Bacterial efflux pump inhibitors from natural sources.

scientific article published on 4 December 2006

Bacterial efflux pump inhibitors from natural sources. is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

External links are
P356DOI10.1093/JAC/DKL460
P698PubMed publication ID17145734
P5875ResearchGate publication ID6652857

P50authorLaura PiddockQ20203247
P2093author name stringSimon Gibbons
Michael Stavri
P2860cites workTetracycline antibiotics: mode of action, applications, molecular biology, and epidemiology of bacterial resistanceQ24548472
Active efflux of tetracycline encoded by four genetically different tetracycline resistance determinants in Escherichia coliQ24613078
Synergy in a medicinal plant: antimicrobial action of berberine potentiated by 5'-methoxyhydnocarpin, a multidrug pump inhibitorQ24650801
Potent synergism of the combination of fluconazole and cyclosporine in Candida albicansQ28344597
Microbial fermentation-derived inhibitors of efflux-pump-mediated drug resistanceQ30667520
Discovery and biological evaluation of a new family of potent modulators of multidrug resistance: reversal of multidrug resistance of mouse lymphoma cells by new natural jatrophane diterpenoids isolated from Euphorbia speciesQ30695267
Flavonolignan and flavone inhibitors of a Staphylococcus aureus multidrug resistance pump: structure-activity relationshipsQ31917006
The threat of vancomycin resistanceQ33646840
Aminoglycoside-modifying enzymesQ33745231
Vancomycin-resistant enterococciQ33975592
Mechanisms of action and resistance of older and newer fluoroquinolonesQ34030757
Version 2000: the new beta-lactamases of Gram-negative bacteria at the dawn of the new millenniumQ34047473
The emergence and evolution of methicillin-resistant Staphylococcus aureusQ34094813
Multidrug pump inhibitors uncover remarkable activity of plant antimicrobials.Q34143579
Piperine, a phytochemical potentiator of ciprofloxacin against Staphylococcus aureusQ34352260
Antimalarial activity of Artemisia annua flavonoids from whole plants and cell culturesQ34384045
Mechanisms of bacterial biocide and antibiotic resistanceQ34631438
Clinically relevant chromosomally encoded multidrug resistance efflux pumps in bacteriaQ34647294
Inducible NorA-mediated multidrug resistance in Staphylococcus aureusQ35120701
Efflux-mediated fluoroquinolone resistance in Staphylococcus aureusQ35814875
Update on acquired tetracycline resistance genesQ36101214
Efflux-mediated antimicrobial resistanceQ36138147
Role of mycobacterial efflux transporters in drug resistance: an unresolved questionQ36378353
The functions and structure of ABC transporters: implications for the design of new inhibitors of Pgp and MRP1 to control multidrug resistance (MDR).Q36536579
Multidrug-resistance efflux pumps - not just for resistanceQ36538111
Emergence of quinolone resistance among clinical isolates of methicillin-resistant Staphylococcus aureus in Ontario, CanadaQ36754974
Staphylococcus aureus with reduced susceptibility to vancomycin isolated from a patient with fatal bacteremiaQ37064359
Bacterial resistance to macrolide, lincosamide, and streptogramin antibiotics by target modificationQ37416736
Efflux-mediated multidrug resistance in Bacillus subtilis: similarities and dissimilarities with the mammalian systemQ37522093
Metabolites of the "smoke tree", Dalea spinosa, potentiate antibiotic activity against multidrug-resistant Staphylococcus aureusQ38901490
Phenothiazines alter resistance of methicillin-resistant strains of Staphylococcus aureus (MRSA) to oxacillin in vitroQ39148696
Evidence for the existence of a multidrug efflux transporter distinct from NorA in Staphylococcus aureusQ39473922
Identification and characterization of inhibitors of multidrug resistance efflux pumps in Pseudomonas aeruginosa: novel agents for combination therapyQ39475894
Use of an efflux-deficient streptococcus pneumoniae strain panel to identify ABC-class multidrug transporters involved in intrinsic resistance to antimicrobial agentsQ39610470
Accumulation of 10 fluoroquinolones by wild-type or efflux mutant Streptococcus pneumoniae.Q39653038
The baeSR two-component regulatory system activates transcription of the yegMNOB (mdtABCD) transporter gene cluster in Escherichia coli and increases its resistance to novobiocin and deoxycholateQ39679827
Contributions of MexAB-OprM and an EmrE homolog to intrinsic resistance of Pseudomonas aeruginosa to aminoglycosides and dyesQ39730828
