scholarly article | Q13442814 |
P50 | author | Pengyu Ren | Q45710729 |
Jiney Jose | Q61822666 | ||
P2093 | author name string | Chunli Yan | |
Yue Shi | |||
Qiantao Wang | |||
Kevin N Dalby | |||
Ashwini K Devkota | |||
Tamer S Kaoud | |||
Eun Jeong Cho | |||
Ramakrishna Edupuganti | |||
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Calcium/calmodulin stimulates the autophosphorylation of elongation factor 2 kinase on Thr-348 and Ser-500 to regulate its activity and calcium dependence | Q28259597 | ||
The Role of Eukaryotic Elongation Factor 2 Kinase in Rapid Antidepressant Action of Ketamine | Q28276943 | ||
The eEF2 kinase confers resistance to nutrient deprivation by blocking translation elongation | Q28291406 | ||
Targeting cancer with small molecule kinase inhibitors | Q29547395 | ||
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NMDA receptor blockade at rest triggers rapid behavioural antidepressant responses | Q30471587 | ||
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Cytoprotective effect of the elongation factor-2 kinase-mediated autophagy in breast cancer cells subjected to growth factor inhibition | Q33543073 | ||
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Targeted silencing of elongation factor 2 kinase suppresses growth and sensitizes tumors to doxorubicin in an orthotopic model of breast cancer | Q34387697 | ||
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Purification and characterization of tagless recombinant human elongation factor 2 kinase (eEF-2K) expressed in Escherichia coli. | Q36075643 | ||
Activated ERK2 Is a Monomer in Vitro with or without Divalent Cations and When Complexed to the Cytoplasmic Scaffold PEA-15 | Q36107198 | ||
From in Silico Discovery to intra-Cellular Activity: Targeting JNK-Protein Interactions with Small Molecules | Q36243062 | ||
Activity and regulation by growth factors of calmodulin-dependent protein kinase III (elongation factor 2-kinase) in human breast cancer | Q36617301 | ||
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1-Benzyl-3-cetyl-2-methylimidazolium iodide (NH125) induces phosphorylation of eukaryotic elongation factor-2 (eEF2): a cautionary note on the anticancer mechanism of an eEF2 kinase inhibitor | Q39454084 | ||
Irreversible Nek2 kinase inhibitors with cellular activity | Q39533198 | ||
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Silencing of elongation factor-2 kinase potentiates the effect of 2-deoxy-D-glucose against human glioma cells through blunting of autophagy | Q39879662 | ||
Structural bioinformatics-based design of selective, irreversible kinase inhibitors | Q40307105 | ||
Identification and characterization of an inhibitor of eukaryotic elongation factor 2 kinase against human cancer cell lines | Q40622035 | ||
Transient inhibition of protein synthesis induces expression of proto-oncogenes and stimulates resting cells to enter the cell cycle | Q41263722 | ||
Cysteine mapping in conformationally distinct kinase nucleotide binding sites: application to the design of selective covalent inhibitors. | Q42750517 | ||
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Cysteine Proteases and Their Inhibitors | Q61066438 | ||
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P433 | issue | 16 | |
P304 | page(s) | 2435-2442 | |
P577 | publication date | 2014-09-15 | |
P1433 | published in | ChemBioChem | Q634395 |
P1476 | title | Reversible covalent inhibition of eEF-2K by carbonitriles | |
P478 | volume | 15 |
Q54978227 | Structural Dynamics of the Activation of Elongation Factor 2 Kinase by Ca2+-Calmodulin. |
Q27727833 | Structure of the C-Terminal Helical Repeat Domain of Eukaryotic Elongation Factor 2 Kinase |
Q38931379 | Targeted Covalent Inhibitors for Drug Design. |
Q40608421 | Using docking and alchemical free energy approach to determine the binding mechanism of eEF2K inhibitors and prioritizing the compound synthesis |
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