Epidermal growth factor receptor tyrosine kinase inhibitors as anticancer agents

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Epidermal growth factor receptor tyrosine kinase inhibitors as anticancer agents is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

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P6179Dimensions Publication ID1001305932
P356DOI10.2165/00003495-200060001-00003
P698PubMed publication ID11129169

P2093author name stringF Ciardiello
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Anti-epidermal growth factor receptor antibody C225 inhibits angiogenesis in human transitional cell carcinoma growing orthotopically in nude miceQ40971116
Tyrosine kinase inhibitors. 14. Structure-activity relationships for methylamino-substituted derivatives of 4-[(3-bromophenyl)amino]-6-(methylamino)-pyrido[3,4-d]pyrimidine (PD 158780), a potent and specific inhibitor of the tyrosine kinase activityQ41056981
4,5-bis(4-fluoroanilino)phthalimide: A selective inhibitor of the epidermal growth factor receptor signal transduction pathway with potent in vivo antitumor activity.Q41313922
Inhibitors of tyrosine kinaseQ41643303
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In vivo toxicity, pharmacokinetics, and anticancer activity of Genistein linked to recombinant human epidermal growth factor.Q48025147
Antitumor effect and potentiation of cytotoxic drugs activity in human cancer cells by ZD-1839 (Iressa), an epidermal growth factor receptor-selective tyrosine kinase inhibitorQ57424632
Antitumor Activity of Combined Blockade of Epidermal Growth Factor Receptor and Protein Kinase AQ57424743
Cytotoxicity against human tumor cells mediated by the conjugate of anti-epidermal growth factor receptor monoclonal antibody to recombinant ricin A chainQ69739616
Antitumor effect of anti-epidermal growth factor receptor monoclonal antibodies plus cis-diamminedichloroplatinum on well established A431 cell xenograftsQ70487549
Tyrosine kinase inhibitors. 10. Isomeric 4-[(3-bromophenyl)amino]pyrido[d]-pyrimidines are potent ATP binding site inhibitors of the tyrosine kinase function of the epidermal growth factor receptorQ71072552
Tyrphostins. 6. Dimeric benzylidenemalononitrile tyrophostins: potent inhibitors of EGF receptor tyrosine kinase in vitroQ71875718
Epidermal growth factor receptors in human breast carcinoma cells: a potential selective target for transforming growth factor alpha-Pseudomonas exotoxin 40 fusion proteinQ72132785
Antitumor effects of doxorubicin in combination with anti-epidermal growth factor receptor monoclonal antibodiesQ72856071
Epidermal growth factor receptor family and chemosensitizationQ73133036
Epidermal growth factor receptor blockade with C225 plus gemcitabine results in regression of human pancreatic carcinoma growing orthotopically in nude mice by antiangiogenic mechanismsQ73803447
Induction of apoptosis and cell cycle arrest by CP-358,774, an inhibitor of epidermal growth factor receptor tyrosine kinaseQ73838278
Blockade of the epidermal growth factor receptor signaling by a novel tyrosine kinase inhibitor leads to apoptosis of endothelial cells and therapy of human pancreatic carcinomaQ73886918
Genistein exerts multiple suppressive effects on human breast carcinoma cellsQ77536071
PD153035, a tyrosine kinase inhibitor, prevents epidermal growth factor receptor activation and inhibits growth of cancer cells in a receptor number-dependent mannerQ77553678
Biological efficacy of a chimeric antibody to the epidermal growth factor receptor in a human tumor xenograft modelQ77555291
Phase I clinical trial of the flavonoid quercetin: pharmacokinetics and evidence for in vivo tyrosine kinase inhibitionQ77556839
P304page(s)25-32; discussion 41-2
P577publication date2000-01-01
P1433published inDrugsQ3040094
P1476titleEpidermal growth factor receptor tyrosine kinase inhibitors as anticancer agents
P478volume60 Suppl 1

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