A One-Pot Three-Component Double-Click Method for Synthesis of [67Cu]-Labeled Biomolecular Radiotherapeutics

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A One-Pot Three-Component Double-Click Method for Synthesis of [67Cu]-Labeled Biomolecular Radiotherapeutics is …
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scholarly articleQ13442814

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P6179Dimensions Publication ID1085378959
P356DOI10.1038/S41598-017-02123-2
P932PMC publication ID5432496
P698PubMed publication ID28507297

P2093author name stringYoshinori Murakami
Shinya Yano
Takeshi Ito
Katsunori Tanaka
Hiromitsu Haba
Yuki Kumagai
Katsumasa Fujiki
Osamu Kamigaito
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In vivo positron emission tomography (PET) imaging with an alphavbeta6 specific peptide radiolabeled using 18F-"click" chemistry: evaluation and comparison with the corresponding 4-[18F]fluorobenzoyl- and 2-[18F]fluoropropionyl-peptidesQ39941022
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Significant acceleration of 6 pi-azaelectrocyclization resulting from a remarkable substituent effect and formal synthesis of the ocular age pigment A2-E by a new method for substituted pyridine synthesisQ43590070
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MicroPET and autoradiographic imaging of breast cancer alpha v-integrin expression using 18F- and 64Cu-labeled RGD peptideQ44735123
Development of highly stereoselective asymmetric 6pi-azaelectrocyclization of conformationally flexible linear 1-azatrienes. from determination of multifunctional chiral amines, 7-alkyl cis-1-amino-2-indanols, to application as a new synthetic stratQ45063216
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P275copyright licenseCreative Commons Attribution 4.0 InternationalQ20007257
P6216copyright statuscopyrightedQ50423863
P433issue1
P407language of work or nameEnglishQ1860
P304page(s)1912
P577publication date2017-05-15
P1433published inScientific ReportsQ2261792
P1476titleA One-Pot Three-Component Double-Click Method for Synthesis of [67Cu]-Labeled Biomolecular Radiotherapeutics
P478volume7

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cites work (P2860)
Q92431398211At-labeled immunoconjugate via a one-pot three-component double click strategy: practical access to α-emission cancer radiotherapeutics
Q92921658Evaluation of a 68Ga-Labeled DOTA-Tetrazine as a PET Alternative to 111In-SPECT Pretargeted Imaging
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Q92424208Monoclonal antibody-based molecular imaging strategies and theranostic opportunities
Q91083729Multifunctional Clickable Reagents for Rapid Bioorthogonal Astatination and Radio-Crosslinking