Interaction of sulfonylurea with the pancreatic B-cell

scientific article published on October 1984

Interaction of sulfonylurea with the pancreatic B-cell is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

External links are
P356DOI10.1007/BF01971460
P698PubMed publication ID6436052

P50authorErik GylfeQ43049285
P2093author name stringJ Sehlin
B Hellman
B Täljedal
P2860cites workOn the Possible Role of Thiol Groups in the Insulin-Releasing Action of Mercurials, Organic Disulfides, Alkylating Agents, and SulfonylureasQ28320917
Inhibition of glucose-induced release of insulin by aldose reductase inhibitorsQ34708157
Effect of glibenclamide on the osmotic resistance of pancreatic beta-cellsQ36605047
The mechanism of sulfonylurea stimulation of insulin release.Q38355789
Potentiating effects of drugs on the binding of glibenclamide to pancreatic beta cellsQ38361033
Effects of various modifiers of insulin release on the lanthanum-nondisplaceable45ca2+ uptake by isolated pancreatic isletsQ40049071
Insulin secretion in diabetes mellitusQ40302183
On insulin secretionQ40313938
Effect of glucose on K+handling by pancreatic isletsQ40828194
D-Glucose inhibits potassium efflux from pancreatic islet cellsQ40850833
Uptake of tolbutamide by islets of Langerhans and other tissuesQ40991688
Stimulus-secretion coupling of glucose-induced insulin release. XXIX. Regulation of 86Rb+ efflux from perfused isletsQ41002036
Transport of rubidium and sodium in pancreatic isletsQ41514972
Insulinotropic effects of hypoglycaemic and hyperglycaemic sulphonamides: The ionophoretic hypothesisQ41549286
L-leucine and a nonmetabolized analogue activate pancreatic islet glutamate dehydrogenaseQ41614642
Chronic chlorpropamide therapy of noninsulin-dependent diabetes augments basal and stimulated insulin secretion by increasing islet sensitivity to glucoseQ41618502
The pentose cycle and insulin release in mouse pancreatic isletsQ41838893
Interrelationship of islet metabolism, adenosine triphosphate content and insulin releaseQ42105569
Synergistic effects of hypoglycaemic sulphonylureas and antibiotic ionophores upon calcium translocationQ42633250
Effects of glucose and other modifiers of insulin release on the oxidative metabolism of amino acids in micro-dissected pancreatic isletsQ42922523
Glucose metabolism in mouse pancreatic isletsQ42925548
The kinetics of electrical activity of beta cells in response to a "square wave" stimulation with glucose or glibenclamideQ43433034
The pancreatic beta-cell recognition of insulin secretagogues. Inhibitory effects of a membrane probe on the islet uptake and insulin-releasing action of glibenclamideQ43527081
Is there a common beta cell insulin compartment stimulated by glucose and tolbutamide?Q43600937
The biophysical effects of insulin-releasing agents on islet cellsQ44091608
Ionic effects on the uptake of sulfonylurea (glibenclamide) by pancreatic isletsQ44762937
The pancreatic β-cell recognition of insulin secretagogues. II. Site of action of tolbutamideQ47736543
Specific receptors for sulfonylureas in brain and in a B-cell tumor of the ratQ48966318
Role of cyclic AMP in insulin release evoked by glucose and other secretagogues.Q52231354
Ionophoretic activity of hypoglycemic sulfonylureasQ53734336
Role of glucose as a regulator and precursor of amino acids in the pancreatic beta-cells.Q53848688
The pancreatic -cell recognition of insulin secretagogues. IV. Islet uptake of sulfonylureas.Q54105575
Requirement for calcium ion in insulin secretion by the perfused rat pancreas.Q54282379
Adenosine Triphosphate Levels of Mammalian Pancreatic B Cells after Stimulation with Glucose and Hypoglycemic SulfonylureasQ54361249
Glucose-induced decrease in Rb+ permeability in pancreatic β cellsQ59084984
