In vivo binding affinities of cholecystokinin agonists and antagonists determined using the selective CCKB agonist [3H]pBC 264

scientific article published on December 17, 1991

In vivo binding affinities of cholecystokinin agonists and antagonists determined using the selective CCKB agonist [3H]pBC 264 is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1016/0014-2999(91)90168-P
P953full work available at URLhttps://api.elsevier.com/content/article/PII:001429999190168P?httpAccept=text/plain
https://api.elsevier.com/content/article/PII:001429999190168P?httpAccept=text/xml
P698PubMed publication ID1797561

P2093author name stringB. P. Roques
C. Durieux
M. Ruiz-Gayo
P2860cites workEvidence that CCKB receptors mediate the regulation of exploratory behaviour in the ratQ70198484
Cholecystokinin receptors: biochemical demonstration and autoradiographical localization in rat brain and pancreas using [3H] cholecystokinin8 as radioligandQ70202430
Cholecystokinin receptors: presence and axonal flow in the rat vagus nerveQ72645114
Pathway of inactivation of cholecystokinin octapeptide (CCK-8) by synaptosomal fractionsQ84269092
Opposite actions of CCK-8 on amphetamine-induced hyperlocomotion and stereotypy following intracerebroventricular and intra-accumbens injections in ratsQ41876087
A behavioural pharmacological study on intracerebroventricularly administered CCK-8 related peptides in miceQ41877188
Binding in vivo of selective mu and delta opioid receptor agonists: opioid receptor occupancy by endogenous enkephalinsQ42189417
Autoradiographic localization of cholecystokinin receptors in rodent brainQ42452814
Reduction of food intake by central administration of cholecystokinin octapeptide in the rat is dependent upon inhibition of brain peptidasesQ42848281
[3H]pBC 264, first highly potent and very selective radioligand for CCK-B receptorsQ46560963
Benzodiazepine gastrin and brain cholecystokinin receptor ligands: L-365,260.Q46782752
Occurrence of two cholecystokinin binding sites in guinea-pig brain cortexQ46798688
Autoradiography of CCK receptors in the rat brain using [(3)H]Boc[Nle(28)(31)]CCK(27)-(33) and [(125)I]bolton-hunter CCK(8). Functional significance of subregional distributions.Q47797242
Autoradiographic localization and biochemical characterization of peripheral type CCK receptors in rat CNS using highly selective nonpeptide CCK antagonistsQ48212288
Antinociceptive profile of sulfated CCK-8. Comparison with CCK-4, unsulfated CCK-8 and other neuropeptidesQ48312564
Intracerebroventricular injections of cholecystokinin octapeptide suppress feeding in rats--pharmacological characterization of this actionQ48324212
Investigation on the metabolism of CCK8 analogues by rat brain slicesQ48409939
Two brain cholecystokinin receptors: implications for behavioral actionsQ48417682
Endopeptidase-24.11 and aminopeptidase activity in brain synaptic membranes are jointly responsible for the hydrolysis of cholecystokinin octapeptide (CCK-8)Q48622391
In rats, the behavioral profile of CCK-8 related peptides resembles that of antipsychotic agentsQ48738164
Cholecystokinin octa- and tetrapeptide degradation by synaptic membranes. II. Solubilization and separation of membrane-bound CCK-8 cleaving enzymesQ48846221
Cholecystokinin receptors of A type in the human dorsal medulla oblongata and meningiomas, and of B type in small cell lung carcinomasQ48896243
Investigation of behavioral and electrophysiological responses induced by selective stimulation of CCKB receptors by using a new highly potent CCK analog, BC 264.Q48906138
Cholecystokinin tetrapeptide induces panic-like attacks in healthy volunteers. Preliminary findings.Q51176483
Cholecystokinin decreases food intake in rats.Q52320733
Enzyme-resistant CCK analogs with high affinities for central receptors.Q54380742
The enkephalinase inhibitor thiorphan shows antinociceptive activity in miceQ59063903
Postponement of satiety by blockade of brain cholecystokinin (CCK-B) receptorsQ60054766
Inhibitory effect of cholecystokinin octapeptide on neurons in the nucleus tractus solitariusQ67292773
Characterization of [3H] CCK4 binding sites in mouse and rat brainQ68059398
Antinociceptive action of cholecystokinin octapeptide (CCK 8) and related peptides in rats and mice: effects of naloxone and peptidase inhibitorsQ68156534
The selective CCK-B receptor antagonist L-365,260 enhances morphine analgesia and prevents morphine tolerance in the ratQ28278422
Development of a class of selective cholecystokinin type B receptor antagonists having potent anxiolytic activityQ28334293
Distinct cholecystokinin receptors in brain and pancreasQ28366068
A serine peptidase responsible for the inactivation of endogenous cholecystokinin in brainQ33666542
PD134308, a selective antagonist of cholecystokinin type B receptor, enhances the analgesic effect of morphine and synergistically interacts with intrathecal galanin to depress spinal nociceptive reflexesQ33792380
Design of potent, orally effective, nonpeptidal antagonists of the peptide hormone cholecystokininQ35615472
Evidence for an involvement of the brain cholecystokinin B receptor in anxietyQ37395948
Cholecystokinin and anxietyQ37948721
The role of CCK caerulein, and CCK antagonists in nociceptionQ38759937
P433issue3
P407language of work or nameEnglishQ1860
P921main subjectpharmacologyQ128406
phenylurea compoundsQ77806913
cholecystokininQ60315441
P304page(s)185-193
P577publication date1991-12-01
1991-12-17
P1433published inEuropean Journal of PharmacologyQ1376712
P1476titleIn vivo binding affinities of cholecystokinin agonists and antagonists determined using the selective CCKB agonist [3H]pBC 264
P478volume209

Reverse relations

cites work (P2860)
Q44344851Antidepressant-like effects of CCK(B) receptor antagonists: involvement of the opioid system
Q34341269CCK-B antagonists exhibit antidepressant-like effects and potentiate endogenous enkephalin analgesia. Correlation with in vivo binding affinities and brain penetration
Q28137628CCK-B receptor: chemistry, molecular biology, biochemistry and pharmacology
Q42446053Cholecystokinin (CCK-8) modulates vesicular release of excitatory amino acids in rat hippocampal nerve endings
Q63966523Cholecystokinin receptor agonists block the jumping behaviour precipitated in morphine-dependent mice by naloxone
Q44443009Effect of peripheral cholecystokinin receptor agonists on c-Fos expression in brain sites mediating food consumption in rats
Q73850248Multiple emulsion technology for the design of microspheres containing peptides and oligopeptides

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