On chiral drug action

scientific article published on July 1, 1984

On chiral drug action is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

External links are
P356DOI10.1002/MED.2610040304
P953full work available at URLhttps://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fmed.2610040304
https://onlinelibrary.wiley.com/doi/full/10.1002/med.2610040304
P698PubMed publication ID6087043
P5875ResearchGate publication ID17099347

P2093author name stringM. Simonyi
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Chronic propranolol treatment decreases cardiac β-adrenoceptors in spontaneously hypertensive ratsQ72929412
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The presence of histamine and acetylcholine in the spleen of the ox and the horseQ80326828
Modulation of GABA binding sites by CNS depressants and CNS convulsantsQ84268741
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Letter: Drug-induced illnessQ93742511
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Pharmacodynamic effects and possible therapeutic uses of THIP, a specific GABA-agonistQ40132011
Effects of the optical isomers of propranolol on neuromuscular transmission in the ratQ40145462
Interaction of barbiturates with dihydropicrotoxinin binding sites related to the GABA receptor-ionophore systemQ40161259
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Is stimulation of benzodiazepine receptor binding mediated by a novel GABA receptor?Q40219716
Benzodiazepines in the elderly.Q40245244
Pindolol--the pharmacology of a partial agonistQ40335577
Determination of the Vacant Amount of High-Affinity Bilirubin Binding Site on Serum AlbuminQ28330549
Plasma binding and the affinity of propranolol for a beta receptor in manQ28333902
The effect of pindolol on plasma renin activity and blood pressure in hypertensive patientsQ28334539
On the transmitter function of 5-hydroxytryptamine at excitatory and inhibitory monosynaptic junctionsQ28362819
Structure and activity of acetylcholineQ29541933
Prediction of creatinine clearance from serum creatinineQ29615603
A NEW ADRENERGIC BETARECEPTOR ANTAGONISTQ33971458
Identification of two related pentapeptides from the brain with potent opiate agonist activityQ34134593
Three acetylcholine receptors inAplysianeuronesQ34216251
Opiate Receptor: Demonstration in Nervous TissueQ34216480
The relevance of β-receptor blockade to ouabain-induced cardiac arrhythmiasQ34239595
(-)Baclofen decreases neurotransmitter release in the mammalian CNS by an action at a novel GABA receptor.Q34251383
3H-baclofen and 3H-GABA bind to bicuculline-insensitive GABAB sites in rat brainQ34252242
PhencyclidineQ34280939
Unaltered serum propranolol binding by meal-induced variations in fatty acidsQ34449997
Renal function, protein binding and pharmacological response to diazoxideQ34515000
Factors affecting drug binding in plasma of elderly patientsQ34515177
A comparison of some physiological and psychological effects of propranolol and diazepam in normal subjectsQ34515265
Bromocriptine and dopamine receptor stimulationQ34515404
Altered distribution of digoxin in renal failure--a cause of digoxin toxicity?Q34515437
Adrenoceptor responsiveness in bronchial asthma: effect of isoprenaline inhalation on plasma cyclic 3',5'-AMP levelsQ34515452
(+)-Propranolol clearance, an estimation of hepatic blood flow in manQ34516519
Kinetics and clinical importance of displacement of warfarin from albumin by acidic drugs.Q34702247
Differentiation of Receptor Systems activated by Sympathomimetic AminesQ34706728
Resolution of DL-Tryptophan by Affinity Chromatography on Bovine-Serum Albumin-Agarose ColumnsQ34737986
Receptors mediating some actions of histamineQ34794929
A study of the adrenotropic receptorsQ34854653
Identification of cardiac beta-adrenergic receptors by (minus) [3H]alprenolol bindingQ35076839
Gamma-aminobutyric acid binding to receptor sites in the rat central nervous system.Q35119680
