Discovery of estrogen sulfotransferase inhibitors from a purine library screen

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Discovery of estrogen sulfotransferase inhibitors from a purine library screen is …
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scholarly articleQ13442814

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P356DOI10.1021/JM010171U
P698PubMed publication ID11495578
P5875ResearchGate publication ID11848390

P50authorCarolyn BertozziQ7442
P2093author name stringNegishi M
Chang YT
Schultz PG
Ge X
Leary JA
Gray NS
Cancilla MT
Verdugo DE
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The sulfuryl transfer mechanism. Crystal structure of a vanadate complex of estrogen sulfotransferase and mutational analysisQ27765678
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Synthesis and application of functionally diverse 2,6,9-trisubstituted purine libraries as CDK inhibitorsQ33178547
Carbohydrate sulfotransferases: mediators of extracellular communicationQ34487662
In vitro sulfotransferase activity of NodH, a nodulation protein of Rhizobium meliloti required for host-specific nodulationQ39838962
A novel, high endothelial venule-specific sulfotransferase expresses 6-sulfo sialyl Lewis(x), an L-selectin ligand displayed by CD34.Q41683619
Enzymatic radiolabelling to a high specific activity of legume lipo-oligosaccharidic nodulation factors from Rhizobium melilotiQ41905480
In vitro inhibition of estrogen sulfoconjugation by some 2- and 4-substituted estra-1,3,5(10)-trien-17 beta-ols1aQ42216038
Tyrosine sulfation of the amino terminus of CCR5 facilitates HIV-1 entryQ43694761
Bioactivation of the cooked food mutagen N-hydroxy-2-amino-1-methyl-6- phenylimidazo[4,5-b]pyridine by estrogen sulfotransferase in cultured human mammary epithelial cellsQ61696721
Facile and Clean Oxidation of Alcohols in Water Using Hypervalent Iodine(III) ReagentsQ64029102
Inhibition of human liver steroid sulfotransferase activities by drugs: a novel mechanism of drug toxicity?Q67554535
Quercetin and resveratrol potently reduce estrogen sulfotransferase activity in normal human mammary epithelial cellsQ73169406
Comparison of estrogen concentrations, estrone sulfatase and aromatase activities in normal, and in cancerous, human breast tissuesQ73580683
Picture story. Agony and antagonismQ73853282
Estrone sulfatase versus estrone sulfotransferase in human breast cancer: potential clinical applicationsQ78036291
P433issue17
P407language of work or nameEnglishQ1860
P304page(s)2683-2686
P577publication date2001-08-01
P1433published inJournal of Medicinal ChemistryQ900316
P1476titleDiscovery of estrogen sulfotransferase inhibitors from a purine library screen
P478volume44

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cites work (P2860)
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