Opiate Analgesia: Evidence for Mediation by a Subpopulation of Opiate Receptors

scientific article published on May 2, 1980

Opiate Analgesia: Evidence for Mediation by a Subpopulation of Opiate Receptors is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1126/SCIENCE.6245448
P953full work available at URLhttps://syndication.highwire.org/content/doi/10.1126/science.6245448
P698PubMed publication ID6245448

P50authorGavril W. PasternakQ92217073
P2093author name stringS. H. Snyder
S. R. Childers
P2860cites workJournal of Pharmacology and Experimental TherapeuticsQ1500272
6.beta.-[N,N-Bis(2-chloroethyl)amino]-17-(cyclopropylmethyl)-4,5.alpha.-epoxy-3,14-dihydroxymorphinan (chloranaltrexamine), a potent opioid receptor alkylating agent with ultralong narcotic antagonist activityQ34141607
Chloroxymorphamine, an Opioid Receptor Site-Directed Alkylating Agent Having Narcotic Agonist ActivityQ34377850
Endogenous opioid peptides: multiple agonists and receptorsQ34986433
Differentiation of opiate agonist and antagonist receptor binding by protein modifying reagentsQ39313497
Identification of novel high affinity opiate receptor binding in rat brainQ48476166
Long-acting opiate agonists and antagonists: 14-hydroxydihydromorphinone hydrazonesQ72612035
P433issue4443
P407language of work or nameEnglishQ1860
P304page(s)514-516
P577publication date1980-05-01
1980-05-02
P1433published inScienceQ192864
P1476titleOpiate analgesia: evidence for mediation by a subpopulation of opiate receptors
Opiate Analgesia: Evidence for Mediation by a Subpopulation of Opiate Receptors
P478volume208