Stereospecific Binding of Propranolol and Catecholamines to the β-Adrenergic ReceptorQ35129754
Interconverting mu and delta forms of the opiate receptor in rat striatal patchesQ35456112
The beta-adrenergic receptor: rapid purification and covalent labeling by photoaffinity crosslinkingQ36293412
Phencyclidine (angel dust)/sigma "opiate" receptor: visualization by tritium-sensitive filmQ36371090
3HPhencyclidine: a probe for the ionic channel of the nicotinic receptorQ36420038
Elevation of beta-adrenergic receptor density in human lymphocytes after propranolol administrationQ37021810
Changes in γ-aminobutyric acid-shunt enzymes in regions of rat brain with ketamine anaesthesiaQ51867372
Effects of autonomic blockade by methylatropine and optical isomers and propranolol on plasma insulin levels in the basal state and after stimulation.Q51867889
An endogenous substance from porcine brain antagonizes the anticonvulsant effect of diazepam.Q51867997
Comparison of dihydrodiazepam enantiomers: metabolism, serum binding and brain receptor binding.Q51874120
Ketamine-induced changes in the GABA system of mouse brain.Q51874936
Serum protein binding of drugs and bilirubin in newborn infants and their mothers.Q51875546
Increase of myocardial pH by 1- and d-propranolol during ischemia of the heart in dogs.Q51875797
The interaction of ketamine with the opiate receptorQ51877206
Pharmacology of ketamine isomers in surgical patients.Q51877487
Identification of an endogenous peptide-ligand for the benzodiazepine receptor.Q51877908
Benzodiazepines: selective use to avoid addiction.Q52270013
Physostigmine, a highly potent antidote for acute experimental diazepam intoxication.Q52705387
Application of ultrafiltration and CD spectroscopy for studying stereoselective binding of racemic ligands.Q52712538
Mechanism of action of beta-adrenergic receptor blocking agents in angina pectoris: comparison of action of propranolol with dexpropranolol and practolol.Q52744918
Determine rate constants of interaction of steroid receptors with non-labelled ligands.Q52755388
Differences in anaesthetic properties between the optical antipodes of hexobarbital in the ratQ52758001
Kinetics of the hormone-receptor interaction competition experiments with slowly equilibrating ligandsQ52764359
Binding of some fatty acids and drugs to immobilized bovine serum albumin studied by column affinity chromatographyQ52770450
Sernyl (CI-395) in clinical anaesthesia.Q52770612
The dissolution times of spherical particles.Q53724866
Pharmacokinetics of dextro-, laevo- and racemic propranolol in man.Q53750445
Increase of ovarian progesterone secretion by beta 2-adrenergic stimulation in oestrous rats.Q54512048
Regional hemodynamic effects of beta-adrenergic blockade with propranolol in the unanesthetized primateQ54653336
Pharmacokinetics and pharmacodynamics of the enantiomers of warfarin in manQ54693988
Beta-adrenergic blocking agents. I. Pronethalol and related N-alkyl and N-aralkyl derivatives of 2-amino-1-(2-naphythyl)ethanol.Q54789636
Cutaneous and ocular reactions to practolol.Q55109534
Beta-blockers and plasma triglycerides.Q55145583
Spezifikation der molekularen ChiralitätQ56657053
A Specific Sympathomimetic Ergone in Adrenergic Nerve Fibres (Sympathin) and its Relations to Adrenaline and Nor-AdrenalineQ56687597
Interaction of clofibrate with warfarin. I. Effect of clofibrate on the disposition of the optical enantiomorphs of warfarinQ58817421
Muscarinic ReceptorsQ58972468
Selective antagonists of benzodiazepinesQ59057876
The CatecholaminesQ59065158
Ethyl β-carboline-3-carboxylate shows differential benzodiazepine receptor interactionQ59075672
Optical Isomers of PropranololQ59085467
Direct evidence for an interaction of β-adrenergic blockers with the 5-HT receptorQ59095140
Toxicity and Teratogenicity of Optical Isomers of ThalidomideQ59099301
Conformation of histamine derivatives. 5. Molecular orbital calculation of the H1-receptor essential conformation of histamineQ66960051
