Synthetic hydrophobic peptides are substrates for P-glycoprotein and stimulate drug transport

scientific article published on December 1996

Synthetic hydrophobic peptides are substrates for P-glycoprotein and stimulate drug transport is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1042/BJ3200421
P932PMC publication ID1217947
P698PubMed publication ID8973548
P5875ResearchGate publication ID14233429

P2093author name stringX Yu
J W Chu
F J Sharom
G DiDiodato
P2860cites workPhosphatidylcholine translocase: a physiological role for the mdr2 geneQ24319732
Homozygous disruption of the murine mdr2 P-glycoprotein gene leads to a complete absence of phospholipid from bile and to liver diseaseQ24322810
A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye bindingQ25938984
ABC Transporters: From Microorganisms to ManQ28181688
Biochemistry of multidrug resistance mediated by the multidrug transporterQ29616476
Photoaffinity labeling of the multidrug-resistance-related P-glycoprotein with photoactive analogs of verapamilQ33651186
Disruption of the mouse mdr1a P-glycoprotein gene leads to a deficiency in the blood-brain barrier and to increased sensitivity to drugsQ34059522
ATP-dependent bacterial transporters and cystic fibrosis: analogy between channels and transportersQ35323989
Interaction of multidrug-resistant Chinese hamster ovary cells with amphiphilesQ35977177
Multidrug resistance and chemosensitization: therapeutic implications for cancer chemotherapy.Q38014962
Characterization and functional reconstitution of the multidrug transporterQ40456754
Allosteric regulation of [3H]vinblastine binding to P-glycoprotein of MCF-7 ADR cells by dexniguldipineQ41334626
Tamoxifen aziridine, a novel affinity probe for P-glycoprotein in multidrug resistant cellsQ41454968
Characterization of the ATPase activity of purified Chinese hamster P-glycoproteinQ41461421
Stoichiometric labeling of peptides by iodination on tyrosyl or histidyl residuesQ41561181
Characterization of the adenosine triphosphatase activity of Chinese hamster P-glycoprotein.Q41572777
The effects of lipids and detergents on ATPase-active P-glycoproteinQ41572851
Transport properties of P-glycoprotein in plasma membrane vesicles from multidrug-resistant Chinese hamster ovary cellsQ41607862
Peptide transport by the multidrug resistance pumpQ41634191
Physical-chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells.Q41912189
Interaction of bioactive hydrophobic peptides with the human multidrug transporterQ42068296
Interaction of prenylcysteine methyl esters with the multidrug resistance transporterQ42068347
Characterization of the ATPase activity of P-glycoprotein from multidrug-resistant Chinese hamster ovary cellsQ42486411
Detection of P-glycoprotein in multidrug-resistant cell lines by monoclonal antibodiesQ42812351
ATPase activity of purified and reconstituted P-glycoprotein from Chinese hamster ovary cells.Q54214354
Functional complementation of yeast ste6 by a mammalian multidrug resistance mdr geneQ54272057
Strategies for the purification of P-glycoprotein from multidrug-resistant Chinese hamster ovary cellsQ54291890
Identification of the multidrug resistance-related membrane glycoprotein as an acceptor for calcium channel blockers.Q54405185
ATPase activity of partially purified P-glycoprotein from multidrug-resistant Chinese hamster ovary cellsQ67520844
The intracellular content of dihydrofolate reductase: possibilities for control and implications for chemotherapyQ70605968
Interaction of multidrug-resistant Chinese hamster ovary cells with the peptide ionophore gramicidin DQ71611332
The effect of verapamil on the transport of peptides across the blood-brain barrier in rats: kinetic evidence for an apically polarized efflux mechanismQ72151415
Interaction of the P-glycoprotein multidrug transporter with peptides and ionophoresQ72191051
Functional reconstitution of drug transport and ATPase activity in proteoliposomes containing partially purified P-glycoproteinQ72656274
Covalent inhibitors of P-glycoprotein ATPase activityQ72671369
P407language of work or nameEnglishQ1860
P921main subjecthydrophobicityQ41854968
P304page(s)421-428
P577publication date1996-12-01
P1433published inBiochemical JournalQ864221
P1476titleSynthetic hydrophobic peptides are substrates for P-glycoprotein and stimulate drug transport
P478volume320 ( Pt 2)

Reverse relations

cites work (P2860)
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