Synthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L.

scientific article published on 25 September 2015

Synthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/J.BMC.2015.09.036
P932PMC publication ID4824049
P698PubMed publication ID26462052

P50authorDhivya R SudhanQ85954937
Erica N ParkerQ86476571
Kevin G. PinneyQ39948043
Michael R. HorsmanQ47792821
P2093author name stringAmanda K Charlton-Sevcik
David J Chaplin
G D Kishore Kumar
Gustavo E Chavarria
Mary Lynn Trawick
Tracy E Strecker
Jiangli Song
Dietmar W Siemann
Thomas R Wittenborn
Samuel O Odutola
Ashleigh L Barnes
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P433issue21
P407language of work or nameEnglishQ1860
P304page(s)6974-6992
P577publication date2015-09-25
P1433published inBioorganic & Medicinal ChemistryQ2904200
P1476titleSynthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L
P478volume23

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cites work (P2860)
Q89634052A Review of Small Molecule Inhibitors and Functional Probes of Human Cathepsin L
Q92702993A Review of the Structure-Activity Relationship of Natural and Synthetic Antimetastatic Compounds
Q90355647Cathepsin L secretion by host and neoplastic cells potentiates invasion
Q48332154Hydrazone Derivatives Enhance Antileishmanial Activity of Thiochroman-4-ones.

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