Depolarization-independent net uptake of calcium into clonal insulin-releasing cells exposed to glucoseQ60032740
Uptake of glibornuride by microdissected pancreatic isletsQ67296577
Comparison of the effects of leucines, non-metabolizable leucine analogues and other insulin secretagogues on the activity of glutamate dehydrogenaseQ67855971
Factors affecting the uptake of glibenclamide in microdissected pancreatic islets rich in beta-cellsQ68342154
The Stimulus-Secretion Coupling of Glucose-Induced Insulin Release VIII. Combined Effects of Glucose and SulfonylureasQ69175744
The stimulus-secretion coupling of glucose-induced insulin release XII. Effects of diazoxide and gliclazide upon45calcium efflux from perifused isletsQ69258165
Acid Amyloglucosidase and Carbohydrate Regulation - III. The Induction of Sulphonylurea-Stimulated Insulin Release and its Dependence on Intracellular MonoaminesQ69380224
Properties of ionophores with broad range cation selectivityQ69580559
Electrical activity in pancreatic islet cellsQ69845749
Action of some hypoglycaemic sulphonylureas on the oxygen consumption of isolated pancreatic islets of miceQ69894220
Energy Metabolism in Pancreatic Islets of Rats: Studies with Tolbutamide and HypoxiaQ69946345
Tolbutamide stimulation of 45Ca fluxes in microdissected pancreatic islets rich in beta-cellsQ70183865
Opposite effects of tolbutamide and diazoxide on 86Rb+ fluxes and membrane potential in pancreatic B cellsQ70245055
Receptor binding sites of hypoglycemic sulfonylureas and related [(acylamino)alkyl]benzoic acidsQ70309196
Transport of Pr3+ by hypoglycemic sulfonylureas across liposomal membranesQ70428165
Effect of a hypoglycaemic sulphonylurea (HB419) and a non-metabolizable amino acid (BCH) on the insulin release and endogenous substrate metabolism of rat pancreatic isletsQ70436043
Binding of hypoglycaemic sulphonylureas to an artificial phospholipid bilayerQ70470826
Lack of Ca2+ ionophoretic activity of hypoglycemic sulfonylureas in excitable cells and isolated secretory granulesQ70548666
Calcium transport in liposomes containing hypoglycemic and hyperglyemic sulfonamidesQ71428372
Modalities of gliclazide-induced Ca2+ influx into the pancreatic B-cellQ71462687
Opposite effects of hypoglycemic and hyperglycemic sulfonamides upon ionophore-mediated calcium transportQ71511027
Changes in glucose-stimulated insulin secretion after long-term treatment of C57BL mice with glibenclamideQ71528481
Long-term effects of glibenclamide on the insulin production, oxidative metabolism and quantitative ultrastructure of mouse pancreatic islets maintained in tissue culture at different glucose concentrationsQ71540171
Are Cl- mechanisms in mouse pancreatic islets involved in insulin release?Q71583942
Differences between the effect of tolbutamide and Ca2+-ionophores on Ca2+ efflux from pancreatic beta-cellsQ71631023
Tolbutamide stimulation and inhibition of insulin release: studies of the underlying ionic mechanisms in isolated rat isletsQ72129897
Metabolic, cationic and secretory effects of hypoglycemic sulfonylureas in pancreatic isletsQ72145797
Carbutamide stimulation of glutamic dehydrogenase activity in the pancreatic β cells from obese-hyperglycemic miceQ72314196
Effect of hypoglycemic sulfonylureas on Ca2+ fluxes across lipid bilayersQ72732454
Glibenclamide is exceptional among hypoglycaemic sulphonylureas in accumulating progressively in β-cell-rich pancreatic isletsQ72809187
Levels of α-Ketoglutarate and Glutamate in Stimulated Pancreatic β-CellsQ93833034
P433issue10
P304page(s)1126-1134
P577publication date1984-10-01
P1433published inExperientiaQ21385347
P1476titleInteraction of sulfonylurea with the pancreatic B-cell
P478volume40

