Palladium-catalyzed difluoromethylation of heteroaryl chlorides, bromides and iodides.

scientific article published on 24 April 2017

Palladium-catalyzed difluoromethylation of heteroaryl chlorides, bromides and iodides. is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1039/C7SC00691H
P932PMC publication ID5603793
P698PubMed publication ID28959407

P50authorQilong ShenQ88474774
P2093author name stringJiang Wu
Yang Gu
Changhui Lu
Yucheng Gu
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Unexpected H2O-induced Ar-X activation with trifluoromethylpalladium(II) arylsQ83085930
A new method for aromatic difluoromethylation: copper-catalyzed cross-coupling and decarboxylation sequence from aryl iodidesQ85006215
Copper- and iron-catalyzed decarboxylative tri- and difluoromethylation of α,β-unsaturated carboxylic acids with CF3SO2Na and (CF2HSO2)2Zn via a radical processQ85886898
Cooperative dual palladium/silver catalyst for direct difluoromethylation of aryl bromides and iodidesQ85924093
Sandmeyer difluoromethylation of (hetero-)arenediazonium saltsQ85929835
Pd-catalyzed difluoromethylation of vinyl bromides, triflates, tosylates, and nonaflatesQ86890598
Direct Difluoromethylation of Aryl Halides via Base Metal Catalysis at Room TemperatureQ87306458
Visible light-mediated C-H difluoromethylation of electron-rich heteroarenesQ87846565
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Analysis of the structural diversity, substitution patterns, and frequency of nitrogen heterocycles among U.S. FDA approved pharmaceuticalsQ38254225
Pd-catalyzed α-arylation of α,α-difluoroketones with aryl bromides and chlorides. A route to difluoromethylarenesQ38736425
Copper-mediated difluoromethylation of aryl and vinyl iodidesQ42216204
Practical and innate carbon-hydrogen functionalization of heterocyclesQ42403853
Visible light-promoted metal-free C-H activation: diarylketone-catalyzed selective benzylic mono- and difluorinationQ42773523
A designed P1 cysteine mimetic for covalent and non-covalent inhibitors of HCV NS3 protease.Q43036547
Selective difluoromethylation and monofluoromethylation reactionsQ43213764
Concise synthesis of acyl migration-blocked 1,1-difluorinated analogues of lysophosphatidic acidQ44158213
Copper-mediated difluoromethylation of (hetero)aryl iodides and β-styryl halides with tributyl(difluoromethyl)stannaneQ44779644
Copper-Catalyzed Difluoromethylation of Aryl Iodides with (Difluoromethyl)zinc Reagent.Q51239539
Palladium-Catalyzed Negishi Cross-Coupling Reaction of Aryl Halides with (Difluoromethyl)zinc Reagent.Q51239594
Visible-light-mediated fluoroalkylation of isocyanides with ethyl bromofluoroacetates: unified synthesis of mono- and difluoromethylated phenanthridine derivatives.Q51733460
P433issue7
P407language of work or nameEnglishQ1860
P304page(s)4848-4852
P577publication date2017-04-24
P1433published inChemical ScienceQ2962267
P1476titlePalladium-catalyzed difluoromethylation of heteroaryl chlorides, bromides and iodides
P478volume8

Reverse relations

cites work (P2860)
Q52598206Diastereoselective [3 + 2] cycloaddition of 3-ylideneoxindoles with in situ generated CF2HCHN2: syntheses of CF2H-containing spirooxindoles.
Q48295974Difluoroacetic Acid as a New Reagent for Direct C-H Difluoromethylation of Heteroaromatic Compounds
Q90686384Metallaphotoredox Difluoromethylation of Aryl Bromides
Q92062591Sustainable Knowledge-Driven Approaches in Transition-Metal-Catalyzed Transformations

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