Covalent modification as a strategy to block protein-protein interactions with small-molecule drugs

scientific article

Covalent modification as a strategy to block protein-protein interactions with small-molecule drugs is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

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P356DOI10.1016/S1367-5931(99)00049-6
P698PubMed publication ID10679371

P2093author name stringWay JC
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P433issue1
P921main subjectprotein-protein interactionQ896177
P304page(s)40-46
P577publication date2000-02-01
P1433published inCurrent Opinion in Chemical BiologyQ15758415
P1476titleCovalent modification as a strategy to block protein-protein interactions with small-molecule drugs
P478volume4

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cites work (P2860)
Q24649147Beyond picomolar affinities: quantitative aspects of noncovalent and covalent binding of drugs to proteins
Q38011256Drug discovery for a new generation of covalent drugs
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Q46691166Inhibition of the calcineurin-NFAT interaction by small organic molecules reflects binding at an allosteric site
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Q38693434New drug design with covalent modifiers.
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Q29617758Small-molecule inhibitors of protein-protein interactions: progressing towards the dream
Q42245644Structure-based design of alpha-amido aldehyde containing gluten peptide analogues as modulators of HLA-DQ2 and transglutaminase 2.
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