2-Carbaborane-3-phenyl-1H-indoles--synthesis via McMurry reaction and cyclooxygenase (COX) inhibition activity.

scientific article published on 09 January 2013

2-Carbaborane-3-phenyl-1H-indoles--synthesis via McMurry reaction and cyclooxygenase (COX) inhibition activity. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1002/CMDC.201200455
P932PMC publication ID3849512
P698PubMed publication ID23303738
P5875ResearchGate publication ID234099397

P50authorWilma NeumannQ59565575
Matthias ScholzQ83444557
Markus LaubeQ84072955
Lawrence J. MarnettQ86531334
Torsten KniessQ88109481
Evamarie Hey-HawkinsQ21259593
Jens PietzschQ39503167
P2093author name stringPeter Lönnecke
Brenda Crews
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Radiosynthesis of a ¹⁸F-labeled 2,3-diarylsubstituted indole via McMurry coupling for functional characterization of cyclooxygenase-2 (COX-2) in vitro and in vivo.Q39353397
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[I]-Celecoxib Analogues as SPECT Tracers of Cyclooxygenase-2 in InflammationQ42189926
Synthesis and biological evaluation of substituted 2-sulfonyl-phenyl-3-phenyl-indoles: a new series of selective COX-2 inhibitorsQ44356861
Discovery of 2-phenyl-3-sulfonylphenyl-indole derivatives as a new class of selective COX-2 inhibitorsQ44671764
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Exploration of physicochemical properties and molecular modelling studies of 2-sulfonyl-phenyl-3-phenyl-indole analogs as cyclooxygenase-2 inhibitors.Q51907410
P433issue2
P304page(s)329-335
P577publication date2013-01-09
P1433published inChemMedChemQ2962252
P1476title2-Carbaborane-3-phenyl-1H-indoles--synthesis via McMurry reaction and cyclooxygenase (COX) inhibition activity
P478volume8

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cites work (P2860)
Q107552783Carbaboranes – more than just phenyl mimetics
Q90850871Carboranyl Analogues of Celecoxib with Potent Cytostatic Activity against Human Melanoma and Colon Cancer Cell Lines
Q92945552Carboranyl Analogues of Ketoprofen with Cytostatic Activity against Human Melanoma and Colon Cancer Cell Lines
Q90372572Carboranyl Derivatives of Rofecoxib with Cytostatic Activity against Human Melanoma and Colon Cancer Cells
Q26750933Development of Antioxidant COX-2 Inhibitors as Radioprotective Agents for Radiation Therapy-A Hypothesis-Driven Review
Q107552670Half- and mixed-sandwich metallacarboranes for potential applications in medicine
Q38808788Recent developments with boron as a platform for novel drug design
Q36987287nido-Dicarbaborate Induces Potent and Selective Inhibition of Cyclooxygenase-2

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