Mass Spectrometry Reveals That the Antibiotic Simocyclinone D8 Binds to DNA Gyrase in a “Bent-Over” Conformation: Evidence of Positive Cooperativity in Binding

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Mass Spectrometry Reveals That the Antibiotic Simocyclinone D8 Binds to DNA Gyrase in a “Bent-Over” Conformation: Evidence of Positive Cooperativity in Binding is …
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scholarly articleQ13442814

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P356DOI10.1021/BI101691K
P698PubMed publication ID21338149

P50authorMark A WilliamsQ55743744
Anthony MaxwellQ37380949
P2093author name stringAdam R McKay
Marcus J Edwards
P2860cites workSimocyclinones, Novel Cytostatic Angucyclinone Antibiotics Produced by Streptomyces antibioticus Tue 6040. II. Structure Elucidation and Biosynthesis.Q78429069
Simocyclinones, Novel Cytostatic Angucyclinone Antibiotics Produced by Streptomyces antibioticus Tue 6040. I. Taxonomy, Fermentation, Isolation and Biological Activities.Q104949753
P433issue17
P407language of work or nameEnglishQ1860
P921main subjectantibioticQ12187
P1104number of pages9
P304page(s)3432-3440
P577publication date2011-04-05
P1433published inBiochemistryQ764876
P1476titleMass spectrometry reveals that the antibiotic simocyclinone D8 binds to DNA gyrase in a "bent-over" conformation: evidence of positive cooperativity in binding
P478volume50