Antiacetylcholine Drugs: Chemistry, Stereochemistry, and Pharmacology

scientific article published on January 1, 1974

Antiacetylcholine Drugs: Chemistry, Stereochemistry, and Pharmacology is …
instance of (P31):
scholarly articleQ13442814
review articleQ7318358

External links are
P356DOI10.1016/S0074-7742(08)60195-6
P698PubMed publication ID4606226

P2093author name stringT. D. Inch
R. W. Brimblecombe
P2860cites workClinical Pharmacology & TherapeuticsQ1101529
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Relationships between chemical structure and affinity for acetylcholine receptorsQ41380208
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Some pharmacological properties common to atropine, pethidine, procaine, and quinidineQ42160042
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pA, a new scale for the measurement of drug antagonismQ42367410
THE OCCURRENCE AND DISTRIBUTION OF ATROPINESTERASE, AND THE SPECIFICITY OF TROPINESTERASES.Q42841689
Parabolic dependence of drug action upon lipophilic character as revealed by a study of hypnoticsQ43433424
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The central and peripheral activities of anti-acetylcholine drugs. Some concepts of practical relevanceQ46672813
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The significance of differences in the potency of enantiomers of anti-acetylcholine drugsQ46872562
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Differential anticholinergic activity, metabolism and excretion of the optical isomers of 14C-benzetimide hydrochlorideQ49029243
The Fate of Intracerebroventricular Injection of Atropine and Methylatropine in Relation to their Pharmacological Effects*Q49073672
Distribution and Metabolism of H3-atropine in MiceQ49159698
Behavioural Actions of Anticholinergic DrugsQ51111283
Effects of DFP and obidoxime on brain acetylcholine levels on brain and peripheral cholinesterases.Q51118382
Decreased distribution of oxotremorine to brain after pharmacological blockade of its peripheral acetylcholine-like effects.Q51120483
The Effect of Physostigmine and Atropine on some Behavioral and Electrophysiological Functions in RatsQ51194359
The peripheral and central actions of some anticholinergic substancesQ51196883
The influence of DFP, atropine and pyridinium aldoximes on the rate of clearance of diisopropyl phosphate (DI32P) from the mouse circulatory system.Q51203975
Distribution of DF32P in mouse organs. II. The effect of prophylactically administered oximes and atropine on incorporation and toxicity.Q51227913
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THE IMPORTANCE OF LIPID-SOLUBILITY FOR THE CENTRAL ACTION OF CHOLINOLYTIC DRUGS.Q51249961
TREMORINE AND OXOTREMORINE EFFECTS ON ACETYLCHOLINESTERASE AND CHOLINE ACETYLASE FROM RAT BRAIN.Q51255791
Cholinergic mechanisms in the control of behavior by the brainQ51290127
The effect of drugs on arousal responses produced by electrical stimulation of the reticular formation of the brain.Q51322490
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Structure--activity correlations in the metabolism of drugs.Q53019613
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Structure-activity relations for anticholinergic 2(1-aryl(or cyclohexyl)-1-hydroxy-1-phenyl)methyl-1,3-dioxolansQ68756277
The stereoselectivity of some anti-acetylcholine acetylenic compoundsQ68759709
Analogues and homologues of atropine: anti-acetylcholine activitiesQ68766012
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Effects of several anticholinergic drugs on the post-tetanic potentiation in the phrenic nerve-diaphragm preparation of the ratQ71101263
The effects of scopolamine hydrobromide and methyl scopolamine hydrobromide upon the discrimination of interoceptive and exteroceptive stimuliQ71238555
Atropine metabolism in manQ71427896
Scopolamine effects on go-no go avoidance discriminations: influence of stimulus factors and primacy of trainingQ71511273
Reassignment of the absolute configuration of 3-acetoxyquinuclidine methiodide and the absolute configuration of receptor-bound acetylcholineQ71525016
Interaction of Atropine with the Muscarinic ReceptorQ71580890
Spasmolytics. 3. 3-Tropanyl 2,3-diarylacrylates. A case history of pi-sigma structure-function correlationQ71592775
Contrasting effects of scopolamine on mice trained simultaneously with two different schedules of avoidance conditioningQ71909359
The metabolism and excretion of benzetimide hydrochloride (R 4929) by ratsQ72029448
Central and peripheral anticholinergic potency of some drugs antagonistic to anticholinesterase poisoningQ72084421
Charge-transfer complexes in medicinal chemistry. I. Correlations with the psychotropic activity of piperidinol esters and related compoundsQ72133525
P433issue0
P407language of work or nameEnglishQ1860
P921main subjectpharmacologyQ128406
P304page(s)67-144
P577publication date1974-01-01
P1433published inInternational Review of NeurobiologyQ15754273
P1476titleAntiacetylcholine Drugs: Chemistry, Stereochemistry, and Pharmacology
P478volume16

Reverse relations

cites work (P2860)
Q72506801Acute extrapyramidal side effects: Serum levels of neuroleptics and anticholinergics
Q34334991Adverse central effects of drugs in man: Predictive value of behavioral studies in rodents and primates
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Q36004398Muscarinic receptor occupation and receptor activation in the guinea-pig ileum by some acetamides related to oxotremorine
Q40076893On chiral drug action
Q40149918Pharmacological properties of oxotremorine and its analogs
Q39932016Stereochemical requirements for central and peripheral muscarinic and antimuscarinic activity of some acetylenic compounds related to oxotremorine
Q38931116Structure-activity requirements for hypotension and α-adrenergic receptor blockade by analogues of atropine
Q39169266The central and peripheral effectiveness of two oxotremorine-antagonists determined using oxotremorine-induced tremor and salivation

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