| scholarly article | Q13442814 |
| P50 | author | Myles H. Akabas | Q42684151 |
| P2093 | author name string | Moez Bali | |
| P2860 | cites work | Structure and gating mechanism of the acetylcholine receptor pore | Q27641514 |
| Refined structure of the nicotinic acetylcholine receptor at 4A resolution | Q28306592 | ||
| A unique amino acid of the Drosophila GABA receptor with influence on drug sensitivity by two mechanisms | Q28367616 | ||
| Mechanisms of channel gating of the ligand-gated ion channel superfamily inferred from protein structure. | Q30341434 | ||
| Structural determinants of fast desensitization and desensitization-deactivation coupling in GABAa receptors. | Q31839971 | ||
| A single amino acid in gamma-aminobutyric acid rho 1 receptors affects competitive and noncompetitive components of picrotoxin inhibition | Q33720641 | ||
| Interaction of picrotoxin with GABAA receptor channel-lining residues probed in cysteine mutants. | Q34047528 | ||
| Pore conformations and gating mechanism of a Cys-loop receptor | Q34116031 | ||
| Gamma-aminobutyric acid increases the water accessibility of M3 membrane-spanning segment residues in gamma-aminobutyric acid type A receptors | Q34171714 | ||
| Minimal structural rearrangement of the cytoplasmic pore during activation of the 5-HT3A receptor | Q34319244 | ||
| An energy-efficient gating mechanism in the acetylcholine receptor channel suggested by molecular and Brownian dynamics | Q34353204 | ||
| A point mutation in a Drosophila GABA receptor confers insecticide resistance. | Q34356098 | ||
| GABAA receptor structure-function studies: a reexamination in light of new acetylcholine receptor structures | Q34365717 | ||
| Emerging structure of the nicotinic acetylcholine receptors | Q34522883 | ||
| Picrotoxin-like channel blockers of GABAA receptors | Q34597191 | ||
| Acetylcholine receptor channel structure in the resting, open, and desensitized states probed with the substituted-cysteine-accessibility method | Q34657454 | ||
| The beta-lactam antibiotics, penicillin-G and cefoselis have different mechanisms and sites of action at GABA(A) receptors | Q35044055 | ||
| Life at the top: the transition state of AChR gating | Q35161669 | ||
| Cys-loop receptors: new twists and turns | Q35785730 | ||
| Convulsant doses of penicillin shorten the lifetime of GABA-induced channels in cultured central neurones | Q35887135 | ||
| Block of muscle nicotinic receptors by choline suggests that the activation and desensitization gates act as distinct molecular entities | Q36295744 | ||
| Trapping of organic blockers by closing of voltage-dependent K+ channels: evidence for a trap door mechanism of activation gating. | Q36411850 | ||
| State-dependent accessibility and electrostatic potential in the channel of the acetylcholine receptor. Inferences from rates of reaction of thiosulfonates with substituted cysteines in the M2 segment of the alpha subunit | Q36412074 | ||
| Identification of channel-lining residues in the M2 membrane-spanning segment of the GABA(A) receptor alpha1 subunit | Q36415753 | ||
| Desensitization of mouse nicotinic acetylcholine receptor channels. A two-gate mechanism | Q36852265 | ||
| Allosteric transitions of the acetylcholine receptor probed at the amino acid level with a photolabile cholinergic ligand | Q37529696 | ||
| Genetic manipulation of ion channels: a new approach to structure and mechanism | Q38211954 | ||
| Local anaesthetics transiently block currents through single acetylcholine-receptor channels | Q40676934 | ||
| Desensitization mechanism of GABA receptors revealed by single oocyte binding and receptor function. | Q40704823 | ||
| Interaction of Tetraethylammonium Ion Derivatives with the Potassium Channels of Giant Axons | Q41761074 | ||
| Dual mechanisms of GABAA response inhibition by beta-lactam antibiotics in the pyramidal neurones of the rat cerebral cortex | Q42040871 | ||