Resolution of (±)‐PropranololQ66962631
Circular dichroism and gel filtration study of binding of prochiral and chiral 1,4-benzodiazepin-2-ones to human serum albuminQ66970911
Stereospecific plasma binding of gliflumide, a new antidiabetic drugQ67015499
Ritodrine in the treatment of preterm labour. A clinical trial to compare a standard treatment with three regimens involving the use of ritodrineQ67241868
Characterization of the mammalian beta-2 receptor in 8 M ureaQ67242304
The effect of racemic, D-, or L-propranolol and practolol on the response to cold by the newborn rabbitQ67421885
Effect of d- and dl-propranolol on glucose-stimulated insulin releaseQ67467893
Chromatographic separation on phosphocellulose of activated and nonactivated forms of steroid-receptor complex. Purification of the activated complexQ67526231
Absolute configuration of glycerol derivatives.3.1 Synthesis and cupra A circular dichroism spectra of some chiral 3-aryloxy-1,2-propanediols and 3-aryloxy-1-amino-2-propanolsQ67550639
The stereoselective interaction of warfarin and metronidazole in manQ67745717
Studies on the binding of benzodiazepines to human serum albumin by circular dichroism measurementsQ67851436
Effects of d-propranolol and estradiol on the cervicovaginal epitheliumQ67863589
Characterization of the binding of benzodiazepines to human serum albuminQ68522466
Properties of γ-aminobutyric acid (GABA) receptor binding in rat brain synaptic membrane fractionsQ40346759
Warfarin. Stereochemical aspects of its metabolism and the interaction with phenylbutazoneQ40373479
A trial of oral ritodrine for the prevention of premature labourQ40754985
Plasma and tissue protein binding of drugs in pharmacokineticsQ40809296
The inhibitory action of noradrenaline and adrenaline on acetylcholine output by guinea-pig ileum longitudinal muscle stripQ41334304
Effects of racemic, dextro-laevo-propranolol and isoxuprine on the metabolic and endocrine response to cold in the newborn rabbitQ41375847
Further studies on the site of action of diazepam: anticonvulsant effect in the rabbitQ41425150
Studies of the action of nicotine in guinea-pig tracheal smooth muscle: Interaction with β-adrenoceptor antagonistsQ41531252
Effects of age and cigarette smoking on propranolol dispositionQ41617556
Inhibition of [3H]adenosine binding by stereoisomers of oxazepam hemisuccinate in guinea-pig brain synaptosomesQ41625546
Kinetics of the glucocorticoid hormone-receptor interaction. False association constants determined in slowly equilibrating systemsQ41669494
Partial agonists for brain GABA/benzodiazepine receptor complexQ41700518
Warfarin metabolism in man: identification of metabolites in urineQ41710726
Biotransformation and excretion of lorazepam in patients with chronic renal failureQ41787246
Studies on the relationship between chemical constitution and physiological action: Molecular dissymmetry and physiological activityQ41869994
The alpha- and beta-adrenoceptor blocking potencies of labetalol and its individual stereoisomers in anaesthetized dogs and in isolated tissuesQ41893893
Educating doctors to use drugs wellQ42101455
Drug advertising in medical journalsQ42161508
Studies on 1,2,3,4-tetrahydroisoquinolines. IV. .BETA.-Adrenoceptor activity and absolute stereochemistry of (-)-5,7-dihydroxy-1-(3,4,5-trimethoxybenzyl)-1,2,3,4-tetrahydroisoquinolineQ42245764
Stereochemical characterization of interactions of chiral 1,4-benzodiazepine-2-ones with liver microsomesQ42264868
Pirenzepine distinguishes between different subclasses of muscarinic receptorsQ42271324
Factors affecting drug-protein binding in the plasma of newborn infantsQ42407260
The beta-adrenergic system and allergic bronchial asthma: changes in lymphocyte beta-adrenergic receptor number and adenylate cyclase activity after an allergen-induced asthmatic attackQ42452372
Increased plasma propranolol binding in myocardial infarctionQ43244558
Drugs for the Third WorldQ43254537