Reverse relations

cites work (P2860)
Q3416993114-Methoxymetopon, a very potent mu-opioid receptor-selective analgesic with an unusual pharmacological profile
Q39158190A "tail" of opioid receptor variants.
Q44330554A comparative study in rats of the respiratory depression and analgesia induced by μ- and δ-opioid agonists
Q72913920ACTH-induced grooming involves high-affinity opiate receptors
Q48536754Actions of opioids on respiratory activity via activation of brainstem mu-, delta- and kappa-receptors; an in vitro study
Q49108187Alterations of synaptic high and low affinity opiate binding sites after acute and chronic morphine administration in mice
Q71809737Analgesic and immunomodulatory effects of codeine and codeine 6-glucuronide
Q35563397Anatomy and physiology of chronic pain
Q68753976Antagonism of morphine analgesia by nonopioid cold-water swim analgesia: direct evidence for collateral inhibition
Q44334055Antisense mapping the MOR‐1 opioid receptor: evidence for alternative splicing and a novel morphine‐6β‐glucuronide receptor
Q73190576Antisense mapping: assessing functional significance of genes and splice variants
Q44275456CJ-15,208, a novel kappa opioid receptor antagonist from a fungus, Ctenomyces serratus ATCC15502.
Q48094185Cardiovascular and renal responses produced by central orphanin FQ/nociceptin occur independent of renal nerves
Q48643732Cardiovascular responses to microinjections of endomorphin-2 into the nucleus of the solitary tract are attenuated in the spontaneously hypertensive rat.
Q36374248Classification of multiple morphine and enkephalin binding sites in the central nervous system
Q34675455Clinical features and management of intoxication due to hallucinogenic drugs
Q79991386Codeine and 6-acetylcodeine analgesia in mice
Q40853885Comparative immunohistochemical distributions of carboxy terminus epitopes from the mu-opioid receptor splice variants MOR-1D, MOR-1 and MOR-1C in the mouse and rat CNS.
Q34253888Cross-tolerance studies distinguish morphine- and metkephamid-induced analgesia
Q37170275Development of delta opioid peptides as nonaddicting analgesics
Q52297184Developmental differences between high and low affinity opiate binding sites: Their relationship to analgesia and respiratory depression
Q44333400Differential involvement of mu(1)-opioid receptors in endomorphin- and beta-endorphin-induced G-protein activation in the mouse pons/medulla
Q44345097Differential sensitivity of opioid-induced feeding to naloxone and naloxonazine
Q36412585Differentiation of delta and mu opiate receptor localizations by light microscopic autoradiography
Q72880466Differentiation of opiate receptors in the brain by the selective development of tolerance
Q43921681Effects of adrenoceptor agonists and antagonists on morphine-induced Straub tail in mice
Q42452233Effects of clozapine on the delta- and kappa-opioid receptors and the G-protein-activated K+ (GIRK) channel expressed in Xenopus oocytes
Q41533628Electrophysiological support in favor of multiple opiate receptors in the caudate and the central gray of the rat
Q40085590Endogenous opiates: 1980
Q44352723Endogenous opioid systems in brain
Q42537695Endomorphins fully activate a cloned human mu opioid receptor
Q28295151Erinacine E as a kappa opioid receptor agonist and its new analogs from a basidiomycete, Hericium ramosum
Q33950375Generation of the mu opioid receptor (MOR-1) protein by three new splice variants of the Oprm gene
Q44344657Genetic analysis of the murine mu opioid receptor: increased complexity of Oprm gene splicing
Q47934009Genetic dissociation of morphine analgesia from hyperalgesia in mice
Q34671312Identification and characterization of seven new exon 11-associated splice variants of the rat μ opioid receptor gene, OPRM1.
Q44330378Isolation and expression of a novel alternatively spliced mu opioid receptor isoform, MOR-1F.
Q52275773Kinetic behavior of a receptor-enzyme system: a model for drug addiction.
Q34253970Metkephamid (Tyr-D-Ala-Gly-Phe-N(Me)Met-NH2), a potent opioid peptide: Receptor binding and analgesic properties
Q44341747Micro1-opioid antagonist naloxonazine alters ethanol discrimination and consumption
Q38331826Modification of phosphorothioate oligonucleotides yields potent analogs with minimal toxicity for antisense experiments in the CNS.
Q41550189Morphiceptin (NH 4 -Tyr-Pro-Phe-Pro-COHN 2 ): a Potent and Specific Agonist for Morphine (μ) Receptors
Q70774870Morphine differentially affects ventral tegmental and substantia nigra brain reward thresholds
Q33581970Mu opioid receptors in pain management
Q37236111Mu opioids and their receptors: evolution of a concept
Q40123055Multiple Neurotransmitter Receptors
Q24613589Multiple opiate receptors: [3H]ethylketocyclazocine receptor binding and ketocyclazocine analgesia
Q72903604Naloxazone irreversibly inhibits the high affinity binding of [125I]D-ala2-D-leu5-enkephalin
Q42246481Naloxozone pretreatment modifies cardiorespiratory, temperature, and behavioral effects of morphine
Q42391159New advances in analgesic and anxiolytic agents: implications for continued support of basic research
Q44352975Ontogeny of opioid pharmacology and receptors: High and low affinity site differences
Q48941537Opiate Receptors from Different Tissue Sources: Solubilization and Characterization
Q44353157Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity
Q72912832Opiates and enkephalins: A common binding site mediates their analgesic actions in rats
Q34250337Oxymorphazone: A long-acting opiate analgesic
Q62028952Perioperative anxiety: psychobiology and effects in postoperative recovery
Q34125112Pharmacologic characterization in the rat of a potent analgesic lacking respiratory depression, IBNtxA.
Q52591971Pharmacological Characterization of Levorphanol, a G-Protein Biased Opioid Analgesic.
Q69848797Quantitative autoradiographic distribution of meptazinol-sensitive binding sites in rat brain
Q48459094Quantitative autoradiography of the development of mu opiate binding sites in rat brain
Q28262450Receptor binding and analgesic properties of oxymorphazone
Q38254516Site and mechanism of morphine tolerance in the gastrointestinal tract
Q53816815Site of action of intrathecal morphine.
Q44353442Spinal and supraspinal opioid analgesia in the mouse: the role of subpopulations of opioid binding sites
Q72920302Spinal and supraspinal sites for morphine and nefopam analgesia in the mouse
Q37693807Spinal endomorphin 2 antinociception and the mechanisms that produce it are both sex- and stage of estrus cycle-dependent in rats.
Q34948489The N-terminally truncated µ3 and µ3-like opioid receptors are transcribed from a novel promoter upstream of exon 2 in the human OPRM1 gene
Q72903597The actions of naloxazone on the binding and analgesic properties of morphiceptin (NH2 Tyr-Pro-Phe-Pro-CONH2), a selective mu-receptor ligand
Q24541287The analgesic activity of morphine-6-glucuronide
Q70217521The effects of chronic naloxone on pituitary hormone secretion in female rats
Q34333349The pharmacology of mu analgesics: from patients to genes
Q40088281The practical use of narcotic analgesics
Q52295955Threshold differences for naloxone and naltrexone in the hypothalamus and midbrain using fixed ratio brain self-stimulation in rats.
Q72878937μ- and δ-opiate receptors: Correlation with high and low affinity opiate binding sites

Search more.