Studies of the biogenic amine transporters. 12. Identification of novel partial inhibitors of amphetamine-induced dopamine release.

scientific article published on 25 April 2008

Studies of the biogenic amine transporters. 12. Identification of novel partial inhibitors of amphetamine-induced dopamine release. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1124/JPET.108.139675
P932PMC publication ID2562894
P698PubMed publication ID18441249
P5875ResearchGate publication ID5411640

P50authorJoseph J PariserQ41650337
P2093author name stringRichard B Rothman
John S Partilla
Subramaniam Ananthan
Christina M Dersch
P2860cites workStudies of the biogenic amine transporters. VII. Characterization of a novel cocaine binding site identified with [125I]RTI-55 in membranes prepared from human, monkey and guinea pig caudateQ48501061
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Inhibition and dissociation of [3H]-paroxetine binding to human plateletsQ69320679
Amphetamine-type central nervous system stimulants release norepinephrine more potently than they release dopamine and serotoninQ28143430
Therapeutic potential of monoamine transporter substratesQ28266724
SSRIs and SNRIs: broad spectrum of efficacy beyond major depressionQ33543679
Anxiety disorders: a review of tricyclic antidepressants and selective serotonin reuptake inhibitors.Q34053653
In vitro characterization of ephedrine-related stereoisomers at biogenic amine transporters and the receptorome reveals selective actions as norepinephrine transporter substratesQ34227794
Distinct effects of imipramine on 5-hydroxytryptamine uptake mediated by the recombinant rat serotonin transporter SERT1.Q34469567
G protein-coupled receptor allosterism and complexingQ34523552
Allosteric enhancers, allosteric agonists and ago-allosteric modulators: where do they bind and how do they act?Q34581080
Binding surface analysis: an intuitive yet quantitative method for the design and analysis of ligand binding studiesQ39501827
Studies of the biogenic amine transporters. XI. Identification of a 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR12909) analog that allosterically modulates the serotonin transporterQ40429339
Characterization of an allosteric citalopram-binding site at the serotonin transporter.Q40479596
From synapse to vesicle: the reuptake and storage of biogenic amine neurotransmittersQ40713073
Nongenomic steroidal modulation of high-affinity serotonin transportQ40967286
Studies of the biogenic amine transporters. VIII: identification of a novel partial inhibitor of dopamine uptake and dopamine transporter bindingQ42164303
3H cocaine labels a binding site associated with the serotonin transporter in guinea pig brain: allosteric modulation by paroxetineQ43710268
Salvinorin A: allosteric interactions at the mu-opioid receptorQ44332543
Identification and characterization of a novel allosteric modulator (SoRI-6238) of the serotonin transporterQ44965402
P433issue1
P407language of work or nameEnglishQ1860
P304page(s)286-295
P577publication date2008-04-25
P1433published inJournal of Pharmacology and Experimental TherapeuticsQ1500272
P1476titleStudies of the biogenic amine transporters. 12. Identification of novel partial inhibitors of amphetamine-induced dopamine release
P478volume326

Reverse relations

cites work (P2860)
Q33808035Allosteric modulatory effects of SRI-20041 and SRI-30827 on cocaine and HIV-1 Tat protein binding to human dopamine transporter.
Q36248541Binding of the amphetamine-like 1-phenyl-piperazine to monoamine transporters
Q38098582Examining the complex regulation and drug-induced plasticity of dopamine release and uptake using voltammetry in brain slices
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Q37672037HIV-1 transgenic rats display an increase in [(3)H]dopamine uptake in the prefrontal cortex and striatum.
Q64054571Mutational effects of human dopamine transporter at tyrosine88, lysine92, and histidine547 on basal and HIV-1 Tat-inhibited dopamine transport
Q26853319Nonclassical pharmacology of the dopamine transporter: atypical inhibitors, allosteric modulators, and partial substrates
Q36912735Recombinant human immunodeficiency virus-1 transactivator of transcription1-86 allosterically modulates dopamine transporter activity.
Q34467830Studies of the biogenic amine transporters 15. Identification of novel allosteric dopamine transporter ligands with nanomolar potency
Q24655326Studies of the biogenic amine transporters. 13. Identification of "agonist" and "antagonist" allosteric modulators of amphetamine-induced dopamine release
Q34249270Studies of the biogenic amine transporters. 14. Identification of low-efficacy "partial" substrates for the biogenic amine transporters
Q41922188The role of human dopamine transporter in NeuroAIDS.

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