Discovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an in vivo active potent VEGFR-2 inhibitor.

scientific article

Discovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an in vivo active potent VEGFR-2 inhibitor. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1021/JM051106D
P698PubMed publication ID16570908

P50authorJ T HuntQ67487747
P2093author name stringAmrita Kamath
Ligang Qian
Punit Marathe
Zhen-Wei Cai
Arvind Mathur
Barri Wautlet
Donna Wei
Joseph Fargnoli
Louis J Lombardo
Robert Jeyaseelan
Robert M Borzilleri
Xiaoping Zheng
Joel C Barrish
Leslie Leith
Rajeev S Bhide
Aberra Fura
Sam Chao
Yong-Zheng Zhang
Celia D'Arienzo
Soong-Hoon Kim
Steven Mortillo
Kenneth Leavitt
Viral Vyas
Daniel Kukral
George Derbin
Laurence I Wu
Stephanie Barbosa
P433issue7
P407language of work or nameEnglishQ1860
P304page(s)2143-2146
P577publication date2006-04-01
P1433published inJournal of Medicinal ChemistryQ900316
P1476titleDiscovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an in vivo active potent VEGFR-2 inhibitor
P478volume49

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