Probing of NMDA channels with fast blockers

scientific article published on December 1999

Probing of NMDA channels with fast blockers is …
instance of (P31):
scholarly articleQ13442814

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P698PubMed publication ID10594045

P2093author name stringKhodorov BI
Sobolevsky AI
Koshelev SG
P2860cites workMechanism of memantine block of NMDA-activated channels in rat retinal ganglion cells: uncompetitive antagonismQ24530210
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Dimensions of the narrow portion of a recombinant NMDA receptor channelQ34128656
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Kinetic analysis of pancuronium interaction with sodium channels in squid axon membranesQ36407698
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Alternative splicing generates functionally distinct N-methyl-D-aspartate receptorsQ37199611
Two blocking sites of amino-adamantane derivatives in open N-methyl-D-aspartate channelsQ40116843
N-methyl-D-aspartic acid receptor structure and functionQ40674725
Local anaesthetics transiently block currents through single acetylcholine-receptor channelsQ40676934
Multiple sites of action of neomycin, Mg2+ and spermine on the NMDA receptors of rat hippocampal CA1 pyramidal neuronesQ41010615
Calcium-dependent inactivation of recombinant N-methyl-D-aspartate receptors is NR2 subunit specific.Q41148644
Actions of ketamine, phencyclidine and MK-801 on NMDA receptor currents in cultured mouse hippocampal neuronesQ41152868
Trapping of an open-channel blocker at the frog neuromuscular acetylcholine channelQ41158135
Structural basis for explaining open-channel blockade of the NMDA receptor.Q41664696
Voltage-gated ion channels and electrical excitabilityQ41737177
Interaction of Tetraethylammonium Ion Derivatives with the Potassium Channels of Giant AxonsQ41761074
The Inhibition of Sodium Currents in Myelinated Nerve by Quaternary Derivatives of LidocaineQ41920650
Simulation of Na channel inactivation by thiazine dyesQ41934311
A kinetic analysis of the modulation of N-methyl-D-aspartic acid receptors by glycine in mouse cultured hippocampal neuronesQ42084783
Voltage-dependent interaction of open-channel blocking molecules with gating of NMDA receptors in rat cortical neuronsQ42637358
Both open and closed NMDA receptor channels desensitizeQ42673990
N-terminal domains in the NR2 subunit control desensitization of NMDA receptorsQ48039856
Tetrahydroaminoacridine blocks and prolongs NMDA receptor-mediated responses in a voltage-dependent mannerQ48173255
Interactions between the glycine and glutamate binding sites of the NMDA receptor.Q48328504
Inactivation of NMDA channels in cultured hippocampal neurons by intracellular calciumQ48344157
Interaction of memantine and amantadine with agonist-unbound NMDA-receptor channels in acutely isolated rat hippocampal neuronsQ48399177
Evidence for a tetrameric structure of recombinant NMDA receptors.Q48487196
Glycine-independent NMDA receptor desensitization: localization of structural determinantsQ48517849
NMDA channel behavior depends on agonist affinityQ48543141
High probability opening of NMDA receptor channels by L-glutamateQ48546296
Vibrodissociation of sliced mammalian nervous tissueQ48700946
NMDAR channel segments forming the extracellular vestibule inferred from the accessibility of substituted cysteinesQ48921111
Concentration-jump experiments with NMDA antagonists in mouse cultured hippocampal neuronsQ48965413
Structure of the NMDA receptor channel M2 segment inferred from the accessibility of substituted cysteines.Q50760890
Synaptic NMDA receptor channels have a low open probability.Q54012474
Regulation of NMDA receptor desensitization in mouse hippocampal neurons by glycine.Q54112154
Trapping of glutamate and glycine during open channel block of rat hippocampal neuron NMDA receptors by 9‐aminoacridineQ54179283
Glycine-insensitive desensitization of NMDA responses in cultured mouse embryonic neuronsQ68461323
Dynamics of the actions of tetrahydro-9-aminoacridine and 9-aminoacridine on glutamatergic currents: concentration-jump studies in cultured rat hippocampal neuronsQ71608640
Novel adamantane derivatives act as blockers of open ligand-gated channels and as anticonvulsantsQ71684723
Hydrophobic interactions of n-alkyl diamines with the N-methyl-D-aspartate receptor: voltage-dependent and -independent blocking sitesQ72759229
Trapping channel block of NMDA-activated responses by amantadine and memantineQ73271990
Binding sites for permeant ions in the channel of NMDA receptors and their effects on channel blockQ77299364
Two-component blocking kinetics of open NMDA channels by organic cationsQ77796382
P433issue24
P407language of work or nameEnglishQ1860
P304page(s)10611-10626
P577publication date1999-12-01
P1433published inJournal of NeuroscienceQ1709864
P1476titleProbing of NMDA channels with fast blockers
P478volume19

Reverse relations

cites work (P2860)
Q41981072Actions of bupivacaine, a widely used local anesthetic, on NMDA receptor responses
Q43953372Blocker studies of the functional architecture of the NMDA receptor channel
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Q88789953Effects of Mg2+ on recovery of NMDA receptors from inhibition by memantine and ketamine reveal properties of a second site
Q28366918Free intracellular Mg(2+) concentration and inhibition of NMDA responses in cultured rat neurons
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Q64937337Influences: Russian training.
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Q34059951Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists
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Q39267480Specific mechanism of use-dependent channel block of calcium-permeable AMPA receptors provides activity-dependent inhibition of glutamatergic neurotransmission
Q34179425Staggering of subunits in NMDAR channels.
Q90425146Structure, function, and allosteric modulation of NMDA receptors
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Q85844030The differential contribution of GluN1 and GluN2 to the gating operation of the NMDA receptor channel
Q53907480The trapping block of NMDA receptor channels in acutely isolated rat hippocampal neurones.

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