Co-amorphous solid dispersion systems of lacidipine-spironolactone with improved dissolution rate and enhanced physical stability

scientific article published on 14 November 2018

Co-amorphous solid dispersion systems of lacidipine-spironolactone with improved dissolution rate and enhanced physical stability is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1016/J.AJPS.2018.11.001
P932PMC publication ID7032115
P698PubMed publication ID32104442

P2093author name stringQing Ye
Tian Liu
Jin Sun
Zhonggui He
Xiao Tan
Dun Wang
Zhaomeng Wang
Mengchi Sun
Zisen Gao
Yanxian Hou
P2860cites workInfluence of physicochemical properties on dissolution of drugs in the gastrointestinal tractQ34190317
Rod shaped nanocrystals exhibit superior in vitro dissolution and in vivo bioavailability over spherical like nanocrystals: a case study of lovastatinQ35576407
Solid state characterization of azelnidipine-oxalic acid co-crystal and co-amorphous complexes: The effect of different azelnidipine polymorphsQ36290858
Effective management of hypertension with dihydropyridine calcium channel blocker-based combination therapy in patients at high cardiovascular riskQ36572955
Pharmaceutical excipients - quality, regulatory and biopharmaceutical considerationsQ38677702
Recent advances in co-amorphous drug formulationsQ38710042
Influence of variation in molar ratio on co-amorphous drug-amino acid systemsQ39638481
Formation Mechanism of Coamorphous Drug-Amino Acid Mixtures.Q40854029
Mechanism-based selection of stabilization strategy for amorphous formulations: Insights into crystallization pathwaysQ41016139
Supersaturating drug delivery systems: The potential of co-amorphous drug formulations.Q47718326
Viewing Molecular and Interface Interactions of Curcumin Amorphous Solid Dispersions for Comprehending Dissolution Mechanisms.Q47783687
Moisture-Induced Amorphous Phase Separation of Amorphous Solid Dispersions: Molecular Mechanism, Microstructure, and Its Impact on Dissolution PerformanceQ47810974
Probing Pharmaceutical Mixtures during Milling: The Potency of Low-Frequency Raman Spectroscopy in Identifying Disorder.Q47865775
Facile formation of co-amorphous atenolol and hydrochlorothiazide mixtures via cryogenic-milling: Enhanced physical stability, dissolution and pharmacokinetic profileQ47891325
Experimental observations and dissipative particle dynamic simulations on microstructures of pH-sensitive polymer containing amorphous solid dispersionsQ48921407
Coamorphous Active Pharmaceutical Ingredient-Small Molecule Mixtures: Considerations in the Choice of Coformers for Enhancing Dissolution and Oral BioavailabilityQ49496136
Solvent-shift strategy to identify suitable polymers to inhibit humidity-induced solid-state crystallization of lacidipine amorphous solid dispersions.Q50881261
Solid-state flurbiprofen and methyl-β-cyclodextrin inclusion complexes prepared using a single-step, organic solvent-free supercritical fluid process.Q51338534
Use of conventional surfactant media as surrogates for FaSSIF in simulating in vivo dissolution of BCS class II drugs.Q51379052
Coamorphous drug systems: enhanced physical stability and dissolution rate of indomethacin and naproxen.Q51542358
Physical Stability and Dissolution Behavior of Ketoconazole-Organic Acid Coamorphous Systems.Q53436393
Enhanced oral absorption of pemetrexed by ion-pairing complex formation with deoxycholic acid derivative and multiple nanoemulsion formulations: preparation, characterization, and in vivo oral bioavailability and anticancer effect.Q55248249
Predicting final product properties of melt extruded solid dispersions from process parameters using Raman spectrometryQ57162915
Co-amorphous simvastatin and glipizide combinations show improved physical stability without evidence of intermolecular interactionsQ59234583
Clinical Position of Lacidipine, a New Dihydropyridine Calcium Antagonist, in the Treatment of HypertensionQ67712776
Calcium channel antagonist effects of spironolactone, an aldosterone antagonistQ68463591
P433issue1
P304page(s)95-103
P577publication date2018-11-14
P1433published inAsian Journal of Pharmaceutical SciencesQ50552622
P1476titleCo-amorphous solid dispersion systems of lacidipine-spironolactone with improved dissolution rate and enhanced physical stability
P478volume14

Search more.