Novel epoxysuccinyl peptides. Selective inhibitors of cathepsin B, in vitro

scientific article published on 01 March 1991

Novel epoxysuccinyl peptides. Selective inhibitors of cathepsin B, in vitro is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/0014-5793(91)80318-W
P698PubMed publication ID2013328

P2093author name stringM Murata
S Miyashita
N Katunuma
T Towatari
K Hanada
M Tamai
K Hatayama
C Yokoo
T Nikawa
P2860cites workL-trans-Epoxysuccinyl-leucylamido(4-guanidino)butane (E-64) and its analogues as inhibitors of cysteine proteinases including cathepsins B, H and LQ24531160
Cathepsin B, Cathepsin H, and cathepsin LQ28277583
Crystal structure of a papain-E-64 complexQ34524433
Studies of a calcium-activated neutral protease from chicken skeletal muscle. I. Purification and characterizationQ39208753
Purification and Properties of a New Cathepsin from Rat Liver1Q39222386
Action of rat liver cathepsin L on collagen and other substratesQ42167985
Elastinolytic activity of human cathepsin L.Q42867583
Crystallization and amino acid composition of cathepsin B from rat liver lysosomesQ44795805
Mode of binding of E-64-c, a potent thiol protease inhibitor, to papain as determined by X-ray crystal analysis of the complexQ69963173
Novel epoxysuccinyl peptides. A selective inhibitor of cathepsin B, in vivoQ70136102
In vitro and in vivo inhibition of cysteine proteinases by EST, a new analog of E-64Q70154545
Inhibitions of cathepsin B and cathepsin L by E-64 in vivo. II. Incorporation of [3H]E-64 into rat liver lysosomes in vivoQ70402950
Papain inhibitions by optically active E-64 analogsQ70945463
Inhibitions by E-64 derivatives of rat liver cathepsin B and cathepsin L in vitro and in vivoQ71479486
Inhibition of epoxide derivatives on chicken calcium-activated neutral protease (CANP) in vitro and in vivoQ72127659
P433issue2
P407language of work or nameEnglishQ1860
P304page(s)307-310
P577publication date1991-03-01
P1433published inFEBS LettersQ1388051
P1476titleNovel epoxysuccinyl peptides. Selective inhibitors of cathepsin B, in vitro
P478volume280

Reverse relations

cites work (P2860)
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