| Subunit composition determines picrotoxin and bicuculline sensitivity of Drosophila gamma-aminobutyric acid receptors. | Q42065545 | ||
| Loose protein packing around the extracellular half of the GABA(A) receptor beta1 subunit M2 channel-lining segment | Q42616990 | ||
| Mutations in the channel domain alter desensitization of a neuronal nicotinic receptor | Q42617071 | ||
| Structural and electrostatic properties of the 5-HT3 receptor pore revealed by substituted cysteine accessibility mutagenesis. | Q42659707 | ||
| Evidence for a centrally located gate in the pore of a serotonin-gated ion channel. | Q42671582 | ||
| Contribution of the beta subunit M2 segment to the ion-conducting pathway of the acetylcholine receptor | Q42678441 | ||
| Rings of negatively charged amino acids determine the acetylcholine receptor channel conductance | Q43509560 | ||
| Mapping the lipid-exposed regions in the Torpedo californica nicotinic acetylcholine receptor | Q43509856 | ||
| Two novel residues in M2 of the gamma-aminobutyric acid type A receptor affecting gating by GABA and picrotoxin affinity. | Q43511697 | ||
| Evidence for distinct conformations of the two alpha 1 subunits in diazepam-bound GABA(A) receptors | Q43757149 | ||
| Evidence that the M2 membrane-spanning region lines the ion channel pore of the nicotinic receptor | Q43866558 | ||
| GABA(A) receptor M2-M3 loop secondary structure and changes in accessibility during channel gating. | Q44133863 | ||
| Site-specific fluorescence reveals distinct structural changes with GABA receptor activation and antagonism | Q44170924 | ||
| Gating-enhanced accessibility of hydrophobic sites within the transmembrane region of the nicotinic acetylcholine receptor's {delta}-subunit. A time-resolved photolabeling study | Q45234380 | ||
| The α7 nicotinic acetylcholine receptor: molecular modelling, electrostatics, and energetics. | Q46646720 | ||
| The location of the gate in the acetylcholine receptor channel | Q47877077 | ||
| How quickly can GABAA receptors open? | Q48196098 | ||
| Multiple mechanisms of picrotoxin block of GABA-induced currents in rat hippocampal neurons | Q48297581 | ||
| Point mutations in the M2 region of the alpha, beta, or gamma subunit of the GABAA channel that abolish block by picrotoxin | Q49071081 | ||
| Identification of acetylcholine receptor channel-lining residues in the entire M2 segment of the alpha subunit | Q49088255 | ||
| Local and global ligand-induced changes in the structure of the GABA(A) receptor. | Q50648350 | ||
| Benzodiazepines induce a conformational change in the region of the gamma-aminobutyric acid type A receptor alpha(1)-subunit M3 membrane-spanning segment. | Q50722415 | ||
| Desensitized states prolong GABAA channel responses to brief agonist pulses. | Q54007822 | ||
| Kinetics of open channel block by penicillin of single GABAA receptor channels from mouse spinal cord neurones in culture | Q54070900 | ||
| On the mechanism of action of picrotoxin on GABA receptor channels in dissociated sympathetic neurones of the rat. | Q55036933 | ||
| Agonist-induced changes in the structure of the acetylcholine receptor M2 regions revealed by photoincorporation of an uncharged nicotinic noncompetitive antagonist | Q68225987 | ||
| Desensitization of the nicotinic acetylcholine receptor mainly involves a structural change in solvent-accessible regions of the polypeptide backbone | Q73299152 | ||
| Desensitization characteristics of rat recombinant GABA(A) receptors consisting of alpha1beta2gamma2S and alpha1beta2 subunits expressed in HEK293 cells | Q73374903 | ||
| P433 | issue | 2 | |
| P304 | page(s) | 145-159 | |
| P577 | publication date | 2007-01-16 | |
| P1433 | published in | The Journal of General Physiology | Q1092259 |
| P1476 | title | The location of a closed channel gate in the GABAA receptor channel | |
| P478 | volume | 129 |
