Structure based development of novel specific inhibitors for cathepsin L and cathepsin S in vitro and in vivo

scientific article published on 01 September 1999

Structure based development of novel specific inhibitors for cathepsin L and cathepsin S in vitro and in vivo is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0014-5793(99)01107-2
P698PubMed publication ID10518923

P50authorHideaki TsugeQ46648414
P2093author name stringV Turk
D Turk
N Katunuma
A Matsui
M Fukushima
H Tsuzuki
Y Tada
E Murata
T Asao
H Kakegawa
P2860cites workMolecular cloning of human cDNA for cathepsin K: novel cysteine proteinase predominantly expressed in boneQ24309351
The refined 2.15 A X-ray crystal structure of human liver cathepsin B: the structural basis for its specificityQ27651464
Crystal structure of cathepsin B inhibited with CA030 at 2.0-A resolution: A basis for the design of specific epoxysuccinyl inhibitorsQ27730182
Crystal structure of human cathepsin K complexed with a potent inhibitorQ27734780
Crystal structure of human osteoclast cathepsin K complex with E-64Q27734783
Binding of chloromethyl ketone substrate analogues to crystalline papainQ27749019
The crystal structure of human cathepsin L complexed with E-64Q28237390
Cathepsin B, Cathepsin H, and cathepsin LQ28277583
Proteolytic activity of human osteoclast cathepsin K. Expression, purification, activation, and substrate identificationQ28280533
Crystal structure of a papain-E-64 complexQ34524433
Purification and characterization of cathepsin J from rat liverQ46117343
Molecular cloning and sequencing of cDNA for rat cathepsin L.Q48336760
Folding and activation of human procathepsin S from inclusion bodies produced in Escherichia coli.Q52519243
Amino acid sequence of rat liver cathepsin LQ68466403
Novel epoxysuccinyl peptides. Selective inhibitors of cathepsin B, in vitroQ70136099
Novel epoxysuccinyl peptides. A selective inhibitor of cathepsin B, in vivoQ70136102
37 Structure, properties, mechanisms, and assays ofcysteine protease inhibitors: Cystatins and E-64 derivativesQ71999767
Specific assay method for the activities of cathepsin L-type cysteine proteinasesQ72411002
P433issue1
P304page(s)6-10
P577publication date1999-09-01
P1433published inFEBS LettersQ1388051
P1476titleStructure based development of novel specific inhibitors for cathepsin L and cathepsin S in vitro and in vivo
P478volume458

Reverse relations

cites work (P2860)
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