Phenothiazines and thioxanthenes inhibit multidrug efflux pump activity in Staphylococcus aureusQ39740497
Mutations affecting substrate specificity of the Bacillus subtilis multidrug transporter Bmr.Q39845092
Fluoroquinolone resistance protein NorA of Staphylococcus aureus is a multidrug efflux transporterQ39864846
Jatrophane diterpenes as modulators of multidrug resistance. Advances of structure-activity relationships and discovery of the potent lead pepluanin A.Q40592854
Prevention of drug access to bacterial targets: permeability barriers and active effluxQ40737334
Epigallocatechin-gallate enhances the activity of tetracycline in staphylococci by inhibiting its efflux from bacterial cellsQ40882710
Berberis aetnensis C. Presl. extracts: antimicrobial properties and interaction with ciprofloxacinQ42035117
Global transcriptome analysis of the responses of a fluoroquinolone-resistant Streptococcus pneumoniae mutant and its parent to ciprofloxacinQ43181777
Linezolid resistance in a clinical isolate of Staphylococcus aureusQ43690311
The multidrug efflux pump NorA is not required for salicylate-induced reduction in drug accumulation by Staphylococcus aureusQ44183691
Identification and characterization of a novel efflux-related multidrug resistance phenotype in Staphylococcus aureusQ44235729
Bacterial resistance modifying agents from Lycopus europaeusQ44244613
A novel inhibitor of multidrug efflux pumps in Staphylococcus aureusQ44257253
Two flavonols from Artemisa annua which potentiate the activity of berberine and norfloxacin against a resistant strain of Staphylococcus aureusQ44257849
Polyacylated neohesperidosides from Geranium caespitosum: bacterial multidrug resistance pump inhibitorsQ44442921
Isoflavones as potentiators of antibacterial activityQ44571372
Phenylpiperidine selective serotonin reuptake inhibitors interfere with multidrug efflux pump activity in Staphylococcus aureusQ44588035
Phenolic metabolites of Dalea versicolor that enhance antibiotic activity against model pathogenic bacteriaQ44813822
In Pseudomonas aeruginosa ethidium bromide does not induce its own degradation or the assembly of pumps involved in its effluxQ45107516
Identification and biological evaluation of grapefruit oil components as potential novel efflux pump modulators in methicillin-resistant Staphylococcus aureus bacterial strainsQ45124008
Antibacterial and resistance modifying activity of Rosmarinus officinalisQ45160744
Catechin gallates inhibit multidrug resistance (MDR) in Staphylococcus aureusQ45219347
Remarkable synergies between baicalein and tetracycline, and baicalein and beta-lactams against methicillin-resistant Staphylococcus aureusQ46446180
Multidrug resistance reversal agent from Jatropha ellipticaQ46624130
Isopimaric acid from Pinus nigra shows activity against multidrug-resistant and EMRSA strains of Staphylococcus aureusQ46662052
Synergic interaction between pomegranate extract and antibiotics against Staphylococcus aureus.Q46713748
Synthesis of functionalized 2-aryl-5-nitro-1H-indoles and their activity as bacterial NorA efflux pump inhibitorsQ46734710
Antimicrobial, resistance-modifying effects, antioxidant and free radical scavenging activities of Mezoneuron benthamianum Baill., Securinega virosa Roxb. &Wlld. and Microglossa pyrifolia Lam.Q46883325
A new chloramphenicol and florfenicol resistance gene flanked by two integron structures in Salmonella typhimurium DT104.Q47961406
Inhibitors of multidrug resistance (MDR) have affinity for MDR substratesQ47972803
Staphylococcus aureus MDR efflux pump inhibitors from a Berberis and a Mahonia (sensu strictu) species.Q54004587
Activity of the tea component epicatechin gallate and analogues against methicillin-resistant Staphylococcus aureus.Q54031266
The effect of a component of tea (Camellia sinensis) on methicillin resistance, PBP2' synthesis, and beta-lactamase production in Staphylococcus aureus.Q54125094
Rapid development of ciprofloxacin resistance in methicillin-susceptible and -resistant Staphylococcus aureus.Q54294777
In-vitro sensitivity of amoxicillin/clavulanic acid (Augmentin) to isolated beta-lactamases and in-vitro antibacterial activity.Q54322163
P433issue6
P407language of work or nameEnglishQ1860
P1104number of pages14
P304page(s)1247-1260
P577publication date2006-12-04
P1433published inJournal of Antimicrobial ChemotherapyQ6294770
P1476titleBacterial efflux pump inhibitors from natural sources
P478volume59

Reverse relations

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