review article | Q7318358 |
scholarly article | Q13442814 |
P2093 | author name string | George Varvounis | |
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Identification and synthesis of major metabolites of Vasopressin V2-receptor agonist WAY-151932, and antagonist, Lixivaptan | Q81249679 | ||
Observation of the reversibility of a covalent pyrrolobenzodiazepine (PBD) DNA adduct by HPLC/MS and CD spectroscopy | Q83257464 | ||
Nuclear magnetic resonance solution structures of inter- and intrastrand adducts of DNA cross-linker SJG-136 | Q83848571 | ||
Iridium catalyzed asymmetric hydrogenation of cyclic imines of benzodiazepinones and benzodiazepines | Q84576320 | ||
γ-Turn Mimicry with Benzodiazepinones and Pyrrolobenzodiazepinones Synthesized from a Common Amino Ketone Intermediate | Q85497098 | ||
Intramolecular azide to alkene cycloadditions for the construction of pyrrolobenzodiazepines and azetidino-benzodiazepines | Q85829558 | ||
Mutasynthesis of a potent anticancer sibiromycin analogue | Q36035377 | ||
SG2285, a novel C2-aryl-substituted pyrrolobenzodiazepine dimer prodrug that cross-links DNA and exerts highly potent antitumor activity | Q36496775 | ||
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Effect of hairpin loop structure on reactivity, sequence preference and adduct orientation of a DNA-interactive pyrrolo[2,1-c][1,4]benzodiazepine (PBD) antitumour agent | Q38300702 | ||
The minor groove-binding agent ELB-21 forms multiple interstrand and intrastrand covalent cross-links with duplex DNA and displays potent bactericidal activity against methicillin-resistant Staphylococcus aureus | Q38336785 | ||
DNA Sequence Preference and Adduct Orientation of Pyrrolo[2,1-c][1,4]benzodiazepine Antitumor Agents | Q38339530 | ||
Dithiocarbamate/piperazine bridged pyrrolobenzodiazepines as DNA-minor groove binders: synthesis, DNA-binding affinity and cytotoxic activity | Q38911469 | ||
GC-targeted C8-linked pyrrolobenzodiazepine-biaryl conjugates with femtomolar in vitro cytotoxicity and in vivo antitumor activity in mouse models | Q39178091 | ||
Synthesis, anticancer activity and apoptosis inducing ability of bisindole linked pyrrolo[2,1-c][1,4]benzodiazepine conjugates | Q39439385 | ||
Synthesis and anticancer activity of chalcone-pyrrolobenzodiazepine conjugates linked via 1,2,3-triazole ring side-armed with alkane spacers | Q39523980 | ||
Synthesis and biological evaluation of estradiol linked pyrrolo[2,1-c][1,4]benzodiazepine (PBD) conjugates as potential anticancer agents | Q39565636 | ||
DNA interstrand cross-linking and in vivo antitumor activity of the extended pyrrolo[2,1-c][1,4]benzodiazepine dimer SG2057. | Q39579617 | ||
Hybrids of privileged structures benzothiazoles and pyrrolo[2,1-c] [1,4]benzodiazepin-5-one, and diversity-oriented synthesis of benzothiazoles | Q39653628 | ||
Remarkable enhancement in the DNA-binding ability of C2-fluoro substituted pyrrolo[2,1-c][1,4]benzodiazepines and their anticancer potential | Q39891027 | ||
DC-81-Indole conjugate agent induces mitochondria mediated apoptosis in human melanoma A375 cells | Q40127572 | ||
Design, synthesis, and biophysical and biological evaluation of a series of pyrrolobenzodiazepine-poly(N-methylpyrrole) conjugates | Q40238058 | ||
Effect of base sequence on the DNA cross-linking properties of pyrrolobenzodiazepine (PBD) dimers | Q42063199 | ||
Antistaphylococcal activity of DNA-interactive pyrrolobenzodiazepine (PBD) dimers and PBD-biaryl conjugates. | Q42190109 | ||
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Correction: Interaction of Pyrrolobenzodiazepine (PBD) Ligands with Parallel Intermolecular G-Quadruplex Complex Using Spectroscopy and ESI-MS. | Q46004902 | ||
Boseongazepines A-C, pyrrolobenzodiazepine derivatives from a Streptomyces sp. 11A057. | Q46259712 | ||
Pyrrolo[1,2-a][1,4]benzodiazepine: a novel class of non-azole anti-dermatophyte anti-fungal agents | Q46540927 | ||
Computational studies support the role of the C7-sibirosamine sugar of the pyrrolobenzodiazepine (PBD) sibiromycin in transcription factor inhibition | Q46853969 | ||
Diazepines. 5. Synthesis and biological action of 6-phenyl-4H-pyrrolo[1,2-a][1,4]benzodiazepines | Q48207802 | ||
Pyrrolobenzodiazepines and related systems. 2. Synthesis and biological properties of isonoraptazepine derivatives | Q48405829 | ||
P275 | copyright license | Creative Commons Attribution | Q6905323 |
P6216 | copyright status | copyrighted | Q50423863 |
P433 | issue | 2 | |
P407 | language of work or name | English | Q1860 |
P921 | main subject | antineoplastic | Q2853144 |
pyrrole | Q67954132 | ||
anti-HIV agents | Q50377208 | ||
P304 | page(s) | 154 | |
P577 | publication date | 2016-01-28 | |
P1433 | published in | Molecules | Q151332 |
P1476 | title | An Update on the Synthesis of Pyrrolo[1,4]benzodiazepines | |
P478 | volume | 21 |