Dynamic behavior of the active and inactive states of the adenosine A(2A) receptor.

scientific article published on 17 March 2014

Dynamic behavior of the active and inactive states of the adenosine A(2A) receptor. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1021/JP411618H
P932PMC publication ID3983344
P698PubMed publication ID24579769
P5875ResearchGate publication ID260440695

P50authorChristopher G. TateQ41625610
Supriyo BhattacharyaQ80146142
Nagarajan VaidehiQ87724234
P2093author name stringReinhard Grisshammer
Sangbae Lee
P2860cites workStructure of an agonist-bound human A2A adenosine receptorQ24296388
Agonist-bound adenosine A2A receptor structures reveal common features of GPCR activationQ24303747
Crystal structure of the β2 adrenergic receptor-Gs protein complexQ24635327
The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonistQ24654563
High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptorQ24657484
Structure of the Adenosine A2A Receptor in Complex with ZM241385 and the Xanthines XAC and CaffeineQ27672832
VMD: visual molecular dynamicsQ27860554
GROMACS 4:  Algorithms for Highly Efficient, Load-Balanced, and Scalable Molecular SimulationQ27860944
Seven-transmembrane receptorsQ29619896
The occurrence of C-H...O hydrogen bonds in proteinsQ30417905
Implementation of force distribution analysis for molecular dynamics simulationsQ33875825
The Calpha ---H...O hydrogen bond: a determinant of stability and specificity in transmembrane helix interactionsQ33929647
Thermostabilisation of an agonist-bound conformation of the human adenosine A(2A) receptorQ34179174
Molecular signatures of G-protein-coupled receptorsQ34327700
Polar residues drive association of polyleucine transmembrane helicesQ34449670
Limits of ligand selectivity from docking to models: in silico screening for A(1) adenosine receptor antagonistsQ34490693
Polar side chains drive the association of model transmembrane peptidesQ34630825
International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and classification of adenosine receptors--an updateQ34701303
Dimerization of the class A G protein-coupled neurotensin receptor NTS1 alters G protein interactionQ35879672
Role of detergents in conformational exchange of a G protein-coupled receptorQ36332894
Hydrogen-bonding and packing features of membrane proteins: functional implicationsQ36481425
Co-evolving stability and conformational homogeneity of the human adenosine A2a receptorQ36825295
Conformational complexity of G-protein-coupled receptorsQ36880905
Thermostabilization of the β1-adrenergic receptor correlates with increased entropy of the inactive stateQ37032791
Specificity of native-like interhelical hydrophobic contacts in the apomyoglobin intermediate.Q37168151
Structure and activation of the visual pigment rhodopsinQ37700655
Adenosine receptors: what we know and what we are learningQ37724988
The crystallographic structure of the human adenosine A2A receptor in a high-affinity antagonist-bound state: implications for GPCR drug screening and designQ37764224
The role of conformational ensembles of seven transmembrane receptors in functional selectivityQ37798993
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Free energy via molecular simulation: applications to chemical and biomolecular systemsQ38648060
GPCR stabilization using the bicelle-like architecture of mixed sterol-detergent micellesQ40616754
A role for a specific cholesterol interaction in stabilizing the Apo configuration of the human A(2A) adenosine receptorQ42949696
Crystallographic evidence for C alpha-H...O=C hydrogen bonds in a collagen triple helixQ47628348
C-H...O hydrogen bonds in beta-sheetsQ47982629
Packing interactions in the apomyglobin folding intermediateQ71031209
Interhelical hydrogen bonding drives strong interactions in membrane proteinsQ73402358
Asparagine-mediated self-association of a model transmembrane helixQ73402361
P433issue12
P407language of work or nameEnglishQ1860
P304page(s)3355-3365
P577publication date2014-03-17
P1433published inJournal of Physical Chemistry BQ668669
P1476titleDynamic behavior of the active and inactive states of the adenosine A(2A) receptor
P478volume118

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cites work (P2860)
Q37490747Conserved Mechanism of Conformational Stability and Dynamics in G-Protein-Coupled Receptors
Q64277579Dynamic Role of the G Protein in Stabilizing the Active State of the Adenosine A Receptor
Q36421791How Can Mutations Thermostabilize G-Protein-Coupled Receptors?
Q30831488How Do Short Chain Nonionic Detergents Destabilize G-Protein-Coupled Receptors?
Q38259766Novel approaches for targeting the adenosine A2A receptor
Q92594361Prediction of Conformation Specific Thermostabilizing Mutations for Class A G Protein-Coupled Receptors
Q34503044Rapid Computational Prediction of Thermostabilizing Mutations for G Protein-Coupled Receptors.
Q38843185Safety issues of compounds acting on adenosinergic signalling
Q28543560Structural and energetic effects of A2A adenosine receptor mutations on agonist and antagonist binding
Q36044571Structural dynamics and thermostabilization of neurotensin receptor 1
Q57922209Validating a 14-Drug Microtiter Plate Containing Bedaquiline and Delamanid for Large-Scale Research Susceptibility Testing of Mycobacterium tuberculosis

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