scholarly article | Q13442814 |
P356 | DOI | 10.1002/CMDC.201600539 |
P698 | PubMed publication ID | 28264138 |
P50 | author | András Kotschy | Q73252492 |
P2093 | author name string | Csaba Wéber | |
Francisco Cruzalegui | |||
Balázs Bálint | |||
Mike Burbridge | |||
P2860 | cites work | Sequence characteristics, subcellular localization, and substrate specificity of DYRK-related kinases, a novel family of dual specificity protein kinases | Q24316021 |
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Synthesis and biological evaluation of N(9)-substituted harmine derivatives as potential anticancer agents | Q38758935 | ||
Synthesis, cytotoxic, anti-lipoxygenase and anti-acetylcholinesterase capacities of novel derivatives from harmine. | Q38782393 | ||
Hydroxybenzothiophene Ketones Are Efficient Pre-mRNA Splicing Modulators Due to Dual Inhibition of Dyrk1A and Clk1/4 | Q41739576 | ||
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A novel DYRK1A (dual specificity tyrosine phosphorylation-regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro. | Q42702995 | ||
High-affinity binding of beta-carbolines to imidazoline I2B receptors and MAO-A in rat tissues: norharman blocks the effect of morphine withdrawal on DOPA/noradrenaline synthesis in the brain | Q46629739 | ||
First selective dual inhibitors of tau phosphorylation and Beta-amyloid aggregation, two major pathogenic mechanisms in Alzheimer's disease | Q48523309 | ||
Computational & experimental evaluation of the structure/activity relationship of β-carbolines as DYRK1A inhibitors. | Q55071094 | ||
Localization of monoamine oxidases in human peripheral tissues | Q61849213 | ||
P433 | issue | 12 | |
P304 | page(s) | 932-939 | |
P577 | publication date | 2017-04-06 | |
P1433 | published in | ChemMedChem | Q2962252 |
P1476 | title | Structure-Based Design and Synthesis of Harmine Derivatives with Different Selectivity Profiles in Kinase versus Monoamine Oxidase Inhibition | |
P478 | volume | 12 |
Q96958956 | A Dual Inhibitor of DYRK1A and GSK3β for β-Cell Proliferation: Aminopyrazine Derivative GNF4877 |
Q90610025 | Development of Kinase-Selective, Harmine-Based DYRK1A Inhibitors that Induce Pancreatic Human β-Cell Proliferation |
Q54107922 | Isoform selectivity of harmine-conjugated 1,2,3-triazoles against human monoamine oxidase. |
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