Computational and biological profile of boronic acids for the detection of bacterial serine- and metallo-β-lactamases.

scientific article published on 18 December 2017

Computational and biological profile of boronic acids for the detection of bacterial serine- and metallo-β-lactamases. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1038/S41598-017-17399-7
P932PMC publication ID5735191
P698PubMed publication ID29255163

P50authorJean-Denis DocquierQ28324616
Gabriele CrucianiQ56858982
Donatella TondiQ57975565
Antonio QuotadamoQ60620220
Jesus BlazquezQ68273789
P2093author name stringFrancesca Spyrakis
Alberto Venturelli
Simon Cross
Davide Farina
Maria Paola Costi
Ana Isabel Prieto
Matteo Santucci
Filomena De Luca
Claudia Ibacache
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P275copyright licenseCreative Commons Attribution 4.0 InternationalQ20007257
P6216copyright statuscopyrightedQ50423863
P433issue1
P407language of work or nameEnglishQ1860
P921main subjectboronic acidQ335768
biological profileQ118125750
P304page(s)17716
P577publication date2017-12-18
P1433published inScientific ReportsQ2261792
P1476titleComputational and biological profile of boronic acids for the detection of bacterial serine- and metallo-β-lactamases
P478volume7

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cites work (P2860)
Q906628784-Amino-1,2,4-triazole-3-thione as a Promising Scaffold for the Inhibition of Serine and Metallo-β-Lactamases
Q92728030Forecasting from phenotypic testing to an antimicrobial stewardship strategy: Does the time to positivity of a blue-carba test predict the meropenem susceptibility level among carbapenemase producers?
Q60049273In silico identification and experimental validation of hits active against KPC-2 β-lactamase
Q50093207Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance.
Q90419283Phenylboronic Acids Probing Molecular Recognition against Class A and Class C β-lactamases
Q59830619Targeting Metalloenzymes for Therapeutic Intervention
Q98164385Virtual screening identifies broad-spectrum β-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases
Q93166853X-ray Crystallography Deciphers the Activity of Broad-Spectrum Boronic Acid β-Lactamase Inhibitors

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