Role of 5-HT(1A) receptors in fluoxetine-induced lordosis inhibition

scientific article

Role of 5-HT(1A) receptors in fluoxetine-induced lordosis inhibition is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/J.YHBEH.2010.03.003
P932PMC publication ID3427749
P698PubMed publication ID20223238
P5875ResearchGate publication ID41909577

P2093author name stringCindy Hiegel
Lynda Uphouse
Jhimly Sarkar
Jutatip Guptarak
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A retrospect on the discovery of WAY-100635 and the prospect for improved 5-HT(1A) receptor PET radioligandsQ34016383
5-HT(1A) receptor antagonism reverses and prevents fluoxetine-induced sexual dysfunction in ratsQ34017480
Regulation of 5-HT1A receptor function in brain following agonist or antidepressant administrationQ34174011
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A review and reevaluation of the role of serotonin in the modulation of lordosis behavior in the female ratQ35851456
Neurosteroidogenesis: relevance to neurosteroid actions in brain and modulation by psychotropic drugsQ35974100
Effects of acute fluoxetine on extracellular serotonin levels in the raphe: an in vivo microdialysis studyQ71012065
Female gonadal hormones, serotonin, and sexual receptivityQ73019374
5-HT(1B) receptor-mediated regulation of serotonin clearance in rat hippocampus in vivoQ73081074
The role of 5-HT(1A) and 5-HT(1B/1D) receptors on the modulation of acute fluoxetine-induced changes in extracellular 5-HT: the mechanism of action of (+/-)pindololQ73571947
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A novel approach for predicting antidepressant-induced sexual dysfunction in ratsQ81306017
3alpha-hydroxy-5alpha-pregnan-20-one in the midbrain ventral tegmental area mediates social, sexual, and affective behaviorsQ36329411
Subchronic treatment with fluoxetine attenuates effects of acute fluoxetine on female rat sexual behaviorQ36477275
Strategies for managing antidepressant-induced sexual dysfunction: a reviewQ36649071
Synthesis and function of hypothalamic neuroprogesterone in reproduction.Q36692137
Neuroendocrine regulation of feminine sexual behavior: lessons from rodent models and thoughts about humansQ36901990
Neuroprogesterone: key to estrogen positive feedback?Q36938797
Sexual dysfunction associated with antidepressant therapyQ36993680
Fluoxetine-elicited changes in brain neurosteroid content measured by negative ion mass fragmentographyQ37243720
Solicitation behavior in the estrous female rat: a reviewQ38749487
Pharmacological characterization of selective serotonin reuptake inhibitors (SSRIs).Q40666676
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Changes in sexual function during acute and six-month fluoxetine therapy: a prospective assessmentQ43609177
Effects of selective 5-HT1A receptor antagonists on regional serotonin synthesis in the rat brain: an autoradiographic study with alpha-[14C]methyl-L-tryptophanQ43647927
Extracellular serotonin and 5-hydroxyindoleacetic acid in hypothalamus of the unanesthetized rat measured by in vivo dialysis coupled to high-performance liquid chromatography with electrochemical detection: dialysate serotonin reflects neuronal relQ43661980
Effects on serotonin in rat hypothalamus of D-fenfluramine, aminorex, phentermine and fluoxetineQ44028352
Treatment of cycling female rats with fluoxetine induces desensitization of hypothalamic 5-HT(1A) receptors with no change in 5-HT(2A) receptorsQ44126370
Progesterone attenuates the effect of the 5-HT1A receptor agonist, 8-OH-DPAT, and of mild restraint on lordosis behaviorQ44438197
Fluoxetine may influence lordosis of rats through effects on midbrain 3 alpha,5 alpha-THP concentrationsQ44781888
Estrogen and progesterone dose-dependently reduce disruptive effects of restraint on lordosis behaviorQ44816287
WAY100635 and female rat lordosis behaviorQ44933413
GABAA-5-HT1A receptor interaction in the mediobasal hypothalamusQ45114766
WAY100635 prevents the changes induced by fluoxetine upon the 5-HT1A receptor functionality.Q46352834
Impact of ovarian hormones on the modulation of the serotonin transporter by fluvoxamineQ46716754
Fluoxetine disrupts food intake and estrous cyclicity in Fischer female ratsQ46901407
5-HT1A receptors mediate (+)8-OH-DPAT-stimulation of extracellular signal-regulated kinase (MAP kinase) in vivo in rat hypothalamus: time dependence and regional differences.Q46919563
WAY-100635 inhibits 8-OH-DPAT-stimulated oxytocin, ACTH and corticosterone, but not prolactin secretionQ47887986
Hypothalamic infusion of the 5-HT2/1C agonist, DOI, prevents the inhibitory actions of the 5-HT1A agonist, 8-OH-DPAT, on lordosis behaviorQ48158601
Estrous cycle modulation of extracellular serotonin in mediobasal hypothalamus: role of the serotonin transporter and terminal autoreceptorsQ48159353
Effect of 5,7-dihydroxytryptamine, ovariectomy and gonadal steroids on serotonin receptor binding in rat brainQ48161705
Effect of progesterone on monoamine turnover in the brain of the estrogen-primed rat.Q48222567
5-HT2C receptor involvement in female rat lordosis behaviorQ48228149
Daily injections of fluoxetine induce dose-dependent desensitization of hypothalamic 5-HT1A receptors: reductions in neuroendocrine responses to 8-OH-DPAT and in levels of Gz and Gi proteins.Q48323833
Infusions of 5alpha-pregnan-3alpha-ol-20-one (3alpha,5alpha-THP) to the ventral tegmental area, but not the substantia nigra, enhance exploratory, anti-anxiety, social and sexual behaviours and concomitantly increase 3alpha,5alpha-THP concentrationsQ48382066
Functional integration among 5-hydroxytryptamine receptor families in the control of female rat sexual behaviorQ48389911
Differences in hypothalamic serotonin between estrous phases and gender: an in vivo microdialysis studyQ48456168
Facilitation of female rat lordosis behavior by hypothalamic infusion of 5-HT(2A/2C) receptor agonistsQ48529275
Effect of fluoxetine on serotonin and dopamine concentration in microdialysis fluid from rat striatumQ48589813
5-HT3 receptors in the ventromedial nucleus of the hypothalamus and female sexual behaviorQ48592136
Subchronic administration of fluoxetine impairs estrous behavior in intact female ratsQ48710963
Chronic fluoxetine induces a gradual desensitization of 5-HT1A receptors: reductions in hypothalamic and midbrain Gi and G(o) proteins and in neuroendocrine responses to a 5-HT1A agonist.Q48876980
5-HT1A receptor antagonists and lordosis behaviorQ49022779
In vivo evidence for progesterone dependent decreases in serotonin release in the hypothalamus and midbrain central grey: relation to the induction of lordosisQ49062625
Sexual functioning in chronically depressed patients treated with SSRI antidepressants: a pilot study.Q50919488
WAY-100635 has high selectivity for serotonin 5-HT(1A) versus dopamine D(4) receptors.Q51794751
The forced swimming test as a model for core and component behavioral effects of antidepressant drugs.Q53801502
Estrogen desensitizes 5-HT1A receptors and reduces levels of Gz, Gi1 and Gi3 proteins in the hypothalamusQ62566842
P433issue2
P921main subjectabnormal lordosisQ744305
P304page(s)290-296
P577publication date2010-03-08
P1433published inHormones and BehaviourQ15760887
P1476titleRole of 5-HT(1A) receptors in fluoxetine-induced lordosis inhibition
P478volume58