The effect of end-stage renal failure and haemodialysis on the elimination kinetics of sotalolQ43255348
Preliminary observations on the elimination of acebutolol in severe chronic renal failureQ43256002
Identification of inosine and hypoxanthine as endogenous inhibitors of [3H] diazepam binding in the central nervous systemQ43547275
Differential effects of d- and l-propranolol on dopamine turnover stimulated by oxotremorine in striatal and mesolimbic areas of rat brainQ43785656
Stereospecific benzodiazepine receptor binding by the enantiomers of oxazepam sodium hemisuccinateQ43898694
Dynorphin Is a Specific Endogenous Ligand of the κ Opioid ReceptorQ44352111
Interactions of benzodiazepines with human serum albumin. Circular dichroism studiesQ44363131
Central noradrenergic mechanisms and the cardiovascular effects of intracerebroventricular (+)- and (−)-propranolol in the conscious rabbitQ44369169
Beta-adrenergic blocking agents. 9. Absolute configuration of propranolol and of a number of related aryloxypropanolamines and arylethanolaminesQ44378417
Brain specific benzodiazepine receptorsQ44452528
Absolute configuration and parasympathetic action: pharmacodynamics of enantiomorphic and diastereoisomeric esters of beta-methylcholineQ45022341
Modification by levo-propranolol of tremors induced by harmine in miceQ45095025
Resolution of two biochemically and pharmacologically distinct benzodiazepine receptorsQ45157485
Benzodiazepine receptors in rat brainQ45205253
Evidence favouring the existence of a single adrenergic receptorQ45230922
Protein binding of drugs in uremic and normal serum: the role of endogenous binding inhibitorsQ45286897
Comparison of in vitro potencies in pharmacological and binding assays after inhibition of peptides reveals that dynorphin (1–9) is a potent κ-agonistQ46284848
3H-Codeine binding in the guinea pig lower brain stemQ46344017
Binding characteristics of (+)-, (+/-)- and (-)-[125iodo] cyanopindolol to guinea-pig left ventricle membranesQ46433717
Ketamine alone and combined with diazepam or xylazine in laboratory animals: a 10 year experienceQ46515518
Studies on the stereospecificity of closely related compounds which block postganglionic acetylcholine receptors in the guinea-pig ileumQ46671733
Definition and antagonism of histamine H 2 -receptorsQ46704110
Antihypertensive and adrenergic receptor blocking properties of the enantiomers of medroxalolQ46758288
Two distinct serotonin receptors: regional variations in receptor binding in mammalian brainQ46832632
Presence of a low molecular weight endogenous inhibitor on 3H-muscimol binding in synaptic membranesQ47293923
Pharmacology of cortical inhibitionQ47715638
Binding of psychotropic drugs to isolated alpha-acid glycoproteinQ47777223
Plus and minus-bicuculline methochloride as optical isomers of a GABA antagonistQ47861420
Disposition of propranolol. VI. Independent variation in steady-state circulating drug concentrations and half-life as a result of plasma drug binding in man.Q47980851
Interactions of the Hexobarbital Enantiomers with Rat Liver MicrosomesQ47990443
Stereospecificity of esterases hydrolyzing oxazepam acetateQ48163799
Comparative pharmacology of the optical isomers of ketamine in miceQ48192323
Is there a "hydrophobic effect"?Q37311020
Stimulation of benzodiazepine receptor binding by gamma-aminobutyric acidQ37317413
Glial cell function: uptake of transmitter substancesQ37490801
Competitive inhibition of benzodiazepine binding by fractions from porcine brainQ37597636
Central Actions of Benzodiazepines: General IntroductionQ37826816
Multiple receptors for dopamineQ37876912
Effect of Propranolol on Oxygen Binding to Hemoglobin In Vitro and In VivoQ38361246
Problems with PractololQ39067668
The Role of Renin in the Antihypertensive Action of β-Adrenoreceptor Blocking AgentsQ39097120
(−)-Propranolol inhibits the behavioural responses of rats to increased 5-hydroxytryptamine in the central nervous systemQ39109775
