Design and synthesis of bis-amide and hydrazide-containing derivatives of malonic acid as potential HIV-1 integrase inhibitors.

scientific article published in October 2008

Design and synthesis of bis-amide and hydrazide-containing derivatives of malonic acid as potential HIV-1 integrase inhibitors. is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.3390/MOLECULES13102442
P932PMC publication ID6245433
P698PubMed publication ID18830166
P5875ResearchGate publication ID239273779

P50authorRoberto DallocchioQ59172807
Mario SechiQ38545838
Nicolino PalaQ42750481
Alessandro DessìQ49838493
P2093author name stringNouri Neamati
Ugo Azzena
Alessia Cosseddu
Maria Paola Delussu
P2860cites workOrdered water and ligand mobility in the HIV-1 integrase-5CITEP complex: a molecular dynamics studyQ53886381
Distributed automated docking of flexible ligands to proteins: Parallel applications of AutoDock 2.4Q57976081
Structure of a copper-isoniazid complexQ71578791
Potential anticancer agents. I. Synthesis of some nitrogen mustard containing benzylidenehydrazidesQ72020524
Some derivatives of oxanilideQ83207553
Prostaglandin-H synthase inhibition by malonamides. Ring-opened analogues of phenylbutazoneQ93536677
Structure of the HIV-1 integrase catalytic domain complexed with an inhibitor: a platform for antiviral drug designQ27620348
Iterative partial equalization of orbital electronegativity—a rapid access to atomic chargesQ28096294
Python: a programming language for software integration and developmentQ29614317
HIV-1 integrase inhibitors: past, present, and futureQ34050694
Molecular dynamics studies of the wild-type and double mutant HIV-1 integrase complexed with the 5CITEP inhibitor: mechanism for inhibition and drug resistanceQ34180538
Integrase inhibitors to treat HIV/AIDS.Q34397376
HIV-1 integrase: from biology to chemotherapeutics.Q36879253
HIV-1 integrase inhibitors: update and perspectivesQ37034614
Patented HIV-1 integrase inhibitors (1998-2005).Q37067128
Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitorsQ40547803
Metal-dependent inhibition of HIV-1 integraseQ40684087
Active site binding modes of HIV-1 integrase inhibitorsQ43846931
From ligand to complexes: inhibition of human immunodeficiency virus type 1 integrase by beta-diketo acid metal complexes.Q44619681
P275copyright licenseCreative Commons Attribution 4.0 InternationalQ20007257
P6216copyright statuscopyrightedQ50423863
P433issue10
P407language of work or nameEnglishQ1860
P304page(s)2442-2461
P577publication date2008-10-01
P1433published inMoleculesQ151332
P1476titleDesign and synthesis of bis-amide and hydrazide-containing derivatives of malonic acid as potential HIV-1 integrase inhibitors
P478volume13

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cites work (P2860)
Q41970138Crystal structure of 2-cyano-N'-(cyclo-hexyl-idene)acetohydrazide
Q45998555Efficient synthesis of 4-oxo-4,5-dihydrothieno[3,2-c]quinoline-2-carboxylic acid derivatives from aniline.
Q33991491Microwave assisted organic synthesis (MAOS) of small molecules as potential HIV-1 integrase inhibitors.
Q28534627Mutational analysis of the binding pockets of the diketo acid inhibitor L-742,001 in the influenza virus PA endonuclease
Q87557172Spectroscopic and quantum mechanical investigation of N,N'-bisarylmalonamides: solvent and structural effects
Q33755920Synthesis and bioactivity of 5-substituted-2-furoyl diacylhydazide derivatives with aliphatic chain
Q42720272Synthesis of a new group of aliphatic hydrazide derivatives and the correlations between their molecular structure and biological activity.
Q37156847Synthesis, physiochemical properties, photochemical probe, and antimicrobial effects of novel norfloxacin analogues
Q35960631Virtual Screening and Biological Validation of Novel Influenza Virus PA Endonuclease Inhibitors.

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