Influence of a new 5-HT4 receptor partial agonist, YKP10811, on visceral hypersensitivity in rats triggered by stress and inflammation

scientific article published on 15 October 2014

Influence of a new 5-HT4 receptor partial agonist, YKP10811, on visceral hypersensitivity in rats triggered by stress and inflammation is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1111/NMO.12458
P698PubMed publication ID25316608

P2093author name stringH Han
H Eutamene
L Bueno
H W Kim
M Gilet
P2860cites workThe 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivoQ24671423
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Activation of colonic mucosal 5-HT(4) receptors accelerates propulsive motility and inhibits visceral hypersensitivity.Q36336675
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5-HT(2B) receptors modulate visceral hypersensitivity in a stress-sensitive animal model of brain-gut axis dysfunctionQ39294409
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5-Hydroxytryptamine4 receptor agonists initiate the peristaltic reflex in human, rat, and guinea pig intestineQ45112735
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Stress-induced visceral hypersensitivity to rectal distension in rats: role of CRF and mast cellsQ48548051
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P433issue12
P304page(s)1761-1770
P577publication date2014-10-15
P1433published inNeurogastroenterology and MotilityQ15767493
P1476titleInfluence of a new 5-HT4 receptor partial agonist, YKP10811, on visceral hypersensitivity in rats triggered by stress and inflammation
P478volume26

Reverse relations

cites work (P2860)
Q38376282Animal models of gastrointestinal and liver diseases. Animal models of visceral pain: pathophysiology, translational relevance, and challenges
Q36082843Early investigational therapeutics for gastrointestinal motility disorders: from animal studies to Phase II trials
Q48350930Effect of prucalopride on intestinal gas tolerance in patients with functional bowel disorders and constipation
Q36828610Enteroendocrine cells: a review of their role in brain-gut communication
Q48168717Localization of the 5-hydroxytryptamine 4 receptor in equine enteric neurons and extrinsic sensory fibers.
Q38696256Novel investigational drugs for constipation-predominant irritable bowel syndrome: a review
Q41392745Pharmacological Approach for Managing Pain in Irritable Bowel Syndrome: A Review Article
Q48048742Prokinetic effects of a new 5-HT4 agonist, YKP10811, on gastric motility in dogs
Q88945541Prokinetics in the Management of Functional Gastrointestinal Disorders
Q39303889Sex-Related Differences in GI Disorders
Q47171305Stress-Induced Chronic Visceral Pain of Gastrointestinal Origin

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