| P50 | author | Srinivasan P Venkatachalan | Q63819516 |
| P2093 | author name string | Cynthia Czajkowski | |
| P2860 | cites work | Channel opening by anesthetics and GABA induces similar changes in the GABAA receptor M2 segment | Q24683541 |
| | Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors | Q27631812 |
| | Structure and gating mechanism of the acetylcholine receptor pore | Q27641514 |
| | Crystal structure of the extracellular domain of nAChR alpha1 bound to alpha-bungarotoxin at 1.94 A resolution | Q27646839 |
| | X-ray structure of a prokaryotic pentameric ligand-gated ion channel | Q27650000 |
| | Structure of a potentially open state of a proton-activated pentameric ligand-gated ion channel | Q27652787 |
| | X-ray structure of a pentameric ligand-gated ion channel in an apparently open conformation | Q27652789 |
| | Principles of activation and permeation in an anion-selective Cys-loop receptor | Q27667848 |
| | Structural domains of the human GABAA receptor 3 subunit involved in the actions of pentobarbital | Q73734637 |
| | Dynamics of heteropentameric nicotinic acetylcholine receptor: implications of the gating mechanism | Q80424010 |
| | Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction | Q27860958 |
| | Structures of Aplysia AChBP complexes with nicotinic agonists and antagonists reveal distinctive binding interfaces and conformations | Q28274662 |
| | A single amino acid of the human gamma-aminobutyric acid type A receptor gamma 2 subunit determines benzodiazepine efficacy | Q28304675 |
| | Refined structure of the nicotinic acetylcholine receptor at 4A resolution | Q28306592 |
| | Optimizing the stability of single-chain proteins by linker length and composition mutagenesis | Q32062853 |
| | An epilepsy-related region in the GABA(A) receptor mediates long-distance effects on GABA and benzodiazepine binding sites | Q33574699 |
| | Photochemical proteolysis of an unstructured linker of the GABAAR extracellular domain prevents GABA but not pentobarbital activation | Q34028207 |
| | Linking the Acetylcholine Receptor-Channel Agonist-Binding Sites with the Gate | Q34032739 |
| | Asymmetric structural motions of the homomeric alpha7 nicotinic receptor ligand binding domain revealed by molecular dynamics simulation | Q34183513 |
| | Ligand-induced conformational change in the alpha7 nicotinic receptor ligand binding domain | Q34189724 |
| | GABAA receptor structure-function studies: a reexamination in light of new acetylcholine receptor structures | Q34365717 |
| | Allosteric modulators induce distinct movements at the GABA-binding site interface of the GABA-A receptor | Q34519334 |
| | Benzodiazepine modulation of partial agonist efficacy and spontaneously active GABA(A) receptors supports an allosteric model of modulation | Q35049035 |
| | Mechanism of action of benzodiazepines on GABAA receptors | Q35546302 |
| | A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity | Q36562133 |
| | Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces | Q36907077 |
| | A hydrogen bond in loop A is critical for the binding and function of the 5-HT3 receptor. | Q37112922 |
| | Gamma-aminobutyric acid (GABA) and pentobarbital induce different conformational rearrangements in the GABA A receptor alpha1 and beta2 pre-M1 regions | Q38631543 |
| | Defining affinity with the GABAA receptor. | Q39110587 |
| | Mapping a molecular link between allosteric inhibition and activation of the glycine receptor. | Q39937407 |
| | A stepwise mechanism for acetylcholine receptor channel gating | Q40143954 |
| | A prokaryotic proton-gated ion channel from the nicotinic acetylcholine receptor family | Q40196783 |
| | The role of loop 5 in acetylcholine receptor channel gating. | Q40626492 |
| | Molecular dissection of benzodiazepine binding and allosteric coupling using chimeric gamma-aminobutyric acidA receptor subunits. | Q41060386 |
| | Subunit stoichiometry of a mammalian K+ channel determined by construction of multimeric cDNAs. | Q42604432 |
| | Activation and block of recombinant GABA(A) receptors by pentobarbitone: a single-channel study | Q42626295 |
| | Classic benzodiazepines modulate the open-close equilibrium in alpha1beta2gamma2L gamma-aminobutyric acid type A receptors | Q42651681 |
| | GABA(A) receptor beta 2 Tyr97 and Leu99 line the GABA-binding site. Insights into mechanisms of agonist and antagonist actions | Q42664010 |
| | Different residues in the GABA(A) receptor alpha 1T60-alpha 1K70 region mediate GABA and SR-95531 actions | Q43918728 |
| | The GABAA receptor alpha 1 subunit Pro174-Asp191 segment is involved in GABA binding and channel gating | Q44295686 |
| | Agonist-mediated conformational changes in acetylcholine-binding protein revealed by simulation and intrinsic tryptophan fluorescence | Q45182660 |
| | Agonist- and competitive antagonist-induced movement of loop 5 on the alpha subunit of the neuronal alpha4beta4 nicotinic acetylcholine receptor | Q46875243 |
| | Charged residues in the alpha1 and beta2 pre-M1 regions involved in GABAA receptor activation. | Q46947140 |
| | Complementary regulation of anaesthetic activation of human (alpha6beta3gamma2L) and Drosophila (RDL) GABA receptors by a single amino acid residue | Q48924497 |
| | GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital | Q49124909 |
| | Agonist-, antagonist-, and benzodiazepine-induced structural changes in the alpha1 Met113-Leu132 region of the GABAA receptor. | Q50642710 |
| | Benzodiazepines act on GABAA receptors via two distinct and separable mechanisms. | Q50720910 |
| | A single hydrophobic residue confers barbiturate sensitivity to gamma-aminobutyric acid type C receptor. | Q51472474 |
| | Relationships between inhibition constants and fractional inhibition in enzyme-catalyzed reactions with different numbers of reactants, different reaction mechanisms, and different types and mechanisms of inhibition. | Q52915790 |
| | The major site of photoaffinity labeling of the gamma-aminobutyric acid type A receptor by [3H]flunitrazepam is histidine 102 of the alpha subunit. | Q53725650 |
| | Single channel currents activated by gamma-aminobutyric acid, muscimol, and (-)-pentobarbital in cultured mouse spinal neurons | Q72936590 |
| P433 | issue | 9 | |
| P407 | language of work or name | English | Q1860 |
| P304 | page(s) | 6714-6724 | |
| P577 | publication date | 2012-01-04 | |
| P1433 | published in | Journal of Biological Chemistry | Q867727 |
| P1476 | title | Structural link between γ-aminobutyric acid type A (GABAA) receptor agonist binding site and inner β-sheet governs channel activation and allosteric drug modulation | |
| P478 | volume | 287 | |