Stereospecificity of interaction of neuroleptic drugs with neurotransmitters and correlation with clinical potencyQ39109812
Simultaneous determination of (–)- and (+)- propranolol by gas chromatography-mass spectrometry using a deuterium labeling techniqueQ39122875
The influence of plasma protein binding on distribution and pharmacological activity of tranquilizers of the benzodiazepine group (author's transl)Q39132506
A functional basis for classification of α-adrenergic receptorsQ39165904
High densities of benzodiazepine receptors in human cortical areasQ39176727
Biochemical identification of the site of action of benzodiazepines in human brain by 3H-diazepam bindingQ39189130
Is the hypotensive effect obtained by application of drugs to the ventral surface of the brain stem due to a membrane stabilizing mechanism? A study with beta-blockersQ39209860
Reduced β-adrenoceptor sensitivity in the elderlyQ39256290
Antagonism by propranolol of central dopamine receptor stimulation is not related to β-adrenergic blockadeQ39258107
The anticonvulsant action of the (−)- and (+)-enantiomers of propranololQ39264852
Fundamental difference between the molecular interactions of agonists and antagonists with the β-adrenergic receptorQ39265422
Studies on the structure-activity relationships of adrenergic .BETA.-mimetic benzylamine derivatives. V. 9-Aryl-1H-2,3,7,8,9,10-hexahydrobenzo[d,e]quinolinesQ39268558
Anti-anxiety action op diazepam after intraamygdaloid application in the ratQ39271094
Use of Serum Creatinine Concentrations to Determine Renal Function1Q39806214
Comparative studies of (--)-, (+/-)-propranolol, atenolol, guanethidine, bretylium and tetracaine on adrenergic transmissionQ39930439
Antiacetylcholine Drugs: Chemistry, Stereochemistry, and PharmacologyQ39945613
Presynaptic regulation of catecholamine releaseQ39953110
Hormone Receptors: Studies on the Interaction of Estrogen with the UterusQ39977967
GABA receptor binding with 3H (+) bicuculline–methiodide in rat CNSQ40068234
.gamma.-Aminobutyric acid agonists, antagonists, and uptake inhibitors. Design and therapeutic aspectsQ40085780
Neurotransmitter modulation of steroid action in target cells that mediate reproduction and reproductive behaviorQ40086030
Pindolol-a beta-adrenoceptor blocking drug with partial agonist activity: clinical pharmacological considerationsQ40087513
Pindolol: A Review of Its Pharmacology, Pharmacokinetics, Clinical Uses, and Adverse EffectsQ40090048
Disease-induced changes in the plasma binding of basic drugsQ40098103
Inhibitors of the GABA uptake systemsQ40121757
Multiple opiate receptors in peripheral tissue preparationsQ40125919
Binding of?-adrenoceptor blocking drugs to human serum albumin, to ?1-acid glycoprotein and to human serumQ72532282
Some β-Adrenoceptor Functions of Therapeutic InterestQ72536121
Beta-receptor agonists in pregnancy: long term effects in preterm childrenQ72536125
GABA--an inhibitory neurotransmitter that is involved in cardiovascular controlQ72538091
Serotonergic component of neuroleptic receptorsQ48203921
Benzodiazepine receptor: demonstration in the central nervous systemQ48250292
Influence of gender and castration on liver and CNS N-demethylation of morphine in ratsQ48327678
C fragment of lipotropin has a high affinity for brain opiate receptorsQ48392026
Propranolol inhibits rat brain monoamine oxidaseQ48425145
Plasma tryptophan and 5-HT metabolism in the CNS of the newborn rat.Q48534984
Location of the site of the tranquillizing action of diazepam by intralimbic applicationQ48640984
Localizing 3H-GABA in Nerve Terminals of Rat Cerebral Cortex by Electron Microscopic AutoradiographyQ48846486
Brain levels of tofizopam in the rat and relationship with benzodiazepine receptorsQ48880653
Bicuculline and Central GABA ReceptorsQ48882915
Isolation of a GABA receptor from bovine brain using a benzodiazepine affinity columnQ48886991
