Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters.

scientific article published on 11 December 2013

Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1002/CHEM.201303409
P698PubMed publication ID24339325

P50authorMarkus R. HeinrichQ39402207
Peter GmeinerQ42185465
Olaf PranteQ85917743
P2093author name stringNuska Tschammer
Harald Hübner
Simone Maschauer
Stefanie K Fehler
Amelie L Bartuschat
Sarah B Höfling
P2860cites workThe growing impact of bioorthogonal click chemistry on the development of radiopharmaceuticalsQ26849599
Modeling of PET data in CNS drug discovery and developmentQ30623699
Synopsis of some recent tactical application of bioisosteres in drug designQ34171394
A fluoride-derived electrophilic late-stage fluorination reagent for PET imaging.Q34230071
Single-step syntheses of no-carrier-added functionalized [18F]fluoroarenes as labeling synthons from diaryliodonium salts.Q34284978
No-carrier-added [18F]fluoroarenes from the radiofluorination of diaryl sulfoxides.Q36655909
Radiofluorination of diaryliodonium tosylates under aqueous-organic and cryptand-free conditionsQ37056100
Synthesis using aromatic homolytic substitution--recent advancesQ37063223
Synthesis of 11C, 18F, 15O, and 13N radiolabels for positron emission tomography.Q37318975
Current state of agonist radioligands for imaging of brain dopamine D2/D3 receptors in vivo with positron emission tomographyQ37768194
Recent advances in the search for D3- and D4-selective drugs: probes, models and candidatesQ37828272
Absolute abundances and affinity states of dopamine receptors in mammalian brain: A reviewQ37838858
Modern developments in aryl radical chemistryQ37867035
Positron emission tomography in psychiatric disordersQ37975237
Radiolabelled RGD peptides for imaging and therapyQ37990409
18F labeling of arenes.Q38053980
Radioligands for the dopamine receptor subtypesQ38166968
Labeling and glycosylation of peptides using click chemistry: a general approach to (18)F-glycopeptides as effective imaging probes for positron emission tomographyQ39759909
4-Substituted tert-butyl phenylazocarboxylates--synthetic equivalents for the para-phenyl radical cationQ42823978
Synthesis, biological evaluation and radiolabelling by 18F-fluoroarylation of a dopamine D3-selective ligand as prospective imaging probe for PET.Q42844373
Radiosynthesis and evaluation of [18F]Selectfluor bis(triflate).Q42935493
Fast production of highly reactive no-carrier-added [18F]fluoride for the labeling of radiopharmaceuticalsQ43117766
Three-step, "one-pot" radiosynthesis of 6-fluoro-3,4-dihydroxy-L-phenylalanine by isotopic exchangeQ43275687
A biomathematical modeling approach to central nervous system radioligand discovery and developmentQ44032522
N-(omega-(4-(2-methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as dopamine D2 and D3 receptor ligandsQ44557234
[18F]fluorination of an arylboronic ester using [18F]selectfluor bis(triflate): application to 6-[18F]fluoro-L-DOPA.Q44562624
Dopamine D2, D3, and D4 selective phenylpiperazines as molecular probes to explore the origins of subtype specific receptor binding.Q45927941
Dopamine (D2/3) receptor agonist positron emission tomography radiotracer [11C]-(+)-PHNO is a D3 receptor preferring agonist in vivoQ48429468
Oxalic acid supported Si-18F-radiofluorination: one-step radiosynthesis of N-succinimidyl 3-(di-tert-butyl[18F]fluorosilyl)benzoate ([18F]SiFB) for protein labelingQ48794678
Radiochemistry: Flipping fluoride's reactivity.Q53174138
Positron emission tomography using [18F]Galacto-RGD identifies the level of integrin alpha(v)beta3 expression in man.Q53530857
Radical reactions of arenediazonium ions: An easy entry into the chemistry of the aryl radicalQ57256651
P433issue2
P407language of work or nameEnglishQ1860
P304page(s)370-375
P577publication date2013-12-11
P1433published inChemistry—A European JournalQ898737
P1476titleFast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters.
P478volume20

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cites work (P2860)
Q3826252418F-labelled intermediates for radiosynthesis by modular build-up reactions: newer developments
Q51007789Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior.
Q39369099Fluorine-18 labelled building blocks for PET tracer synthesis
Q38950052Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.
Q48534307In Vitro and In Vivo Characterization of Selected Fluorine-18 Labeled Radioligands for PET Imaging of the Dopamine D3 Receptor.
Q48303344Microwave-Assisted Rapid One-Pot Synthesis of Fused and Non-Fused Indoles and 5-[18 F]Fluoroindoles from Phenylazocarboxylates
Q94600975Synthesis, biological evaluation and radiosynthesis of buprenorphine-derived phenylazocarboxamides as novel μ-opioid receptor ligands
Q50325135[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor

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