E-2078, a potent, selective and stable dynorphin analog with preferential activity for the kappa-opioid receptor subtype on the mouse vas deferens neuroeffector junction

scientific article published on November 1, 1991

E-2078, a potent, selective and stable dynorphin analog with preferential activity for the kappa-opioid receptor subtype on the mouse vas deferens neuroeffector junction is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1016/0196-9781(91)90196-V
P953full work available at URLhttps://api.elsevier.com/content/article/PII:019697819190196V?httpAccept=text/plain
https://api.elsevier.com/content/article/PII:019697819190196V?httpAccept=text/xml
P698PubMed publication ID1687708

P2093author name stringS. Tachibana
J. P. Huidobro-Toro
R. Valenzuela
Huidobro-Toro JP
P2860cites workNaltrindole, a highly selective and potent non-peptide delta opioid receptor antagonistQ28280800
Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonistsQ34559354
Endogenous opioid peptides: multiple agonists and receptorsQ34986433
Porcine pituitary dynorphin: complete amino acid sequence of the biologically active heptadecapeptideQ36380726
Application of an irreversible opiate antagonist (β-FNA, β-funal-trexamine) to demonstrate dynorphin selectivity for K-opioid sitesQ41533856
Pharmacological profile of PD 117302, a selective kappa-opioid agonistQ41813703
Interactions between morphine and the opioid-like peptides in the rat vas deferensQ42116276
Lack of mixed agonist-antagonist properties of [Gln8-Gly31]-beta h-EP-Gly-Gly-NH2 and [Arg9,19,24,28,29]-beta h-EP in the rat vas deferens neuroeffector junction: studies with naloxone, beta-funaltrexamine and ICI 174,864.Q42155805
PD117302: a selective agonist for the kappa-opioid receptorQ42849304
Rabbit vas deferens: A specific bioassay for opioid κ-receptor agonistsQ44352972
Evidence that dynorphin-(1–13) acts as an agonist on opioid κ-receptorsQ44353022
The irreversible narcotic antagonistic and reversible agonistic properties of the fumaramate methyl ester derivative of naltrexoneQ46222547
Synthesis and structure-activity relationships of dynorphin A-(1-8) amide analoguesQ46258920
Dynorphin interaction at the κ-opiate siteQ72480926
P433issue6
P407language of work or nameEnglishQ1860
P921main subjectphysiologyQ521
biochemistryQ7094
endocrinologyQ162606
dynorphinQ324076
P1104number of pages4
P304page(s)1211-1214
P577publication date1991-11-01
P1433published inPeptidesQ7166533
P1476titleE-2078, a potent, selective and stable dynorphin analog with preferential activity for the kappa-opioid receptor subtype on the mouse vas deferens neuroeffector junction
P478volume12