[125I]-HEAT:fifty percent of the ligand can bind to the alpha1-adrenoceptors with extremely high affinity.Q48892978
Opiate receptor binding sites in human brainQ48895431
Diethylstilbestrol regulates the number of α- and β-adrenergic binding sites in incubated hypothalamus and amygdalaQ48895452
The nature of opiate receptors in toad brainQ48895886
Multiple opiate binding sites in human brain regions: Evidence for κ and σ sitesQ48895894
Certain calcium antagonists are potent displacers of [3H]phencyclidine (PCP) binding in rat brainQ48897569
Central Hypotensive Activity of dl- and d-PropranololQ48898299
Changes in populations of cholinergic binding sites in brain after chronic exposure to barbital in ratsQ48910176
Anticonflict effect of the benzodiazepines mediated by a GABAergic mechanism in the amygdalaQ48910623
GABA, bicuculline and central inhibitionQ48911565
Aggressive behavior and benzodiazepine receptor changes in isolated male miceQ48918451
Tofizopam modulates the affinity of benzodiazepine receptors in the rat brainQ48920183
Stereospecific binding of 3H-phencyclidine in brain membranesQ48932317
Effects of caffeine and theophylline on adenosine and benzodiazepine receptors in human brainQ48942844
Beta-carboline binding indicates the presence of benzodiazepine receptor subclasses in the bovine central nervous systemQ48951400
Enhancement of delta- but not mu-opiate agonist binding by calcium.Q48951417
Effects of propranolol and a number of its analogues on sodium channelsQ48951494
Nanomolar concentrations of propranolol inhibit GABA-stimulated benzodiazepine binding to rat cerebral cortexQ48954847
Physicochemical Characterization of Detergent-Solubilized gamma-Aminobutyric Acid and Benzodiazepine Receptor Proteins from Bovine BrainQ48962321
The Binding of the GAB A Agonist [3H]THIP to Rat Brain Synaptic MembranesQ48962755
The influence of sex hormones on antidepressant-induced alterations in neurotransmitter receptor binding.Q48974726
Effect of acute and chronic phenobarbital treatment on GABA and other amino acids contents in seven regions of the rat brainQ49014701
Stereospecificity of the in vitro and in vivo blockade of β-receptors by FM 24, a slowly reversible ligandQ49133197
Benzodiazepines: towards more logical use.Q49133718
Kinetics and clinical effects of flurazepam in young and elderly noninsomniacsQ49161512
Metabolic consequences of atenolol and propranolol in treatment of essential hypertensionQ50275473
Tranquillizing effects of propranolol demonstrated in rats.Q51324894
Stereoselective binding of 4,5-dihydrodiazepam to human serum albumin.Q51853269
Ketamine inhibition of ligand binding to cholinergic receptors and ion channels.Q51862250
Scopolamine-induced locomotor stimulation in mice: effect of diazepam and a benzodiazepine antagonist.Q51864336
Dual Action of Pentobarbitone on GABA Binding: Role of Binding Site IntegrityQ51865235
Relationship between alpha 1-acid glycoprotein and lidocaine disposition in myocardial infarction.Q51866437
Studies on the antihypertensive action of the optical isomers of propranolol in manQ68544174
Inhibition of insulin secretion by aryl-substituted secondary aminoethanolsQ68596988
Interaction of acetylcholine with different cholinergic nerve receptorsQ68603612
Beta-adrenergic blocking agents. 3. The optical isomers of pronethalol, propranolol, and several related compoundsQ68729783
Beta-adrenergic blocking agents. 10. (3-amino-2-hydroxypropoxy)anilidesQ68754781
Configuration and Conformation of Bicuculline, a GABA AntagonistQ69028342
Studies on the optical enantiomorphs of warfarin in manQ69355706
The effect of d(+)- and 1(-)-practolol on ouabain-induced arrhythmiaQ69411595
The Effect in Man of (+)-Propranolol and Racemic Propranolol on Renin Secretion Stimulated by Orthostatic StressQ69494552
Sclerosing peritonitis, an unusual reaction to a beta-adrenergic-blocking drug (practolol)Q70028270
Beta-adrenergic receptor: stereospecific interaction of iodinated beta-blocking agent with high affinity siteQ70053461
