Homologous regulation of the alpha2C-adrenoceptor subtype in human hepatocarcinoma, HepG2.

scientific article published on January 1999

Homologous regulation of the alpha2C-adrenoceptor subtype in human hepatocarcinoma, HepG2. is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1038/SJ.BJP.0702269
P932PMC publication ID1565780
P698PubMed publication ID10051122
P5875ResearchGate publication ID240270867

P50authorCéline GalèsQ73251493
P2093author name stringParis H
Schaak S
Cayla C
Quinchon F
Roquelaine C
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Four consecutive serines in the third intracellular loop are the sites for beta-adrenergic receptor kinase-mediated phosphorylation and desensitization of the alpha 2A-adrenergic receptorQ34319907
The alpha 2-adrenoceptors of the human retinoblastoma cell line (Y79) may represent an additional example of the alpha 2C-adrenoceptorQ35870765
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Dynamin and beta-arrestin reveal distinct mechanisms for G protein-coupled receptor internalizationQ41176691
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Regulation of the alpha 2A-adrenergic receptor in the HT29 cell line. Effects of insulin and growth factorsQ41670263
Alpha 2A- and alpha 2C-adrenoceptor subtypes are differentially down-regulated by norepinephrineQ41674982
Inverse agonism and the regulation of receptor numberQ41698383
Desensitization of the alpha-2 adrenergic receptor in HT29 and opossum kidney cell linesQ41729360
Up-regulation of the levels of expression and function of a constitutively active mutant of the hamster alpha1B-adrenoceptor by ligands that act as inverse agonistsQ42443312
Inverse agonist-induced up-regulation of the human beta2-adrenoceptor in transfected neuroblastoma X glioma hybrid cells.Q42528165
Radioimmunoassay for cyclic nucleotides. I. Preparation of antibodies and iodinated cyclic nucleotidesQ43417658
Selective blockade and recovery of cell surface alpha 2-adrenergic receptors in human erythroleukemia (HEL) cells. Studies with the irreversible antagonist benextramineQ46524300
Analysis of radioligand binding experiments. A collection of computer programs for the IBM PC.Q46875721
Turnover of beta 1- and beta 2-adrenergic receptors after down-regulation or irreversible blockade.Q54136867
Subtype-selective desensitization of alpha 2-adrenergic receptors. Different mechanisms control short and long term agonist-promoted desensitization of alpha 2C10, alpha 2C4, and alpha 2C2Q67867385
[3H]L-657,743 (MK-912): a new, high affinity, selective radioligand for brain alpha 2-adrenoceptorsQ69368411
In vitro study of alpha 2-adrenoceptor turnover and metabolism using the adenocarcinoma cell line HT29Q69909670
G protein-coupled receptor kinase specificity for phosphorylation and desensitization of alpha2-adrenergic receptor subtypesQ71144208
The M(r) 35,000 beta-adrenergic receptor mRNA-binding protein binds transcripts of G-protein-linked receptors which undergo agonist-induced destabilizationQ72259884
P433issue1
P407language of work or nameEnglishQ1860
P304page(s)69-78
P577publication date1999-01-01
P1433published inBritish Journal of PharmacologyQ919631
P1476titleHomologous regulation of the alpha2C-adrenoceptor subtype in human hepatocarcinoma, HepG2
P478volume126

Reverse relations

cites work (P2860)
Q73898065Inverse agonism at alpha(2)-adrenoceptors in native tissue
Q44075447Ligand modulation of [35S]GTPgammaS binding at human alpha(2A), alpha(2B) and alpha(2C) adrenoceptors