The insecticide fipronil and its metabolite fipronil sulphone inhibit the rat alpha1beta2gamma2L GABA(A) receptor

scientific article published on 28 July 2008

The insecticide fipronil and its metabolite fipronil sulphone inhibit the rat alpha1beta2gamma2L GABA(A) receptor is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1038/BJP.2008.309
P932PMC publication ID2584928
P698PubMed publication ID18660823
P5875ResearchGate publication ID51431659

P2093author name stringP Li
G Akk
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Ethanol modulates the interaction of the endogenous neurosteroid allopregnanolone with the alpha1beta2gamma2L GABAA receptorQ48643666
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Dual potentiating and inhibitory actions of a benz[e]indene neurosteroid analog on recombinant alpha1beta2gamma2 GABAA receptorsQ50114260
Local and global ligand-induced changes in the structure of the GABA(A) receptor.Q50648350
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Acute human self-poisoning with the N-phenylpyrazole insecticide fipronil--a GABAA-gated chloride channel blockerQ34313293
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Neuroactive steroids have multiple actions to potentiate GABAA receptorsQ40555555
Effects of gamma2S subunit incorporation on GABAA receptor macroscopic kineticsQ40645605
Which GABAA-receptor subtypes really occur in the brain?Q41003268
Pharmacological and physiological characterization of murine homomeric beta3 GABA(A) receptorsQ41065249
Endogenous subunits can cause ambiguities in the pharmacology of exogenous gamma-aminobutyric acidA receptors expressed in human embryonic kidney 293 cellsQ41163217
Actions of the insecticide fipronil, on dieldrin‐sensitive and ‐resistant GABA receptors of Drosophila melanogasterQ42708156
Unique insecticide specificity of human homomeric rho 1 GABA(C) receptorQ43906479
P433issue5
P407language of work or nameEnglishQ1860
P921main subjectinsecticideQ181322
P304page(s)783-794
P577publication date2008-07-28
P1433published inBritish Journal of PharmacologyQ919631
P1476titleThe insecticide fipronil and its metabolite fipronil sulphone inhibit the rat alpha1beta2gamma2L GABA(A) receptor
P478volume155

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cites work (P2860)
Q27308741A Recombinant Human Pluripotent Stem Cell Line Stably Expressing Halide-Sensitive YFP-I152L for GABAAR and GlyR-Targeted High-Throughput Drug Screening and Toxicity Testing
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Q35531843Synaptic-type α1β2γ2L GABAA receptors produce large persistent currents in the presence of ambient GABA and anesthetic drugs
Q24656617The local anaesthetics proadifen and adiphenine inhibit nicotinic receptors by different molecular mechanisms
Q36199211The pharmacological profile of ELIC, a prokaryotic GABA-gated receptor

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