Modulation of constitutive activity and signaling bias of the ghrelin receptor by conformational constraint in the second extracellular loop

scientific article published on 30 July 2012

Modulation of constitutive activity and signaling bias of the ghrelin receptor by conformational constraint in the second extracellular loop is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1074/JBC.M112.383240
P932PMC publication ID3460450
P698PubMed publication ID22846991
P5875ResearchGate publication ID230588693

P50authorThue W SchwartzQ51291438
Birgitte HolstQ57178867
Jacek MokrosinskiQ38804492
P2093author name stringThomas M Frimurer
Bjørn Sivertsen
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P433issue40
P407language of work or nameEnglishQ1860
P921main subjectbiasQ742736
P1104number of pages15
P304page(s)33488-33502
P577publication date2012-07-30
P1433published inJournal of Biological ChemistryQ867727
P1476titleModulation of constitutive activity and signaling bias of the ghrelin receptor by conformational constraint in the second extracellular loop
P478volume287

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cites work (P2860)
Q96132105Advances in therapeutic peptides targeting G protein-coupled receptors
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Q34580340G Protein and β-arrestin signaling bias at the ghrelin receptor
Q36665235G Protein-coupled Receptor Biased Agonism
Q38113559GHS-R1a constitutive activity and its physiological relevance
Q35062647Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex
Q39145769Structural basis for constitutive activity and agonist-induced activation of the enteroendocrine fat sensor GPR119.
Q90331866The C-terminal Phosphorylation Sites of eel Follicle-Stimulating Hormone Receptor are Important Role in the Signal Transduction
Q24568026The growth hormone secretagogue receptor: its intracellular signaling and regulation
Q57292162Translating biased signaling in the ghrelin receptor system into differential in vivo functions

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