The fatty acid amide hydrolase inhibitor URB 597: interactions with anandamide in rhesus monkeys

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The fatty acid amide hydrolase inhibitor URB 597: interactions with anandamide in rhesus monkeys is …
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scholarly articleQ13442814

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P356DOI10.1111/J.1476-5381.2011.01388.X
P932PMC publication ID3188916
P698PubMed publication ID21449917
P5875ResearchGate publication ID50935465

P50authorLance R McMahonQ60311068
P2093author name stringJennifer L Stewart
P2860cites workSupersensitivity to anandamide and enhanced endogenous cannabinoid signaling in mice lacking fatty acid amide hydrolaseQ24555807
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Synergy between enzyme inhibitors of fatty acid amide hydrolase and cyclooxygenase in visceral nociceptionQ37162136
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Fatty acid amide hydrolase inhibition heightens anandamide signaling without producing reinforcing effects in primatesQ37239653
Evidence for both inverse agonism at the cannabinoid CB1 receptor and the lack of an endogenous cannabinoid tone in the rat and guinea-pig isolated ileum myenteric plexus-longitudinal muscle preparationQ42434209
Fatty acid amide hydrolase (FAAH) inhibition reduces L-3,4-dihydroxyphenylalanine-induced hyperactivity in the 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine-lesioned non-human primate model of Parkinson's diseaseQ42851005
Delta-9-tetrahydrocannabinol differentially suppresses cisplatin-induced emesis and indices of motor function via cannabinoid CB(1) receptors in the least shrewQ43648938
(R)-methanandamide and Delta 9-THC as discriminative stimuli in rats: tests with the cannabinoid antagonist SR-141716 and the endogenous ligand anandamideQ43703172
Cocaine and other indirect-acting monoamine agonists differentially attenuate a naltrexone discriminative stimulus in morphine-treated rhesus monkeys.Q44625328
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Evaluation of cannabimimetic discriminative stimulus effects of anandamide and methylated fluoroanandamide in rhesus monkeysQ45108581
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Characterization of the fatty acid amide hydrolase inhibitor cyclohexyl carbamic acid 3'-carbamoyl-biphenyl-3-yl ester (URB597): effects on anandamide and oleoylethanolamide deactivation.Q45173372
Monoaminergic drugs and directly observable signs of LAAM withdrawal in rhesus monkeysQ45261514
Dysregulation of the endogenous cannabinoid system in adult rats prenatally treated with the cannabinoid agonist WIN 55,212-2.Q48099000
Large receptor reserve for cannabinoid actions in the central nervous system.Q48299894
The endogenous cannabinoid anandamide produces delta-9-tetrahydrocannabinol-like discriminative and neurochemical effects that are enhanced by inhibition of fatty acid amide hydrolase but not by inhibition of anandamide transportQ48315882
Anandamide administration alone and after inhibition of fatty acid amide hydrolase (FAAH) increases dopamine levels in the nucleus accumbens shell in ratsQ48485540
Isotope dilution GC/MS determination of anandamide and other fatty acylethanolamides in rat blood plasmaQ48513242
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Enhancement of Anandamide Formation in the Limbic Forebrain and Reduction of Endocannabinoid Contents in the Striatum of Δ9-Tetrahydrocannabinol-Tolerant RatsQ60690625
P433issue2b
P407language of work or nameEnglishQ1860
P921main subjectfatty acidQ61476
niacinamideQ192423
anandamideQ410228
cannabinoidsQ422936
P304page(s)655-666
P577publication date2011-09-01
P1433published inBritish Journal of PharmacologyQ919631
P1476titleThe fatty acid amide hydrolase inhibitor URB 597: interactions with anandamide in rhesus monkeys
P478volume164

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cites work (P2860)
Q47744626Cannabinoid CB1 Discrimination: Effects of Endocannabinoids and Catabolic Enzyme Inhibitors
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