Targeting mycobacterium protein tyrosine phosphatase B for antituberculosis agents

scientific article

Targeting mycobacterium protein tyrosine phosphatase B for antituberculosis agents is …
instance of (P31):
scholarly articleQ13442814

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P819ADS bibcode2010PNAS..107.4573Z
P356DOI10.1073/PNAS.0909133107
P932PMC publication ID2842023
P698PubMed publication ID20167798
P5875ResearchGate publication ID41486435

P50authorScott G. FranzblauQ39482766
Jie XuQ91794273
P2093author name stringYong Luo
Yan Liu
Zhong-Yin Zhang
Bo Zhou
Xian Zhang
Rebecca J Chan
Yantao He
Yuehong Wang
Jianyu Zheng
Zhenyun Yang
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A potent and highly selective inhibitor of human alpha-1,3-fucosyltransferase via click chemistryQ33188039
Rapid assembly and in situ screening of bidentate inhibitors of protein tyrosine phosphatasesQ33233529
A two stage click-based library of protein tyrosine phosphatase inhibitorsQ33260614
Parallel synthesis of a multi-substituted benzo[b]furan library.Q33378183
Inhibition of MptpB phosphatase from Mycobacterium tuberculosis impairs mycobacterial survival in macrophagesQ33412046
In vitro and in vivo activities of macrolide derivatives against Mycobacterium tuberculosisQ33722005
Identification of p130Cas as a substrate of Yersinia YopH (Yop51), a bacterial protein tyrosine phosphatase that translocates into mammalian cells and targets focal adhesionsQ33886658
Protein tyrosine phosphatases: structure and function, substrate specificity, and inhibitor developmentQ34110887
Combinatorial control of the specificity of protein tyrosine phosphatasesQ34180660
Protein tyrosine phosphatases: prospects for therapeuticsQ34318066
Interleukin-6 gene-deficient mice show impaired defense against pneumococcal pneumoniaQ34433776
Discovery of protein phosphatase inhibitor classes by biology-oriented synthesisQ34771016
Interplay between mycobacteria and host signalling pathwaysQ35745231
Targeting virulence: a new paradigm for antimicrobial therapyQ36914994
Intracellular bacterial growth is controlled by a kinase network around PKB/AKT1.Q40043123
Interferon-gamma induces C/EBP beta expression and activity through MEK/ERK and p38 in T84 colon epithelial cells.Q40680288
ERK1 and ERK2 activate CCAAAT/enhancer-binding protein-beta-dependent gene transcription in response to interferon-gammaQ40854135
The Salmonella effector SptP dephosphorylates host AAA+ ATPase VCP to promote development of its intracellular replicative nicheQ43074065
Fragment-based substrate activity screening method for the identification of potent inhibitors of the Mycobacterium tuberculosis phosphatase PtpB.Q44448705
Disruption of mptpB impairs the ability of Mycobacterium tuberculosis to survive in guinea pigs.Q44655558
In situ click chemistry: enzyme inhibitors made to their own specificationsQ45093957
Brunsvicamides A−C: Sponge-Related Cyanobacterial Peptides withMycobacteriumtuberculosisProtein Tyrosine Phosphatase Inhibitory ActivityQ57007066
New fronts in an old warQ59097546
Structure-based discovery of small molecule inhibitors targeted to protein tyrosine phosphatase 1BQ73390423
Click chemistry in situ: acetylcholinesterase as a reaction vessel for the selective assembly of a femtomolar inhibitor from an array of building blocksQ78687582
P433issue10
P407language of work or nameEnglishQ1860
P304page(s)4573-4578
P577publication date2010-02-18
P1433published inProceedings of the National Academy of Sciences of the United States of AmericaQ1146531
P1476titleTargeting mycobacterium protein tyrosine phosphatase B for antituberculosis agents
P478volume107

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