scholarly article | Q13442814 |
P50 | author | Kenji Maeda | Q55153732 |
P2093 | author name string | Hiroaki Mitsuya | |
Arun K Ghosh | |||
Yasuhiro Hayashi | |||
Debananda Das | |||
Darshan V Desai | |||
Simon B Chang | |||
Navnath Gavande | |||
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Molecular mechanism of action of monocyclam versus bicyclam non-peptide antagonists in the CXCR4 chemokine receptor | Q30832371 | ||
Molecular interactions of cyclam and bicyclam non-peptide antagonists with the CXCR4 chemokine receptor | Q31821860 | ||
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Isolation of a new human retrovirus from West African patients with AIDS. | Q34038984 | ||
Structural and molecular interactions of CCR5 inhibitors with CCR5. | Q34494226 | ||
Novel HIV-1 protease inhibitors (PIs) containing a bicyclic P2 functional moiety, tetrahydropyrano-tetrahydrofuran, that are potent against multi-PI-resistant HIV-1 variants | Q34737640 | ||
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GluVII:06--a highly conserved and selective anchor point for non-peptide ligands in chemokine receptors | Q36570350 | ||
Potent synergistic anti-human immunodeficiency virus (HIV) effects using combinations of the CCR5 inhibitor aplaviroc with other anti-HIV drugs | Q36703042 | ||
Involvement of the second extracellular loop and transmembrane residues of CCR5 in inhibitor binding and HIV-1 fusion: insights into the mechanism of allosteric inhibition. | Q37071732 | ||
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Blockade of X4-tropic HIV-1 cellular entry by GSK812397, a potent noncompetitive CXCR4 receptor antagonist | Q39104422 | ||
Novel low molecular weight spirodiketopiperazine derivatives potently inhibit R5 HIV-1 infection through their antagonistic effects on CCR5. | Q39202247 | ||
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Orally bioavailable isothioureas block function of the chemokine receptor CXCR4 in vitro and in vivo | Q39521135 | ||
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Indicator cell lines for detection of primary strains of human and simian immunodeficiency viruses | Q41104028 | ||
Identification of residues of CXCR4 critical for human immunodeficiency virus coreceptor and chemokine receptor activities | Q45742231 | ||
The different ways through which specificity works in orthosteric and allosteric drugs | Q47577552 | ||
Comparison of Shape-Matching and Docking as Virtual Screening Tools | Q56853909 | ||
Critical Role for the Second Extracellular Loop in the Binding of Both Orthosteric and Allosteric G Protein-coupled Receptor Ligands | Q57838214 | ||
Azamacrocyclic metal complexes as CXCR4 antagonists | Q83396529 | ||
P433 | issue | 4 | |
P407 | language of work or name | English | Q1860 |
P304 | page(s) | 1895-1904 | |
P577 | publication date | 2015-01-12 | |
P1433 | published in | Antimicrobial Agents and Chemotherapy | Q578004 |
P1476 | title | Insights into the mechanism of inhibition of CXCR4: identification of Piperidinylethanamine analogs as anti-HIV-1 inhibitors | |
P478 | volume | 59 |
Q64082901 | Activity and structural analysis of GRL-117C: a novel small molecule CCR5 inhibitor active against R5-tropic HIV-1s |
Q56700832 | Advances in the Development of Shape Similarity Methods and Their Application in Drug Discovery |
Q45325496 | Chemokines and Chemokine Receptors: Accomplices for Human Immunodeficiency Virus Infection and Latency |
Q36212626 | Development of CXCR4 modulators by virtual HTS of a novel amide-sulfamide compound library |
Q27468774 | Membrane-associated GRP78 helps subgroup J avian leucosis virus enter cells |
Q50870345 | Novel anti-inflammatory agents targeting CXCR4: Design, synthesis, biological evaluation and preliminary pharmacokinetic study. |
Q34550666 | Structural Analysis of Chemokine Receptor-Ligand Interactions |
Q39766459 | Symmetrical bis-tertiary amines as novel CXCR4 inhibitors |
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