scholarly article | Q13442814 |
P2093 | author name string | Iva Navratilova | |
Andrew L Hopkins | |||
P2860 | cites work | Discovery of a novel warhead against beta-secretase through fragment-based lead generation | Q27648962 |
Tyramine fragment binding to BACE-1 | Q27649725 | ||
Recent developments in fragment-based drug discovery | Q27650535 | ||
Ligand efficiency: a useful metric for lead selection | Q29617403 | ||
Lessons for fragment library design: analysis of output from multiple screening campaigns | Q30864260 | ||
Fragment library screening and lead characterization using SPR biosensors | Q30904689 | ||
Druggability indices for protein targets derived from NMR-based screening data | Q30986175 | ||
SPR-based fragment screening: advantages and applications | Q33304863 | ||
Label-free primary screening and affinity ranking of fragment libraries using parallel analysis of protein panels | Q33319538 | ||
Fragment-based screening using surface plasmon resonance technology | Q33436591 | ||
Recent progress in fragment-based lead discovery | Q33455221 | ||
Predicting protein druggability | Q36352932 | ||
Do enthalpy and entropy distinguish first in class from best in class? | Q36967464 | ||
From fragment to clinical candidate--a historical perspective. | Q37475509 | ||
Stoichiometry and physical chemistry of promiscuous aggregate-based inhibitors | Q42063999 | ||
Comparative analysis of 10 small molecules binding to carbonic anhydrase II by different investigators using Biacore technology. | Q53010783 | ||
Identification of MMP-12 Inhibitors by Using Biosensor-Based Screening of a Fragment Library | Q56945048 | ||
Thermodynamic benchmark study using Biacore technology | Q57266892 | ||
Surface plasmon resonance based assay for the detection and characterization of promiscuous inhibitors | Q80463480 | ||
P4510 | describes a project that uses | surface plasmon resonance | Q898756 |
P433 | issue | 1 | |
P921 | main subject | surface plasmon resonance | Q898756 |
P304 | page(s) | 44-48 | |
P577 | publication date | 2010-02-04 | |
P1433 | published in | ACS Medicinal Chemistry Letters | Q2819061 |
P1476 | title | Fragment screening by surface plasmon resonance | |
P478 | volume | 1 |
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