| Q35238474 | 5-HT3 receptor ion size selectivity is a property of the transmembrane channel, not the cytoplasmic vestibule portals. |
| Q37954719 | A novel GABA(A) receptor pharmacology: drugs interacting with the α(+) β(-) interface |
| Q42603484 | Agonist- and antagonist-induced conformational changes of loop F and their contributions to the rho1 GABA receptor function |
| Q28245066 | Allosteric activation mechanism of the cys-loop receptors |
| Q36533714 | Assessment of subunit-dependent direct gating and allosteric modulatory effects of carisoprodol at GABA(A) receptors |
| Q37649162 | Atomic structure and dynamics of pentameric ligand-gated ion channels: new insight from bacterial homologues. |
| Q35080454 | Binding sites for bilobalide, diltiazem, ginkgolide, and picrotoxinin at the 5-HT3 receptor |
| Q37382995 | Brain regional distribution of GABA(A) receptors exhibiting atypical GABA agonism: roles of receptor subunits |
| Q36785221 | Bubbles, gating, and anesthetics in ion channels |
| Q63432840 | Cryo-EM structure of the human α1β3γ2 GABA receptor in a lipid bilayer |
| Q38089188 | Discriminating between 5-HT₃A and 5-HT₃AB receptors |
| Q35266466 | Engineering a prokaryotic Cys-loop receptor with a third functional domain |
| Q63432841 | GABA receptor signalling mechanisms revealed by structural pharmacology |
| Q37181047 | GABA-induced intersubunit conformational movement in the GABAA receptor alpha 1M1-beta 2M3 transmembrane subunit interface: experimental basis for homology modeling of an intravenous anesthetic binding site |
| Q36201884 | Gating-induced conformational rearrangement of the γ-aminobutyric acid type A receptor β-α subunit interface in the membrane-spanning domain |
| Q39443162 | Influences on blockade by t-butylbicyclo-phosphoro-thionate of GABA(A) receptor spontaneous gating, agonist activation and desensitization. |
| Q45134796 | Inhibitory effects of insulin on GABAA currents modulated by the GABAA alpha subunit |
| Q36404799 | Modular design of Cys-loop ligand-gated ion channels: functional 5-HT3 and GABA rho1 receptors lacking the large cytoplasmic M3M4 loop |
| Q33623304 | Robust photoregulation of GABA(A) receptors by allosteric modulation with a propofol analogue |
| Q48055229 | Side chain flexibility and the pore dimensions in the GABAA receptor. |
| Q45141518 | String method solution of the gating pathways for a pentameric ligand-gated ion channel. |
| Q34782188 | Structural answers and persistent questions about how nicotinic receptors work |
| Q26852212 | Structure and pharmacology of pentameric receptor channels: from bacteria to brain |
| Q34800089 | Structure of the M2 transmembrane segment of GLIC, a prokaryotic Cys loop receptor homologue from Gloeobacter violaceus, probed by substituted cysteine accessibility. |
| Q37782321 | The Evolution of Pentameric Ligand-Gated Ion Channels |
| Q35795776 | The atypical cation-conduction and gating properties of ELIC underscore the marked functional versatility of the pentameric ligand-gated ion-channel fold. |
| Q39977073 | The desensitization gate of inhibitory Cys-loop receptors. |
| Q30401509 | The dual modulatory effects of efavirenz on GABAA receptors are mediated via two distinct sites |
| Q87892073 | The dual-gate model for pentameric ligand-gated ion channels activation and desensitization |
| Q36977473 | The insecticide fipronil and its metabolite fipronil sulphone inhibit the rat alpha1beta2gamma2L GABA(A) receptor |
| Q37789790 | The structural basis of function in Cys-loop receptors. |
| Q30461963 | Use of the light-dark box to compare the anxiety-related behavior of virgin and postpartum female rats |
| Q37240694 | Using molecular dynamics to elucidate the structural basis for function in pLGICs |
| Q30605151 | X-ray structures of GluCl in apo states reveal a gating mechanism of Cys-loop receptors. |
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