The role of fulvestrant in endometrial cancer

scientific article

The role of fulvestrant in endometrial cancer is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

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P356DOI10.1080/17425255.2016.1244264
P698PubMed publication ID27696906

P50authorChiara CassaniQ85328415
Simone FerreroQ47282621
Arsenio SpinilloQ59159199
P2093author name stringPier Luigi Venturini
Anna Daniela Iacobone
Barbara Gardella
Mattia Dominoni
Stefano Bogliolo
Anna Orlandini
Franco Viazzo
P2860cites workHormonal therapy in advanced or recurrent endometrial cancerQ24235543
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Palbociclib in Hormone-Receptor-Positive Advanced Breast CancerQ33423263
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Effects of short-term antiestrogen treatment of primary breast cancer on estrogen receptor mRNA and protein expression and on estrogen-regulated genesQ59289308
Importance of the regulation of nuclear receptor degradationQ34327269
Fulvestrant: a review of its use in the management of hormone receptor-positive metastatic breast cancer in postmenopausal womenQ34626963
The turnover of estrogen receptor α by the selective estrogen receptor degrader (SERD) fulvestrant is a saturable process that is not required for antagonist efficacyQ35027844
Phase II study of everolimus and letrozole in patients with recurrent endometrial carcinomaQ35144264
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Combined histone deacetylase inhibition and tamoxifen induces apoptosis in tamoxifen-resistant breast cancer models, by reversing Bcl-2 overexpressionQ35201384
Estrogen receptor alpha is a putative substrate for the BRCA1 ubiquitin ligaseQ35749504
Fulvestrant: an oestrogen receptor antagonist with a novel mechanism of actionQ35750078
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ERα phosphorylation at Y537 by Src triggers E6-AP-ERα binding, ERα ubiquitylation, promoter occupancy, and target gene expression.Q36210983
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A phase I trial to assess the pharmacology of the new oestrogen receptor antagonist fulvestrant on the endometrium in healthy postmenopausal volunteersQ36646485
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OTU Domain-containing ubiquitin aldehyde-binding protein 1 (OTUB1) deubiquitinates estrogen receptor (ER) alpha and affects ERalpha transcriptional activityQ37269111
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The effects of estradiol and selective estrogen receptor modulators on gene expression and messenger RNA stability in immortalized sheep endometrial stromal cells and human endometrial adenocarcinoma cellsQ40649825
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The paracrine stimulation of MCF-7 cells by MDA-MB-231 cells: possible role in antiestrogen failureQ41959489
FDA drug approval summaries: fulvestrantQ42691178
Results of the CONFIRM phase III trial comparing fulvestrant 250 mg with fulvestrant 500 mg in postmenopausal women with estrogen receptor-positive advanced breast cancer.Q42882393
Phase II study of fulvestrant 250 mg/month in patients with recurrent or metastatic endometrial cancer: a study of the Arbeitsgemeinschaft Gynäkologische OnkologieQ44208606
The NEDD8 pathway is required for proteasome-mediated degradation of human estrogen receptor (ER)-alpha and essential for the antiproliferative activity of ICI 182,780 in ERalpha-positive breast cancer cellsQ44294730
Pharmacokinetic profile of intramuscular fulvestrant in advanced breast cancerQ44915900
Fulvestrant (ICI 182,780)-dependent interacting proteins mediate immobilization and degradation of estrogen receptor-alphaQ46928900
Treating gynecologic malignancies with selective estrogen receptor downregulators (SERDs): promise and challenges.Q55049851
Endometrial cancer: ESMO Clinical Practice Guidelines for diagnosis, treatment and follow-upQ56019470
P433issue5
P407language of work or nameEnglishQ1860
P304page(s)537-544
P577publication date2016-10-04
P1433published inExpert Opinion on Drug Metabolism & ToxicologyQ5421205
P1476titleThe role of fulvestrant in endometrial cancer
P478volume13