Identification of novel, selective, and stable inhibitors of class II histone deacetylases. Validation studies of the inhibition of the enzymatic activity of HDAC4 by small molecules as a novel approach for cancer therapy

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Identification of novel, selective, and stable inhibitors of class II histone deacetylases. Validation studies of the inhibition of the enzymatic activity of HDAC4 by small molecules as a novel approach for cancer therapy is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1021/JM900555U
P8608Fatcat IDrelease_5qkwwi7oe5e6dnkvx62cnmzzve
P698PubMed publication ID19888759
P5875ResearchGate publication ID38066520

P50authorCarsten Schultz-FademrechtQ59564783
P2093author name stringPhilip Jones
Christian Steinkühler
Michael Rowley
Ralph Laufer
Sergio Altamura
Ester Muraglia
Federica Ferrigno
Jesus M Ontoria
Maria Cecilia Palumbi
Rita Scarpelli
Annalise Di Marco
Sergio Serafini
P433issue21
P407language of work or nameEnglishQ1860
P304page(s)6782-6789
P577publication date2009-11-01
P1433published inJournal of Medicinal ChemistryQ900316
P1476titleIdentification of novel, selective, and stable inhibitors of class II histone deacetylases. Validation studies of the inhibition of the enzymatic activity of HDAC4 by small molecules as a novel approach for cancer therapy
P478volume52

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Q38246144Selective class IIa HDAC inhibitors: myth or reality
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Q36614119Why Hydroxamates May Not Be the Best Histone Deacetylase Inhibitors--What Some May Have Forgotten or Would Rather Forget?

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