The effect of the dextro isomer of propranolol on sinus rate and cardiac arrhythmiasQ70098081
Transfer of propranolol and sotalol across the human placenta. Their effect on maternal and fetal plasma renin activityQ70243832
[The EEG of patients with acute manic psychoses before, during and after treatment with high doses of d-propranolol and dl-propranolol (author's transl)]Q70260523
Propranolol effects on autonomic function in hypertensive menQ70397264
Stereoselective disposition and glucuronidation of propranolol in humansQ70406047
Cardiac safety of acute beta blockade: intrinsic sympathomimetic activity is superior to beta-1 selectivityQ70419742
Ticrynafen-racemic warfarin interaction: hepatotoxic or stereoselective?Q70425480
Dependence of rate constants of the glucocorticoid hormone-receptor interaction on steroid structureQ70433526
Effects of cancer and its treatments on plasma concentration of alpha 1-acid glycoprotein and propranolol bindingQ70476807
Rat lung cholinergic receptor: characterization and regulation by corticosteroidsQ70482455
Atenolol vs. propranolol in essential tremor. A controlled, quantitative studyQ70532030
Phencyclidine, lysergic acid diethylamide, and mescaline: cerebral artery spasms and hallucinogenic activityQ70662687
Withdrawal from chronic treatment with metergoline, dl-propranolol and amitriptyline enhances serotonin receptor mediated behaviour in the ratQ70677316
Systemic and forearm haemodynamic and metabolic effects of racemic propranolol or D-propranolol in healthy subjectsQ70823837
Propranolol, alprenolol and oxprenolol metabolism in the dog. Identification of N-methylated metabolitesQ70901252
Stereoselective interaction of trimethoprim-sulfamethoxazole with the separated enantiomorphs of racemic warfarin in manQ71128161
High-affinity uptake of (RS)-nipecotic acid in astrocytes cultured from mouse brain. Comparison with GABA transportQ71144478
Soluble benzodiazepine receptors: GABAergic regulationQ71218575
Kinetics of R andS warfarin enantiomersQ71236832
D-propranolol and DL-propranolol both decrease conversion of L-thyroxine to L-triiodothyronineQ71291227
Stationary ultrafiltration: a radio-tracer technique for studying stereoselective binding of racemic ligandsQ71467123
Dynamic interaction between disulfiram and separated enantiomorphs of racemic warfarinQ71509185
Resolution by affinity chromatography: stereoselective binding of racemic oxazepam esters to human serum albuminQ71767203
Stereoselective binding of a 2,3-benzodiazepine to human serum albumin. Effect of conformation on tofizopam bindingQ71819508
Paradoxical nature of estrogen agonist and antagonist binding in rat liverQ71844948
Clinical experience of terbutaline in preterm laborQ72050942
The effect of a benzodiazepine, flurazepam, on the response of in vitro skeletal muscle preparations to muscle relaxants: are purines or their receptors involved?Q72115572
.beta.-Adrenergic blocking agents. II. Propranolol and related 3-amino-1-naphthoxy-2-propanolsQ72148178
The effect of various drugs on the binding of warfarin-14C to human albuminQ72296181
Antagonism by propranolol of isolation-induced aggression in mice: correlation with 5-hydroxytryptamine receptor blockadeQ72429427
Increase in 3H-flunitrazepam binding in vitro and in vivo to rat brain benzodiazepine receptors by tofizopam, a 3,4-benzodiazepineQ72465280
Kappa opiate binding sites in human placentaQ72497427
Quantitation of Beta Adrenergic Receptors in Rat Liver: Confounding Effect of Displaceable But Nonstereospecific Antagonist BindingQ72521776
The binding characteristics of some adrenergic beta-receptor antagonists to human serum proteinsQ72525316
P433issue3
P407language of work or nameEnglishQ1860
P921main subjectpharmacologyQ128406
chiralityQ214514
molecular medicineQ3523816
P304page(s)359-413
P577publication date1984-07-01
P1433published inMedicinal Research ReviewsQ2436033
P1476titleOn chiral drug action
P478volume4