2-(3,5-Dimethylphenyl)tryptamine derivatives that bind to the GnRH receptor

scientific article published in April 2001

2-(3,5-Dimethylphenyl)tryptamine derivatives that bind to the GnRH receptor is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0960-894X(01)00134-2
P698PubMed publication ID11327593
P5875ResearchGate publication ID12007923

P2093author name stringLin P
Smith RG
Fisher MH
Wyvratt MJ
Marino D
Cheng K
Goulet MT
Lo JL
Yang YT
P2860cites workDiscovery of a novel, potent, and orally active nonpeptide antagonist of the human luteinizing hormone-releasing hormone (LHRH) receptorQ42538865
A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptorQ43574126
Heterocyclic derivatives of 2-(3,5-dimethylphenyl)tryptamine as GnRH receptor antagonistsQ43591324
Gonadotropin-releasing hormone: one polypeptide regulates secretion of luteinizing and follicle-stimulating hormonesQ47743244
Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequenceQ47747051
A Locus of the Gonadotropin-releasing Hormone Receptor That Differentiates Agonist and Antagonist Binding SitesQ58853853
Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonistQ73022495
Investigation of the 4-O-alkylamine substituent of non-peptide quinolone GnRH receptor antagonistsQ73022498
Initial structure-activity relationship of a novel class of nonpeptidyl GnRH receptor antagonists: 2-arylindolesQ73566599
SAR studies of novel 5-substituted 2-arylindoles as nonpeptidyl GnRH receptor antagonistsQ73566603
Potent antagonists of gonadotropin releasing hormone receptors derived from quinolone-6-carboxamidesQ73613776
Quinolones as gonadotropin releasing hormone (GnRH) antagonists: simultaneous optimization of the C(3)-aryl and C(6)-substituentsQ74151432
P433issue8
P407language of work or nameEnglishQ1860
P304page(s)1073-1076
P577publication date2001-04-01
P1433published inBioorganic & Medicinal Chemistry LettersQ2709483
P1476title2-(3,5-Dimethylphenyl)tryptamine derivatives that bind to the GnRH receptor
P478volume11

Reverse relations

cites work (P2860)
Q438916512-Arylindoles as gonadotropin releasing hormone (GnRH) antagonists: optimization of the tryptamine side chain
Q40691847A novel synthesis of 7-aryl-8-fluoro-pyrrolo[1,2-a]pyrimid-4-ones as potent, stable GnRH receptor antagonists
Q43591324Heterocyclic derivatives of 2-(3,5-dimethylphenyl)tryptamine as GnRH receptor antagonists
Q43868998Initial structure-activity relationship studies of a novel series of pyrrolo[1,2-a]pyrimid-7-ones as GnRH receptor antagonists
Q43733815Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity
Q43653091Potent nonpeptide GnRH receptor antagonists derived from substituted indole-5-carboxamides and -acetamides bearing a pyridine side-chain terminus
Q47323557Recent Development of Non-Peptide GnRH Antagonists.
Q43653090Substituted indole-5-carboxamides and -acetamides as potent nonpeptide GnRH receptor antagonists
Q44593722Synthesis and structure–Activity relationships of thieno[2,3- d ]pyrimidine-2,4-dione derivatives as potent GnRH receptor antagonists

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