Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery

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Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery is …
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scholarly articleQ13442814

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P356DOI10.1021/ACS.JMEDCHEM.6B00228
P698PubMed publication ID27031670

P50authorHenriëtte M.G. WillemsQ52116793
Alison J-A WoolfordQ57837773
P2093author name stringJames F Callahan
Gordon Saxty
Rachel McMenamin
Thomas G Davies
Joseph E Coyle
Sharna J Rich
Tom D Heightman
Joseph P Foley
Caroline Richardson
Yolanda Sanchez
John G Yonchuk
Brian J Bolognese
Patricia L Podolin
David Norton
Joshua E Cottom
Hongxing Yan
Jeffrey K Kerns
Charlotte Griffiths-Jones
Gregory Logan
Heidi G Feldser
Jen-Pyng Kou
Keisha Hearn
William E Wixted
P433issue8
P407language of work or nameEnglishQ1860
P921main subjectprotein-protein interactionQ896177
P304page(s)3991-4006
P577publication date2016-04-28
P1433published inJournal of Medicinal ChemistryQ900316
P1476titleMonoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery
P478volume59

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