Fragment screening by surface plasmon resonance

scientific article

Fragment screening by surface plasmon resonance is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1021/ML900002K
P932PMC publication ID4007845
P698PubMed publication ID24900174
P5875ResearchGate publication ID231712197

P2093author name stringIva Navratilova
Andrew L Hopkins
P2860cites workDiscovery of a novel warhead against beta-secretase through fragment-based lead generationQ27648962
Tyramine fragment binding to BACE-1Q27649725
Recent developments in fragment-based drug discoveryQ27650535
Ligand efficiency: a useful metric for lead selectionQ29617403
Lessons for fragment library design: analysis of output from multiple screening campaignsQ30864260
Fragment library screening and lead characterization using SPR biosensorsQ30904689
Druggability indices for protein targets derived from NMR-based screening dataQ30986175
SPR-based fragment screening: advantages and applicationsQ33304863
Label-free primary screening and affinity ranking of fragment libraries using parallel analysis of protein panelsQ33319538
Fragment-based screening using surface plasmon resonance technologyQ33436591
Recent progress in fragment-based lead discoveryQ33455221
Predicting protein druggabilityQ36352932
Do enthalpy and entropy distinguish first in class from best in class?Q36967464
From fragment to clinical candidate--a historical perspective.Q37475509
Stoichiometry and physical chemistry of promiscuous aggregate-based inhibitorsQ42063999
Comparative analysis of 10 small molecules binding to carbonic anhydrase II by different investigators using Biacore technology.Q53010783
Identification of MMP-12 Inhibitors by Using Biosensor-Based Screening of a Fragment LibraryQ56945048
Thermodynamic benchmark study using Biacore technologyQ57266892
Surface plasmon resonance based assay for the detection and characterization of promiscuous inhibitorsQ80463480
P4510describes a project that usessurface plasmon resonanceQ898756
P433issue1
P921main subjectsurface plasmon resonanceQ898756
P304page(s)44-48
P577publication date2010-02-04
P1433published inACS Medicinal Chemistry LettersQ2819061
P1476titleFragment screening by surface plasmon resonance
P478volume1

Reverse relations

cites work (P2860)
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