TS-071 is a novel, potent and selective renal sodium-glucose cotransporter 2 (SGLT2) inhibitor with anti-hyperglycaemic activity

scientific article published on September 2011

TS-071 is a novel, potent and selective renal sodium-glucose cotransporter 2 (SGLT2) inhibitor with anti-hyperglycaemic activity is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1111/J.1476-5381.2011.01340.X
P932PMC publication ID3171870
P698PubMed publication ID21410690
P5875ResearchGate publication ID50408288

P2093author name stringK Yamamoto
K Takahashi
N Kojima
T Takahashi
K Kitano
S Uchida
M Arai
H Toyoda
H Tomoike
N Fukuhara
A Kozakai
E Gunji
J Asami
L Okumura-Kitajima
P2860cites workEfficient selection for high-expression transfectants with a novel eukaryotic vectorQ27860810
Renal Na(+)-glucose cotransportersQ28141135
Molecular Analysis of the SGLT2 Gene in Patients with Renal GlucosuriaQ28211392
Molecular basis for glucose-galactose malabsorptionQ28215903
Structure, function, and regulation of the mammalian facilitative glucose transporter gene familyQ28292160
Molecular characteristics of Na(+)-coupled glucose transporters in adult and embryonic rat kidneyQ28580452
The human kidney low affinity Na+/glucose cotransporter SGLT2. Delineation of the major renal reabsorptive mechanism for D-glucoseQ34121476
Human cardiomyocytes express high level of Na+/glucose cotransporter 1 (SGLT1)Q34264473
SGLT2 mediates glucose reabsorption in the early proximal tubule.Q34457264
Oral antihyperglycemic therapy for type 2 diabetes: scientific reviewQ34492673
Sergliflozin, a novel selective inhibitor of low-affinity sodium glucose cotransporter (SGLT2), validates the critical role of SGLT2 in renal glucose reabsorption and modulates plasma glucose levelQ34575066
Molecular physiology of sodium-glucose cotransportersQ34724942
Phlorizin: a reviewQ35995949
Dapagliflozin, a selective SGLT2 inhibitor, improves glucose homeostasis in normal and diabetic ratsQ39999985
Insulin regulation of the two glucose transporters in 3T3-L1 adipocytesQ42831625
(1S)-1,5-anhydro-1-[5-(4-ethoxybenzyl)-2-methoxy-4-methylphenyl]-1-thio-D-glucitol (TS-071) is a potent, selective sodium-dependent glucose cotransporter 2 (SGLT2) inhibitor for type 2 diabetes treatmentQ43123822
Remogliflozin etabonate, in a novel category of selective low-affinity sodium glucose cotransporter (SGLT2) inhibitors, exhibits antidiabetic efficacy in rodent modelsQ46516165
Guide to Receptors and Channels (GRAC), 4th EditionQ56639335
T-1095, an inhibitor of renal Na+-glucose cotransporters, may provide a novel approach to treating diabetesQ78238839
Studies on the diabetogenic action of streptozotocin (NSC-37917)Q94295200
P433issue1
P407language of work or nameEnglishQ1860
P921main subjecthyperglycemiaQ271993
P304page(s)181-191
P577publication date2011-09-01
P1433published inBritish Journal of PharmacologyQ919631
P1476titleTS-071 is a novel, potent and selective renal sodium-glucose cotransporter 2 (SGLT2) inhibitor with anti-hyperglycaemic activity
P478volume164

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cites work (P2860)
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