Structure of a human carcinogen-converting enzyme, SULT1A1. Structural and kinetic implications of substrate inhibition

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Structure of a human carcinogen-converting enzyme, SULT1A1. Structural and kinetic implications of substrate inhibition is …
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scholarly articleQ13442814

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P356DOI10.1074/JBC.M207246200
P698PubMed publication ID12471039

P50authorJennifer L. MartinQ17517193
P2093author name stringAmanda C Barnett
Catherine F Latham
Nancy E Liyou
Michael E McManus
Ronald G Duggleby
Michael Tresillian
Niranjali U Gamage
P2860cites workA single amino acid, glu146, governs the substrate specificity of a human dopamine sulfotransferase, SULT1A3Q22008545
Expression and characterization of a novel thyroid hormone-sulfating form of cytosolic sulfotransferase from human liverQ24309363
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Functional characterization of two human sulphotransferase cDNAs that encode monoamine- and phenol-sulphating forms of phenol sulphotransferase: substrate kinetics, thermal-stability and inhibitor-sensitivity studiesQ24528266
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Crystal structure of the sulfotransferase domain of human heparan sulfate N-deacetylase/ N-sulfotransferase 1Q27617860
Crystal structure of human catecholamine sulfotransferaseQ27620124
The structural basis of substrate activation in yeast pyruvate decarboxylase. A crystallographic and kinetic studyQ27621116
Crystal structure of SULT2A3, human hydroxysteroid sulfotransferaseQ27624929
Crystal structure of yeast acetohydroxyacid synthase: a target for herbicidal inhibitorsQ27638401
Crystal structures of Toxoplasma gondii HGXPRTase reveal the catalytic role of a long flexible loopQ27733464
Crystal structure of estrogen sulphotransferaseQ27747076
Raster3D: photorealistic molecular graphicsQ27860557
Errors in protein structuresQ27860776
X-ray crystal structure of human dopamine sulfotransferase, SULT1A3. Molecular modeling and quantitative structure-activity relationship analysis demonstrate a molecular basis for sulfotransferase substrate specificityQ28141090
Human cytosolic sulphotransferases: genetics, characteristics, toxicological aspectsQ28215175
Development and validation of a genetic algorithm for flexible dockingQ28236574
Sulfation and sulfotransferases 1: Sulfotransferase molecular biology: cDNAs and genesQ28303680
Characterization of human liver thermostable phenol sulfotransferase (SULT1A1) allozymes with 3,3',5-triiodothyronine as the substrateQ28646411
Formation of the active site of ribulose-1,5-bisphosphate carboxylase/oxygenase by a disorder-order transition from the unactivated to the activated form.Q36625257
Sulfuryl transfer: the catalytic mechanism of human estrogen sulfotransferaseQ41036966
Human phenol sulfotransferases SULT1A2 and SULT1A1: genetic polymorphisms, allozyme properties, and human liver genotype-phenotype correlationsQ42606037
Differential expression of sulfotransferase enzymes involved in thyroid hormone metabolism during human placental developmentQ43819874
Catecholestrogen sulfation: possible role in carcinogenesisQ43924877
Molecular basis of sulfonylurea herbicide inhibition of acetohydroxyacid synthaseQ44258967
Rat brain phenolsulfotransferase—partial purification and some propertiesQ48611904
Sulfotransferase (SULT) 1A1 polymorphism as a predisposition factor for lung cancer: a case-control analysis.Q53392908
Sulfation and sulfotransferases. Introduction: changing view of sulfation and the cytosolic sulfotransferasesQ73075391
Mutational analysis of the substrate binding/catalytic domains of human M form and P form phenol sulfotransferasesQ73731277
Novel sulfotransferases cloned by RT-PCR: real proteins or PCR artifacts?Q74497630
Phenol sulphotransferase SULT1A1*1 genotype is associated with reduced risk of colorectal cancerQ77113474
Analysis of the substrate specificity of human sulfotransferases SULT1A1 and SULT1A3: site-directed mutagenesis and kinetic studiesQ78108827
P433issue9
P407language of work or nameEnglishQ1860
P921main subjectxenobiotic metabolic processQ14358591
Sulfotransferase family 1A member 1Q21122138
P304page(s)7655-62
P577publication date2003-02-28
P1433published inJournal of Biological ChemistryQ867727
P1476titleStructure of a human carcinogen-converting enzyme, SULT1A1. Structural and kinetic implications of substrate inhibition
P478volume278

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cites work (P2860)
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