Reverse relations

cites work (P2860)
Q38991824Animal Models for the Study of Female Sexual Dysfunction
Q90697470Chronic Fluoxetine Impairs the Effects of 5-HT1A and 5-HT2C Receptors Activation in the PAG and Amygdala on Antinociception Induced by Aversive Situation in Mice
Q37515934Comparison of female Fischer and Sprague-Dawley rats in the response to ketanserin
Q43548532Developmental fluoxetine exposure facilitates sexual behavior in female offspring
Q36204980Factors influencing fluoxetine-induced sexual dysfunction in female rats.
Q22242315Flibanserin and 8-OH-DPAT implicate serotonin in association between female marmoset monkey sexual behavior and changes in pair-bond quality.
Q34672013Fluoxetine prevents 8-OH-DPAT-induced hyperphagia in Fischer inbred rats
Q36840540Genetic approaches for understanding the role of serotonin receptors in mood and behavior.
Q37347736Long-term consequences of chronic fluoxetine exposure on the expression of myelination-related genes in the rat hippocampus
Q48111793Paroxetine-induced reduction of sexual incentive motivation in female rats is not modified by 5-HT1B or 5-HT2C antagonists
Q26861672Pharmacology of serotonin and female sexual behavior
Q35731575Sprague-Dawley and Fischer female rats differ in acute effects of fluoxetine on sexual behavior
Q36777115Synthesis of novel analogs of cabergoline: improving cardiovascular safety by removing 5-HT2B receptor agonism

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