Evidence that methyl arachidonyl fluorophosphonate is an irreversible cannabinoid receptor antagonist

scientific article

Evidence that methyl arachidonyl fluorophosphonate is an irreversible cannabinoid receptor antagonist is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1038/SJ.BJP.0701303
P932PMC publication ID1564861
P698PubMed publication ID9283708
P5875ResearchGate publication ID13936652

P50authorRoger PertweeQ29643420
P2093author name stringS R Fernando
P2860cites work(R)-methanandamide: a chiral novel anandamide possessing higher potency and metabolic stabilityQ28244400
Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amidesQ28295481
Methyl arachidonyl fluorophosphonate: a potent irreversible inhibitor of anandamide amidaseQ28305612
SR141716A, a potent and selective antagonist of the brain cannabinoid receptorQ34332716
Factors influencing the release of acetylcholine from the myenteric plexus of the ileum of the guinea-pig and rabbitQ35177860
Inhibitory effects of certain enantiomeric cannabinoids in the mouse vas deferens and the myenteric plexus preparation of guinea-pig small intestineQ35872513
Further evidence for the presence of cannabinoid CB1 receptors in guinea-pig small intestineQ35874121
Functional identification of the active-site nucleophile of the human 85-kDa cytosolic phospholipase A2.Q41214023
Effect of phenylmethylsulphonyl fluoride on the potency of anandamide as an inhibitor of electrically evoked contractions in two isolated tissue preparationsQ46551529
The origin of acetylcholine released from guinea-pig intestine and longitudinal muscle strips.Q52754983
P433issue8
P407language of work or nameEnglishQ1860
P921main subjectcannabinoid receptorQ421237
cannabinoidsQ422936
CNR2Q17907844
P304page(s)1716-1720
P577publication date1997-08-01
P1433published inBritish Journal of PharmacologyQ919631
P1476titleEvidence that methyl arachidonyl fluorophosphonate is an irreversible cannabinoid receptor antagonist
P478volume121

Reverse relations

cites work (P2860)
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Q44618356Inhibition of Platelet-Activating Factor (PAF) Acetylhydrolase by Methyl Arachidonyl Fluorophosphonate Potentiates PAF Synthesis in Thrombin-Stimulated Human Coronary Artery Endothelial Cells
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Q33644120α-Ketoheterocycle inhibitors of fatty acid amide hydrolase: exploration of conformational constraints in the acyl side chain

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