The simultaneous estimation of the influx and efflux blood-brain barrier permeabilities of gabapentin using a microdialysis-pharmacokinetic approach.

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The simultaneous estimation of the influx and efflux blood-brain barrier permeabilities of gabapentin using a microdialysis-pharmacokinetic approach. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1023/A:1016092525901
P698PubMed publication ID8692732

P2093author name stringY Wang
D F Welty
P2860cites workTransport of gabapentin, a gamma-amino acid drug, by system l alpha-amino acid transporters: a comparative study in astrocytes, synaptosomes, and CHO cellsQ72169569
Gabapentin anticonvulsant action in rats: disequilibrium with peak drug concentrations in plasma and brain microdialysateQ72270715
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Selected CSF biochemistry and gabapentin concentrations in the CSF and plasma in patients with partial seizures after a single oral dose of gabapentinQ45012245
Diet and uptake of aldomet by the brain: competition with natural large neutral amino acidsQ48265693
An in situ brain perfusion technique to study cerebrovascular transport in the rat.Q48627674
The use of an "internal standard" for control of the recovery in microdialysis.Q51720194
Zidovudine transport in the rabbit brain during intravenous and intracerebroventricular infusion.Q52337785
Microdialysis study of zidovudine (AZT) transport in rat brain.Q52387285
A saturable transport mechanism in the intestinal absorption of gabapentin is the underlying cause of the lack of proportionality between increasing dose and drug levels in plasmaQ70618602
Disposition of gabapentin (neurontin) in mice, rats, dogs, and monkeysQ71845183
P433issue3
P921main subjectblood–brain barrierQ221694
pharmacokineticsQ323936
gabapentinQ410352
P304page(s)398-403
P577publication date1996-03-01
P1433published inPharmaceutical ResearchQ7180737
P1476titleThe simultaneous estimation of the influx and efflux blood-brain barrier permeabilities of gabapentin using a microdialysis-pharmacokinetic approach.
P478volume13

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