Reverse relations

cites work (P2860)
Q33554980ATP-sensitive K+ channels that are blocked by hypoglycemia-inducing sulfonylureas in insulin-secreting cells are activated by galanin, a hyperglycemia-inducing hormone
Q44046827ATP-sensitive K-channels in HIT T15 beta-cells studied by patch-clamp methods, 86Rb efflux and glibenclamide binding
Q42173668An inhibitory role for polyamines in protein kinase C activation and insulin secretion in mouse pancreatic islets
Q69913208Beta-cell cytoplasmic Ca2+ balance as a determinant for glucose-stimulated insulin release
Q42856428Biosynthesis of insulin secretory granule membrane proteins. Control by glucose.
Q39504068Calcium transport in pancreatic beta-cells: implications for glucose regulation of insulin release
Q46790732Changes of membrane currents in cardiac cells induced by long whole-cell recordings and tolbutamide
Q57504439Characterization of sulfonylurea receptors in isolated human pancreatic islets
Q54128043Concentration-dependent effects of tolbutamide, meglitinide, glipizide, glibenclamide and diazoxide on ATP-regulated K+ currents in pancreatic B-cells.
Q38351945Direct measurements of increased free cytoplasmic Ca2+ in mouse pancreatic beta-cells following stimulation by hypoglycemic sulfonylureas
Q42857185Effect of perchlorate on calcium uptake and insulin secretion in mouse pancreatic islets
Q42465957Effects of porcine diazepam-binding inhibitor on insulin and glucagon secretion in vitro from the rat endocrine pancreas
Q42848672Effects of sulphonylureas and diazoxide on insulin secretion and nucleotide-sensitive channels in an insulin-secreting cell line
Q54107466Effects of verapamil and nifedipine on gliclazide-induced increase in cytosolic free Ca2+ in pancreatic islet cells.
Q35755181Highly potent and stereoselective effects of the benzoic acid derivative AZ-DF 265 on pancreatic beta-cells
Q69551659How do sulfonylureas approach their receptor in the B-cell plasma membrane?
Q41878159Inhibition by glibenclamide of the vasorelaxant action of cromakalim in the rat.
Q45835469Insulin secretory responses of a clonal cell line of simian virus 40-transformed B cells
Q70289261Internalization of 3H-glibenclamide in pancreatic islet cells
Q69972595Mechanism of the stimulation of insulin release in vitro by HB 699, a benzoic acid derivative similar to the non-sulphonylurea moiety of glibenclamide
Q44961703New mechanisms for sulfonylurea control of insulin secretion
Q44273170Opposite effects of tolbutamide and diazoxide on the ATP-dependent K+ channel in mouse pancreatic beta-cells
Q70222704Oral hypoglycemic agents
Q38631248Pharmacokinetic-pharmacodynamic relationships of oral hypoglycaemic agents. An update
Q38691347Pharmacology and regulation of ATP-sensitive K+ channels.
Q33992531Pharmacotherapy of type 2 diabetes mellitus
Q68922788Regulation of energy metabolism in pancreatic islets by glucose and tolbutamide
Q35043029Relationships between the Na(+)/K(+) pump and ATP and ADP content in mouse pancreatic islets: effects of meglitinide and glibenclamide
Q40078304Stimulus-secretion coupling in the pancreatic B-cell: concluding remarks
Q44119980Sulfonylurea-induced inhibition of glucagon secretion from the perfused rat pancreas: evidence for a direct, non-paracrine effect
Q51314532The effect of glibenclamide on insulin secretion at normal glucose concentrations.
Q44956244The oral hypoglycemic agent, U-56324, inhibits the activity of ATP-sensitive potassium channels in cell-free membrane patches from cultured mouse pancreatic B-cells
Q39662366The relationship between the pharmacokinetics and pharmacodynamic effects of oral hypoglycaemic drugs
Q45163742Tolbutamide potentiates the volume-regulated anion channel current in rat pancreatic beta cells

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