Striking differences of action of lisuride stereoisomers at histamine H1 receptors

scientific article

Striking differences of action of lisuride stereoisomers at histamine H1 receptors is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1007/S00210-006-0111-0
P698PubMed publication ID17106670

P2093author name stringRoland Seifert
Heinz H Pertz
Andrea Strasser
Tilo Görnemann
Björn Schurad
P2860cites workRelationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionQ27860958
Differential actions of antiparkinson agents at multiple classes of monoaminergic receptor. I. A multivariate analysis of the binding profiles of 14 drugs at 21 native and cloned human receptor subtypesQ28208581
Differential actions of antiparkinson agents at multiple classes of monoaminergic receptor. II. Agonist and antagonist properties at subtypes of dopamine D(2)-like receptor and alpha(1)/alpha(2)-adrenoceptorQ28208591
International Union of Pharmacology. XIII. Classification of histamine receptorsQ28249809
Partial agonists, full agonists, antagonists: dilemmas of definitionQ36741987
The classification of seven transmembrane receptors in recombinant expression systemsQ41185384
An analysis of the direct and indirect actions of drugs on the isolated guinea-pig ileumQ41377111
8R-lisuride is a potent stereospecific histamine H1-receptor partial agonistQ42831275
Emerging views of dopamine in modulating sleep/wake state from an unlikely source: PD.Q43882541
Multiple differences in agonist and antagonist pharmacology between human and guinea pig histamine H1-receptorQ44355508
Pharmacological differences between human and guinea pig histamine H1 receptors: Asn84 (2.61) as key residue within an additional binding pocket in the H1 receptorQ45207500
Guinea pig histamine H1 receptor. II. Stable expression in Chinese hamster ovary cells reveals the interaction with three major signal transduction pathwaysQ46184989
Identification of 5HT2-receptors on longitudinal muscle of the guinea pig ileumQ46270600
Increased levels of extracellular dopamine in neostriatum and nucleus accumbens after histamine H1 receptor blockadeQ48344452
Selectivity of some ergot derivatives for 5-HT1 and 5-HT2 receptors of rat cerebral cortexQ48389799
On the statistics of drug-receptor constants for partial agonistsQ52843199
Cumulative dose-response curves. II. Technique for the making of dose-response curves in isolated organs and the evaluation of drug parametersQ79695858
P433issue3
P304page(s)215-222
P577publication date2006-11-08
P1433published inNaunyn-Schmiedeberg's Archives of PharmacologyQ1468251
P1476titleStriking differences of action of lisuride stereoisomers at histamine H1 receptors
P478volume374

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cites work (P2860)
Q461837663D-QSAR CoMFA Study to Predict Orientation of Suprahistaprodifens and Phenoprodifens in the Binding-Pocket of Four Histamine H1 -Receptor Species
Q42020167Comparison of the pharmacological properties of human and rat histamine H3-receptors
Q37327413Functional pharmacology of H1 histamine receptors expressed in mouse preoptic/anterior hypothalamic neurons
Q48812098Interactions of recombinant human histamine H₁R, H₂R, H₃R, and H₄R receptors with 34 antidepressants and antipsychotics
Q46861009Pharmacological properties of a wide array of ergolines at functional alpha(1)-adrenoceptor subtypes

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