Analysis of antimalarial synergy between bestatin and endoprotease inhibitors using statistical response-surface modelling

scientific article

Analysis of antimalarial synergy between bestatin and endoprotease inhibitors using statistical response-surface modelling is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1128/AAC.45.11.3175-3181.2001
P932PMC publication ID90800
P698PubMed publication ID11600374

P2093author name stringA Bell
J P Dalton
S G Machado
C S Gavigan
P2860cites workHemoglobin metabolism in the malaria parasite Plasmodium falciparumQ27973732
Synergistic drug combinations in AIDS therapy. Dipyridamole/3'-azido-3'-deoxythymidine in particular and principles of analysis in generalQ28328662
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Order and specificity of the Plasmodium falciparum hemoglobin degradation pathwayQ34139669
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Lecture on the Antagonism between the Actions of Active Substances.Q48582933
Application of a new approach for the quantitation of drug synergism to the combination of cis-diamminedichloroplatinum and 1-beta-D-arabinofuranosylcytosine.Q52473169
Measurement of the Potencies of Drug MixturesQ52507424
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Localization and characterization of hemoglobin-degrading aspartic proteinases from the malarial parasite Plasmodium falciparumQ68017340
Plasmodium falciparum: differential sensitivity in vitro to E-64 (cysteine protease inhibitor) and Pepstatin A (aspartyl protease inhibitor)Q68041234
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The problem of synergism and antagonism of combined drugsQ73248616
Plasmodium chabaudi chabaudi and P. falciparum: inhibition of aminopeptidase and parasite growth by bestatin and nitrobestatinQ77051404
P433issue11
P407language of work or nameEnglishQ1860
P921main subjectstatisticsQ12483
antimalarialQ521616
P304page(s)3175-3181
P577publication date2001-11-01
P1433published inAntimicrobial Agents and ChemotherapyQ578004
P1476titleAnalysis of antimalarial synergy between bestatin and endoprotease inhibitors using statistical response-surface modelling
P478volume45

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cites work (P2860)
Q27671783Bestatin-based chemical biology strategy reveals distinct roles for malaria M1- and M17-family aminopeptidases
Q36870833Chemical target validation studies of aminopeptidase in malaria parasites using alpha-aminoalkylphosphonate and phosphonopeptide inhibitors
Q39017667Overexpression of leucyl aminopeptidase in Plasmodium falciparum parasites. Target for the antimalarial activity of bestatin
Q27653672Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase
Q36018855The aminopeptidase inhibitor CHR-2863 is an orally bioavailable inhibitor of murine malaria
Q47988678The antimalarial action of FK506 and rapamycin: evidence for a direct effect on FK506-binding protein PfFKBP35.

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